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3-cyclopropyl-5-[2-(1H-imidazol-4-yl)-1-(1H-pyrrol-1-yl)ethyl]-1H-1,2,4-triazole
4-chloro-N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-propanamidobenzamide
N,4-dimethyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-4-yl)methyl]-1,2,5-oxadiazole-3-carboxamide
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-[2-(cyclohex-1-en-1-yl)ethyl]propanamide
5-ethyl-5-(1-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperidin-4-yl)imidazolidine-2,4-dione
1-{2-methyl-1-[2-(3-methyl-1H-1,2,4-triazol-5-yl)pyrrolidin-1-yl]propan-2-yl}piperidine
4,5-dimethyl 1-[(3S,5S)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}-1-(thiophen-3-ylmethyl)pyrrolidin-3-yl]-1H-1,2,3-triazole-4,5-dicarboxylate
(3R,4R)-1-[1-(4-methoxyphenyl)piperidin-4-yl]-4-(4-methylpiperazin-1-yl)piperidin-3-ol
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-1H-pyrazole-4-carboxamide
{1-[4-(ethylamino)-5-methylthieno[2,3-d]pyrimidine-6-carbonyl]piperidin-2-yl}methanol
3-[(3R,7S,8aS)-3-(2-methylpropyl)-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(naphthalen-1-yl)urea
N-[(2R)-3,4-dihydro-2H-1-benzopyran-2-ylmethyl]-5-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-1,5,6-trimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
1-[(2-chloro-6-fluorophenyl)methyl]-4-[2-(pyrrolidine-1-carbonyl)phenoxy]piperidine
(2R,3R,6R)-3-(3-methoxyphenyl)-5-(6-methylpyridine-2-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
2-(4-{[3-(4-fluorophenyl)-1-(4-methylphenyl)-1H-pyrazol-4-yl]methyl}piperazin-1-yl)pyrimidine
1-[(2Z)-2-fluoro-3-phenylprop-2-enoyl]-4-[(2-fluorophenyl)methyl]-1,4-diazepan-5-one
(3aR,6aS)-5-(3-ethyl-1-methyl-1H-pyrazole-5-carbonyl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-[3-(morpholin-4-yl)propyl]-5-(thiomorpholine-4-carbonyl)piperidin-2-one
1-[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-ol
N-ethyl-3-(piperidine-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N,1-dimethyl-N-[2-(pyridin-2-yl)ethyl]-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(4-{[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]methyl}thiophen-2-yl)ethan-1-one
2-(4-{[4-(pyrrolidin-1-ylmethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)pyridine
methyl[(5-methyl-1,2,4-oxadiazol-3-yl)methyl]{[5-(thiophen-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]methyl}amine
1-(2,6-dimethylpyridin-4-yl)-4-(pyrrolidin-3-ylmethyl)piperazine
6-[4-(2-ethyl-4-methyl-1,3-oxazole-5-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
N-({2-methoxy-5-oxo-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)cyclopropanecarboxamide
2-(2,3-dihydro-1H-inden-1-yl)-N-propyl-N-(pyridin-3-ylmethyl)acetamide
N-[2-(4-methoxyphenyl)ethyl]-3-methyl-N-[(1-methylpiperidin-4-yl)methyl]thiophene-2-carboxamide
(5-{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}-1-methyl-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl)methanol
(4aS,7aR)-1-[4-(1H-imidazol-1-yl)butanoyl]-4-(2-methylpropanoyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[1-(3-cyanopyridin-2-yl)piperidin-4-yl]-5-oxopyrrolidine-3-carboxylic acid
3-(1H-indol-5-yl)-1-[1-(methoxymethyl)cyclopentyl]urea
3-methyl-7-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-(3,4-dimethylphenyl)-5-(1H-imidazol-1-ylmethyl)-3-(propan-2-yl)-1H-1,2,4-triazole
N-(2,3-dihydro-1H-inden-2-yl)-1-(9H-purin-6-yl)piperidin-4-amine
N-(butan-2-yl)-N-[(4-chlorophenyl)methyl]-2-(4-oxocyclohexyl)acetamide
3-(2H-1,3-benzodioxol-5-yl)-1-(4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)propan-1-one
(3aS,6aS)-2-(dimethylcarbamoyl)-5-{[5-(propan-2-yl)-1,2-oxazol-3-yl]methyl}-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-[(diethylamino)methyl]-5-ethyl-N-[(4-oxo-3,4-dihydroquinazolin-2-yl)methyl]furan-2-carboxamide
N-cyclopropyl-6-[4-(piperidine-1-carbonyl)piperidin-1-yl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
methyl({[5-methyl-2-(3-methylphenyl)-1,3-oxazol-4-yl]methyl})[(3-methylthiophen-2-yl)methyl]amine
N-{1-[(3-chlorophenyl)methyl]-1H-pyrazol-5-yl}-3,5-dimethyl-4,5-dihydro-1,2-oxazole-5-carboxamide
2-(methylsulfanyl)-6-oxo-N-(pentan-3-yl)-N-(2-phenylethyl)-1,6-dihydropyrimidine-5-carboxamide
methyl 1-[(3R,5S)-1-{[3-(benzyloxy)phenyl]methyl}-5-[4-(4-fluorophenyl)piperazine-1-carbonyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
3-[2-(2H-1,3-benzodioxol-5-ylmethyl)-5-oxopyrrolidin-2-yl]-N-{2-[(1R,5S)-6,6-dimethylbicyclo[3.1.1]hept-2-en-2-yl]ethyl}propanamide
1-(4-acetyl-4-phenylpiperidin-1-yl)-2-(5-acetylthiophen-3-yl)ethan-1-one
3-{[2-(4-chlorophenyl)morpholin-4-yl]methyl}-N-methyl-1,2,4-oxadiazole-5-carboxamide
3-{2-[(5-chloro-2-methoxyphenyl)carbamoyl]ethyl}-N-(2-methoxyethyl)piperidine-1-carboxamide