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4-[3-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]-1,2-dihydroquinolin-2-one
[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)[(6-methylpyridin-2-yl)methyl]amine
3-[({1-[5-(2-methoxyphenoxymethyl)-1,2-oxazole-3-carbonyl]piperidin-3-yl}oxy)methyl]pyridine
3-(4-phenylbenzoyl)-1-(prop-2-ene-1-sulfonyl)piperidine
4-methyl-6-{6-oxa-9-azaspiro[4.5]decan-9-yl}-5-(prop-2-en-1-yl)pyrimidin-2-amine
3-{[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}-4,5-dimethyl-2,3-dihydro-1,3-oxazol-2-one
(2S)-4-(methylsulfanyl)-2-{[5-(pyridin-4-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}butan-1-ol
6-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-5H-[1,3]thiazolo[3,2-a]pyrimidin-5-one
N-[3-(3-methoxyphenyl)phenyl]-1-(1-methyl-1H-pyrazole-5-carbonyl)piperidine-2-carboxamide
[1-(dimethyl-1,3-thiazol-4-yl)ethyl][(8-methoxyquinolin-2-yl)methyl]methylamine
1-(4-hydroxyphenyl)-N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-oxopyrrolidine-3-carboxamide
7-(cyclopropylmethyl)-2-(1-phenyl-1H-1,2,3-triazole-4-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-(1H-1,3-benzodiazol-1-yl)-1-(2-methoxyacetyl)piperidine-4-carboxylic acid
1-(1-propyl-1H-pyrazole-5-carbonyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
N-{[2-(3,4-difluorophenoxy)pyridin-3-yl]methyl}-2-(methylamino)pyridine-4-carboxamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(2-methoxyethoxy)ethan-1-one
5-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}isoquinoline
1-(2-methoxyacetyl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}piperidine-3-carboxamide
2-hydroxy-5-methyl-N-{[1-(1-methylpiperidin-4-yl)pyrrolidin-3-yl]methyl}benzamide
N,N-dimethyl-1-[1-(pyridine-4-carbonyl)piperidine-4-carbonyl]azepan-4-amine
1-(2-{5-hydroxy-1-oxa-9-azaspiro[5.5]undecan-9-yl}-4-methylpyrimidin-5-yl)ethan-1-one
2-(2-{[3-(4-methylpiperazin-1-yl)pyrrolidin-1-yl]methyl}phenoxy)acetic acid
N-methyl-N-[2-(1-methyl-1H-pyrazol-4-yl)ethyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-1-(difluoromethyl)-1H-pyrazole
3-({3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)pyridin-2-amine
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-2-oxo-1-[(1r,4r)-4-hydroxycyclohexyl]-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
(3S,4R)-1-(3,4-diethoxybenzoyl)-4-methylpiperidine-3,4-diol
1-[1-(2,3-dihydroxybenzoyl)piperidin-3-yl]-3-phenylpropan-1-one
4-methyl-N-[(4-phenyloxan-4-yl)methyl]pyrimidin-2-amine
3-cyclopropyl-N-[(2-{methyl[2-(pyridin-2-yl)ethyl]amino}pyridin-3-yl)methyl]-1,2-oxazole-5-carboxamide
(2S,4S)-1-cyclopentyl-N-ethyl-4-[2-(phenylsulfanyl)acetamido]pyrrolidine-2-carboxamide
3-benzyl-8-(butan-2-yl)-1-methyl-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-(4-butylphenyl)-3-[2-(5-methyl-4H-1,2,4-triazol-3-yl)ethyl]urea
3-({6-cyclopentyl-1-methyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}amino)-3-(4-methylphenyl)propan-1-ol
3-[1-(1-methyl-1H-pyrazol-4-yl)propyl]-1-[3-(4-methylpiperazine-1-carbonyl)phenyl]urea
4-[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl]-N-cyclopropylpiperazine-2-carboxamide
3-benzoyl-1-(1-phenylcyclopropanecarbonyl)piperidine
5-{[benzyl(methyl)amino]methyl}-N-[1-(pyridin-3-yl)propyl]-1,2-oxazole-3-carboxamide
1-[1-(3-cyano-4,6-dimethylpyridin-2-yl)piperidin-4-yl]-N-(2-methoxyethyl)piperidine-3-carboxamide
2-[3-oxo-9-(2-phenylacetyl)-2,9-diazaspiro[5.5]undecan-2-yl]propanoic acid
(1S,5R)-6-(2-chloro-6-fluorobenzoyl)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-methyl-7-[(5-propylfuran-2-yl)methyl]-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
3-[2-amino-4-(3-acetamidopyrrolidin-1-yl)-6-methylpyrimidin-5-yl]propanoic acid
2-[4-(2-amino-6-methoxypyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(3-methyl-1-propyl-1H-pyrazol-5-yl)acetamide
N-[3-fluoro-4-(trifluoromethyl)phenyl]-2-(2-methoxyethyl)piperidine-1-carboxamide
4-[(4-ethyl-2-methyl-1,3-thiazol-5-yl)methyl]-2H,3H,4H-pyrido[3,2-b][1,4]oxazin-3-one
1,9-dimethyl-4-{7-methylthieno[3,2-d]pyrimidin-4-yl}-1,4,9-triazaspiro[5.6]dodecan-10-one
3-methyl-N-[(3R,5S)-1-[(5-methylfuran-2-yl)methyl]-5-[(propan-2-yl)carbamoyl]pyrrolidin-3-yl]-1,2-oxazole-5-carboxamide
2-amino-8-[5-(1-methyl-1H-1,3-benzodiazol-2-yl)furan-2-yl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
1-{2-[(1R,5S)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-2-oxoethyl}-2,3-dihydro-1H-1,3-benzodiazol-2-one