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N-(2-methylpropyl)-2-(3-oxo-1-{[3-(trifluoromethyl)phenyl]methyl}piperazin-2-yl)acetamide
4-[(1S,2S)-2-hydroxycyclohexyl]-N-(4-methoxy-2-methylphenyl)piperazine-1-carboxamide
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-5-(methoxymethyl)pyrazolo[1,5-a]pyrimidin-7-amine
[(2-chloro-4-fluorophenyl)methyl][(1-cyclopentylpiperidin-4-yl)methyl](pyridin-3-ylmethyl)amine
N-cyclopropyl-5-methyl-4-{[2-(pyridin-2-yl)ethyl]amino}thieno[2,3-d]pyrimidine-6-carboxamide
N-phenyl-3-(quinoxalin-5-ylformamido)propanamide
1-{4-[(4-methyl-1H-pyrazol-1-yl)methyl]piperidin-1-yl}-2-(morpholin-3-yl)ethan-1-one
5-(4-fluorophenyl)-N-methyl-N-[4-(morpholin-4-yl)butyl]-1,2,4-triazin-3-amine
(3aR,6aR)-2-(2,3-dihydro-1,4-benzodioxin-6-ylmethyl)-5-(pyrimidin-2-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(3-{[(4-{3-[cyclohexyl(methyl)amino]-2-hydroxypropoxy}-3-methoxyphenyl)methyl]amino}propyl)pyrrolidin-2-one
N-[(6-hydroxypyrimidin-4-yl)methyl]pyrazolo[1,5-a]pyridine-7-carboxamide
N-[2-(4,6-dihydroxypyrimidin-2-yl)ethyl]-3-(2-methylphenyl)-3-phenylpropanamide
methyl (2S,4R)-1-[(5-chloro-2-hydroxyphenyl)methyl]-4-(2-phenylbenzamido)pyrrolidine-2-carboxylate
N-[(2-ethoxyphenyl)methyl]-2,6-dihydroxy-N-(prop-2-en-1-yl)benzamide
4-benzyl-2-{2-oxo-2-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]ethyl}-1,2-dihydrophthalazin-1-one
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-{imidazo[1,2-a]pyridin-3-ylmethyl}benzamide
[(1-ethyl-1H-pyrazol-4-yl)methyl]({1-[2-(3-fluorophenyl)ethyl]piperidin-4-yl}methyl)methylamine
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-3-{5-oxo-2-[(4-phenylphenyl)methyl]pyrrolidin-2-yl}propanamide
1-(3-fluoropyridin-4-yl)-4-(3-methoxybenzoyl)piperazine
2-[4-(2,3-dihydro-1H-inden-2-yl)-6-hydroxy-1,4-diazepan-1-yl]pyridine-3-carbonitrile
4-(4-chlorophenyl)-1-[4-(ethoxymethyl)piperidin-1-yl]butan-1-one
3-({[1-({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)piperidin-4-yl]oxy}methyl)pyridine
1-ethyl-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]pyrrolidine-2-carboxamide
1-methyl-8-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
3-(furan-2-yl)-N-[(3-methyloxetan-3-yl)methyl]-3-phenylpropanamide
3-(4-fluorophenoxymethyl)-1-(1,3-thiazol-4-ylmethyl)piperidine
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1-[(2-fluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
1-methyl-4-{5-[3-(2-methylphenyl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}piperazine
N-methyl-2-[1-(2-methylpropyl)-3-oxopiperazin-2-yl]-N-(pyrimidin-4-ylmethyl)acetamide
2-(3-ethylphenyl)-2-(4-hydroxy-4-phenylpiperidin-1-yl)acetic acid
2,5-dimethyl-N-(oxolan-2-ylmethyl)-N-(2-phenoxyethyl)-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
1-benzyl-N-ethyl-4-oxo-5-(3-phenylpiperidine-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
N-[(3-chlorophenyl)methyl]-3-(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-4-yl)propanamide
(1S,5R)-6-(4-chloro-1-methyl-1H-pyrazole-3-carbonyl)-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
8-{[4-(1,2-oxazinane-2-carbonyl)-1,3-oxazol-2-yl]methoxy}quinoline
methyl 2-(ethylsulfamoyl)-6-(3-phenylpropyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(5-{2-[4-(1H-imidazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}-1H-1,2,4-triazol-3-yl)pyridine
N-benzyl-N,1-dimethyl-5-{[(3,4,5-trimethoxyphenyl)methyl]amino}-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-[4-(difluoromethoxy)-2-methylphenyl]-3-[1-(3,5-dimethyl-1H-pyrazol-1-yl)propan-2-yl]urea
N3-benzyl-1-(2-methylpropyl)-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3-hydroxy-3-({methyl[2-(pyrrolidin-1-yl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-2-(oxan-2-ylmethoxy)ethan-1-one
1-(2-oxo-2-{4-[1-(pyridin-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethyl)pyrrolidin-2-one
(1,2-oxazol-3-ylmethyl)({[2-(piperidin-1-yl)-2,3-dihydro-1H-inden-2-yl]methyl})amine
1-benzyl-2-methyl-3-[2-(4H-1,2,4-triazol-4-yl)ethyl]-1H-indole
3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]propanamide
5-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidine-1-carbonyl]-2-methoxyphenol
(benzylsulfamoyl)(methyl)[1-(1,2-oxazol-3-yl)ethyl]amine
4-{2-tert-butyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-methoxypyridine-3-carbonitrile
1-[7-(cyclopropylmethyl)-2,7-diazaspiro[4.5]decan-2-yl]-3-methylbut-2-en-1-one