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3-{5-[(furan-2-ylmethyl)carbamoyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanoic acid
N-(1-{1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-4-methoxybenzamide
2-methoxy-1-[1'-(pyridin-4-ylmethyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-5-yl]ethan-1-one
N-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N,1-dimethyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[2-(2,3-difluorophenoxymethyl)-1,3-oxazole-4-carbonyl]-1,2,3,4-tetrahydroisoquinoline
[(3R,4R)-4-[(dimethylamino)methyl]-1-{[3-(3-methoxyphenyl)phenyl]methyl}pyrrolidin-3-yl]methanol
4-[3-(2-methoxyethyl)-1-[3-(trifluoromethyl)phenyl]-1H-1,2,4-triazol-5-yl]azepane
4-(2-methylpropyl)-3-{2-oxo-2-[4-(quinazolin-4-yl)piperazin-1-yl]ethyl}piperazin-2-one
2-[4-(2,1,3-benzothiadiazol-5-ylmethyl)-1-[(5-methylfuran-2-yl)methyl]piperazin-2-yl]ethan-1-ol
(1R,2R,6S,7S)-4-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
9-[2-(2-methoxy-4-methylphenoxy)ethyl]-2-methyl-2,9-diazaspiro[5.5]undecan-3-one
6-(1-{[2-(furan-2-yl)pyrimidin-5-yl]methyl}piperidin-3-yl)-2-methylpyrimidin-4-ol
4-(2-methyl-1H-imidazol-1-yl)-1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidine-4-carboxylic acid
(2R,3R)-3-{[(4-fluorophenyl)methyl](methyl)amino}-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
6-{3-hydroxy-5-[2-(piperidin-2-yl)ethyl]phenyl}pyridine-3-carboxylic acid
N-[(2-ethyl-3-methyl-1H-indol-5-yl)methyl]-2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetamide
N-[(4-ethyl-1,3-thiazol-2-yl)methyl]-6-{[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]amino}pyridine-3-carboxamide
6-methyl-2-({[1-(pyridin-3-yl)propan-2-yl]amino}methyl)quinolin-4-ol
2-{2-chloro-4-[(3-acetamidopiperidin-1-yl)methyl]-6-methoxyphenoxy}acetamide
2-({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(propyl)amino)ethan-1-ol
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-5-cyclobutyl-1,3,4-oxadiazol-2-amine
2-[(2-methylphenyl)sulfanyl]-N-[(1-methylpyrrolidin-3-yl)methyl]acetamide
N-[(2-chlorophenyl)methyl]-6-oxo-1-[3-(2-oxopyrrolidin-1-yl)propyl]piperidine-3-carboxamide
2-methyl-N-{1-[4-methyl-2-(pyridin-4-yl)pyrimidin-5-yl]ethyl}imidazo[1,2-a]pyridine-3-carboxamide
3-{[({1-[2-(4-fluorophenyl)ethyl]piperidin-4-yl}methyl)(methyl)amino]methyl}-6-methyl-4H-chromen-4-one
3-(3-fluorophenyl)-4-[2-(4-fluorophenyl)azetidine-1-carbonyl]-1H-pyrazole
9-ethyl-1-methyl-4-({1-methyl-4-oxo-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-6-yl}methyl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-ethyl-4-[(3-fluoropyridin-2-yl)methyl]-1-(propan-2-yl)piperazine
N-ethyl-2-[2-oxo-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-8-yl]acetamide
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-2-propyl-1,3-thiazole-4-carboxamide
3-{1-[2-(carbamoylamino)acetyl]piperidin-4-yl}-N-(3-methoxyphenyl)propanamide
{[1-benzyl-2-(2-methoxyethanesulfonyl)-1H-imidazol-5-yl]methyl}bis(prop-2-en-1-yl)amine
5-methyl-4-{1-[3-(5-methylfuran-2-yl)butyl]piperidin-4-yl}pyrimidine
5-methyl-N-{2-[5-(oxolan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}-1,3,4-oxadiazol-2-amine
3-{[4-(pyrrolidin-3-yl)piperidin-1-yl]methyl}pyridine
2-benzyl-N-[1-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-N-methyl-1,3-benzoxazole-5-carboxamide
1-ethyl-3-methyl-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}-1H-pyrazole-4-sulfonamide
4-[(4aS,8aS)-4a-hydroxy-decahydroisoquinolin-2-yl]-N-cyclooctyl-4-oxobutanamide
[(5-chlorothiophen-2-yl)methyl]({[2-(morpholine-4-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl})amine
(4aS,8aR)-6-(1,3-benzoxazol-2-yl)-1-(3-methoxypropyl)-decahydro-1,6-naphthyridin-2-one
2-(1H-pyrazol-1-yl)-N-[1-(pyridin-2-yl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]benzamide
3-butyl-4-ethyl-1-{2-oxo-2-[4-(propan-2-yl)piperazin-1-yl]ethyl}-4,5-dihydro-1H-1,2,4-triazol-5-one
3-[5-(2-cyclopentylacetyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]-N-(2-hydroxyethyl)propanamide
2-(dimethylamino)-2-(4-fluorophenyl)-1-[4-(morpholin-4-yl)piperidin-1-yl]ethan-1-one
(2-{2-[1-(isoquinolin-1-yl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)dimethylamine
(5S,9aS,9bS)-2-[(3-methoxyphenyl)methyl]-5-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
2-[1'-(6-methylpyridine-2-carbonyl)-2-oxo-1,2-dihydrospiro[indole-3,3'-pyrrolidine]-1-yl]acetamide
2-(1H-1,2,4-triazol-1-ylmethyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-({2-methyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}(2-phenylethyl)amino)propanamide
N-{1-[(4-fluorophenyl)methyl]piperidin-3-yl}-2-(propan-2-yl)pyrimidine-5-carboxamide