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N-[2-(benzylsulfanyl)ethyl]-2-(2-oxopyrrolidin-1-yl)propanamide
N-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-[4-(2-methylquinolin-4-yl)-2-(morpholin-4-ylmethyl)phenoxy]acetamide
2-ethyl-8-[2-(3-methyl-6-oxo-1,6-dihydropyridazin-1-yl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
N-(2-methanesulfonamidoethyl)-2-(trimethyl-1H-pyrazol-1-yl)acetamide
N3-cycloheptyl-1-cyclopropyl-N5-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
ethyl 3-[(2,4-difluorophenyl)methyl]-1-(pyridine-3-sulfonyl)piperidine-3-carboxylate
2-(4-methoxy-2-methylphenyl)-2-{methyl[2-(morpholin-4-yl)ethyl]amino}acetic acid
N-(1-phenylbutyl)pyridine-4-carboxamide
1-{4-[(2,3-dihydroxypropyl)(methyl)amino]-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl}ethan-1-one
2-{5-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]-1H-pyrazol-3-yl}phenol
4,4,4-trifluoro-1-{3-[1-(pyrimidin-2-yl)piperidin-4-yl]pyrrolidin-1-yl}butan-1-one
4-hydroxy-N-(2-hydroxy-3-methoxypropyl)-2-phenylpyrimidine-5-carboxamide
2-amino-4-(5-cyclopropyl-1-methyl-1H-pyrazol-4-yl)-6-(4-methoxyphenyl)pyridine-3-carbonitrile
N-[2-(1-{[3-(3-methoxyphenyl)-1-phenyl-1H-pyrazol-4-yl]methyl}piperidin-2-yl)ethyl]acetamide
6-{4-[4-cyclopropyl-5-(1H-imidazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyrimidin-4-amine
2-methoxy-1-{4-[3-(3-methoxyphenyl)-1H-pyrazole-4-carbonyl]-1,4-diazepan-1-yl}ethan-1-one
4-(2,3-dimethoxybenzoyl)-2-(4-methylpentyl)morpholine
(2S)-1-{5-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyridin-2-yl}pyrrolidine-2-carboxamide
1-methanesulfonyl-N-(6-phenoxypyridin-3-yl)piperidine-2-carboxamide
1-methyl-3-{2-methyl-2H,4H,5H,6H-cyclopenta[c]pyrazol-3-yl}-1-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}urea
N-[(4-fluorophenyl)methyl]-3-(1-{[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl}piperidin-4-yl)propanamide
(1R,5R)-6-[(2-methoxyphenyl)methyl]-3-(pyrazine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
2-{3-[3-(pyrimidin-2-yl)phenyl]-1H-pyrazol-1-yl}-N-(1,3-thiazol-2-yl)butanamide
1-(cyclopropylmethyl)-2-(propan-2-yl)-4-(pyrazine-2-carbonyl)-1,4-diazepane
1-(3-chlorophenyl)-4-[3-(4H-1,2,4-triazol-4-yl)benzoyl]piperazin-2-one
(2S)-2-({5-chloro-2-[(1-cyclopentylpiperidin-4-yl)oxy]phenyl}formamido)propanamide
(2S,4R)-4-amino-1-(2,3-dimethyl-1H-indole-7-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
4-{5-fluoro-2-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]pyrimidin-4-yl}morpholine
7-(3-chlorophenyl)-4-cyclopropanecarbonyl-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepine
6-methoxy-N-methyl-N-{2-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]ethyl}pyrimidin-4-amine
N-[(1-ethyl-5-methyl-1H-pyrazol-4-yl)methyl]-N,1,3-trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2,6-dimethyl-5-{2-oxo-2-[4-(2-phenoxyethyl)piperazin-1-yl]ethyl}-3,4-dihydropyrimidin-4-one
1-(2-fluoro-6-methoxybenzoyl)-3-(3-methoxypropyl)piperidine
2-(4-{1-[(4-ethylphenyl)methyl]-1H-1,2,4-triazol-5-yl}piperidin-1-yl)acetamide
7-fluoro-3-methyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-N-(pyridin-4-ylmethyl)-1-benzofuran-2-carboxamide
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-[(3-methyl-1-benzofuran-2-yl)methyl]pyrrolidin-3-yl]methanol
2-({1-[(2S)-2-aminopropanoyl]piperidin-4-yl}oxy)-4-methoxy-N-(2-methoxyethyl)benzamide
4-{7-[2-(furan-2-yl)-2-oxoacetyl]-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl}benzamide
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-[methyl(pyridin-4-ylmethyl)amino]acetamide
N-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-[(quinolin-6-yloxy)methyl]-1,3-oxazole-4-carboxamide
1-[1-(1,3-dimethyl-1H-pyrazole-5-carbonyl)piperidin-3-yl]-4-(2-methylphenyl)piperazine
2-(3-{1-[(1-methylpiperidin-3-yl)methyl]-1H-pyrazol-3-yl}phenyl)pyrazine
3-(4-methyl-1,3-thiazol-5-yl)-N-{pyrazolo[1,5-a]pyridin-3-ylmethyl}propanamide
(3aR,7aS)-N-(2-fluoro-5-methanesulfonamidophenyl)-2,3,3a,4,7,7a-hexahydro-1H-isoindole-2-carboxamide
(1S,5R)-6-benzyl-3-(1H-imidazol-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
N-[(1-hydroxycyclohexyl)methyl]-1-{1-[(6-methylpyridin-2-yl)methyl]piperidin-4-yl}piperidine-4-carboxamide
N-[1-(2-chlorophenyl)cyclopropyl]-1-(methoxymethyl)cyclobutane-1-carboxamide
[(3S,5R)-1-(2-methyl-1H-1,3-benzodiazole-5-carbonyl)-5-(morpholin-4-ylmethyl)piperidin-3-yl]methanol
4-(2-methoxyphenoxy)-1-(piperidin-3-yl)piperidine
methyl 3-[(3S,4R)-4-(morpholin-4-yl)-1-{[2-(prop-2-en-1-yloxy)phenyl]methyl}piperidin-3-yl]propanoate