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6-(4-fluorophenyl)-N-(2-methoxyethyl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
(3R,4S)-N,N-dimethyl-1-[4-methyl-2-(piperidin-1-yl)pyrimidine-5-carbonyl]-4-propylpyrrolidin-3-amine
1-(pyridin-2-yl)-N-[1-(pyridin-2-ylmethyl)piperidin-4-yl]-4,5,6,7-tetrahydro-1H-indazol-4-amine
3-methyl-8-{6-methyl-4-oxa-2,5-diazatricyclo[7.3.0.03,7]dodeca-1(9),2,5,7-tetraene-8-carbonyl}-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-{1-[(3-methoxyphenyl)methyl]piperidin-3-yl}-5-phenyl-1,2-oxazole-3-carboxamide
2-(cyclopropylmethyl)-8-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-2,8-diazaspiro[5.5]undecan-3-one
3,5-dimethyl-2-{[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]methyl}-1,4-dihydropyridin-4-one
N-{[(3S,4S)-3-hydroxy-1-[2-methyl-2-(1H-pyrrol-1-yl)propanoyl]piperidin-4-yl]methyl}furan-2-carboxamide
N-(1-methoxy-2-methylpropan-2-yl)-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N-methyl-2-(phenoxymethyl)-1,3-oxazole-4-carboxamide
N-(2-chloropyridin-3-yl)-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
7-[(dimethyl-1,2-oxazol-4-yl)methyl]-2-oxa-7-azaspiro[4.5]decane
N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-5-[3-(2-methoxyethyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
2,6-difluoro-3-methoxy-N-(2-methoxyethyl)-N-[(1-methyl-1H-pyrazol-4-yl)methyl]benzamide
methyl 2-oxo-1-(prop-2-en-1-yloxy)-8-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,8-diazaspiro[4.5]decane-4-carboxylate
2-[1-(propan-2-yl)piperidin-4-yl]-N-[(4-sulfamoylphenyl)methyl]acetamide
3-cyclopropyl-5-[4-(methoxymethyl)-5-methyl-1,2-oxazol-3-yl]-1H-1,2,4-triazole
(2R,6R)-4-(3-ethyl-4-methyl-1H-pyrazole-5-carbonyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
2-[4-(5-phenyl-1,2,4-oxadiazol-3-yl)-1-(2-phenylethyl)piperazin-2-yl]ethan-1-ol
4-{4-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]phenyl}-2-methylbutan-2-ol
3-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-3-ethyl-1-(2-methyl-1-benzofuran-7-yl)urea
6-(2-fluoro-5-methoxyphenyl)-2H-1,3-benzodioxole-5-carboxamide
6-(hydroxymethyl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}pyridine-2-carboxamide
1-(4-chlorophenyl)-N-{[1-(oxane-4-carbonyl)piperidin-3-yl]methyl}cyclopropane-1-carboxamide
[3-(2-methoxyethyl)-1-(pyrimidin-2-ylmethyl)piperidin-3-yl]methanol
1-[2-(2-chloro-4-fluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-4-methylpiperazine
N-{[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]methyl}-N-methyl-5-oxo-1-(propan-2-yl)pyrrolidine-3-carboxamide
4-(5-{2-phenyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl}-1H-pyrazol-3-yl)pyridine
3-[4-(3-chlorophenyl)piperazine-1-carbonyl]-2-ethyl-1-[(4-methoxyphenyl)methyl]-6-methyl-1,4-dihydropyridin-4-one
(1R,5R)-6-(cyclopropylmethyl)-3-(2-fluoro-5-methylbenzenesulfonyl)-3,6-diazabicyclo[3.2.2]nonane
2-(3,5-dimethyl-1H-pyrazol-1-yl)-1-{3-[4-(4-fluorophenyl)piperazin-1-yl]piperidin-1-yl}ethan-1-one
N-[(3R,4S)-1-(2-methoxyethyl)-4-propylpyrrolidin-3-yl]-4-methyl-1,2,5-oxadiazole-3-carboxamide
N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzamide
2-{1-[2-(thiophen-2-yl)-1,3-thiazole-4-carbonyl]azetidin-3-yl}pyridine
N-{3-oxo-3-[4-(2-phenoxyethyl)piperazin-1-yl]propyl}methanesulfonamide
N-[(3S,4R)-4-ethoxyoxolan-3-yl]-4-{[(3-methylthiophen-2-yl)methyl]amino}benzamide
N-({1-[2-(2-fluorophenyl)ethyl]piperidin-3-yl}methyl)-N,5-dimethyl-1H-indazole-3-carboxamide
1-[2-(4-chlorophenyl)morpholin-4-yl]-2-propoxyethan-1-one
(4S)-4-(methoxymethyl)-3,3-dimethyl-1-[2-(trifluoromethyl)benzoyl]piperidin-4-ol
2-[3-(1-ethyl-1H-imidazol-2-yl)piperidin-1-yl]-6,7-dimethoxyquinazolin-4-amine
6-oxo-N-[(5-phenyl-1,3,4-oxadiazol-2-yl)methyl]-1,4,5,6-tetrahydropyridazine-3-carboxamide
N-({5-acetyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-5-methylpyrazine-2-carboxamide
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N-methyl-2-[3-oxo-1-(propan-2-yl)piperazin-2-yl]acetamide
2-[(5-{[2-(1H-pyrazol-1-ylmethyl)pyrrolidin-1-yl]methyl}furan-2-yl)sulfanyl]pyrimidine
(2S,4R)-4-amino-1-{2-[4-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)phenyl]acetyl}-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[3-(6-hydroxy-2-methylpyrimidin-4-yl)piperidin-1-yl]-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
N-(1H-indol-4-ylmethyl)-1-[(3-methoxyphenyl)methyl]-6-oxopiperidine-3-carboxamide
1-methyl-4-[(1-{[3-(trifluoromethyl)phenyl]methyl}piperidin-3-yl)methyl]piperazine
4-(4-ethyl-1H-pyrazol-5-yl)-1-{[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}piperidine
N-(4-acetylphenyl)-3-(4-phenylpiperazin-1-yl)piperidine-1-carboxamide