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6-methyl-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]pyrazolo[1,5-a]pyrimidine-3-carboxamide
5-[(3-fluorophenyl)methyl]-7-{[(3-hydroxypropyl)amino]methyl}-2H,5H,6H-[1,3]dioxolo[4,5-g]quinolin-6-one
6-(methoxymethyl)-N,1-dimethyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-1H-pyrazolo[3,4-d]pyrimidin-4-amine
1-(pyridin-3-yl)-4-(2,3,4,5-tetrahydro-1-benzoxepine-4-carbonyl)piperazine
5-(3-methyl-1H-pyrazol-1-yl)pyridine-3-carboxamide
N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methyl-N'-(2-methylphenyl)propanediamide
(2S)-2-{[1-methyl-6-(2-phenylethyl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}propanamide
9-[2-(propan-2-ylsulfanyl)ethyl]-2-(pyridin-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
3-(3-chlorophenyl)-3-(3-hydroxyphenyl)-N-methyl-N-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]propanamide
1-[(4-fluorophenyl)methanesulfonyl]-N-(piperidin-4-yl)azepan-3-amine
ethyl 4-{[1-(pyrimidin-2-yl)-1H-pyrrol-2-yl]methyl}piperazine-1-carboxylate
{2-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-oxoethyl}urea
N-{[2-(1H-imidazol-1-yl)phenyl]methyl}-8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-amine
(2R,3R,6R)-3-(2-methoxyphenyl)-5-(5-methylpyridine-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-[2-(3-methoxyphenyl)azetidine-1-carbonyl]-5-(propan-2-yl)-1,2-oxazole
5-{4-[(2-methylphenyl)methyl]piperazine-1-carbonyl}-N-phenylpyrimidin-2-amine
1-[(2-fluorophenyl)methyl]-6-oxo-N-(1-phenylcyclopropyl)piperidine-3-carboxamide
2-(ethylsulfanyl)-5-{[4-(pyrrolidine-1-sulfonyl)piperazin-1-yl]methyl}pyrimidine
1-methoxy-8-[(4-phenyl-1,3-thiazol-2-yl)methyl]-1,8-diazaspiro[4.5]decan-2-one
[2-(2-ethylphenoxy)ethyl](1H-imidazol-2-ylmethyl)methylamine
6-methyl-2-[2-({2,3,5-trimethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]-3,4-dihydropyrimidin-4-one
4-({2-[2-(1H-imidazol-1-yl)ethoxy]-3-methoxyphenyl}methyl)-2-(trifluoromethyl)morpholine
(4aS,7aR)-1-[2-(2H-1,3-benzodioxol-5-yl)acetyl]-4-propyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[6,6-dimethyl-1-(4-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-(1H-1,2,3,4-tetrazol-1-yl)propanamide
1-[(2-chlorophenyl)methyl]-N-[2-(2-oxopiperidin-1-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
(2S,4S)-4-amino-N,N-diethyl-1-(4-propoxybenzoyl)pyrrolidine-2-carboxamide
N,N-dimethyl-5-(1-{[5-(1H-pyrazol-5-yl)thiophen-2-yl]methyl}pyrrolidin-2-yl)thiophene-2-carboxamide
1-ethyl-3-{[4-(5-ethylpyridin-2-yl)-1H-1,2,3-triazol-1-yl]methyl}-1H-indazole
2-[(4-methanesulfonylphenyl)methyl]-1,2-dihydrophthalazin-1-one
N-[4-(4-{[2-methyl-2-(morpholin-4-yl)propyl]amino}piperidin-1-yl)phenyl]-2-phenoxyacetamide
2-(furan-2-yl)-1-[3-(1H-pyrazol-1-yl)benzoyl]azepane
2-({5-[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl]-4-methyl-4H-1,2,4-triazol-3-yl}sulfanyl)acetic acid
4-[(6-methylhept-5-en-2-yl)amino]adamantan-1-ol
4-{[2-methanesulfonyl-1-(2-methylpropyl)-1H-imidazol-5-yl]methyl}-1-(3-methoxyphenyl)piperazin-2-one
3-[2-(2-butyl-2,5-dihydro-1H-pyrrol-1-yl)-2-oxoethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-(6-cyclopropylpyrimidin-4-yl)-N-(pyridin-3-ylmethyl)-1H-pyrrolo[2,3-b]pyridin-6-amine
1-[4-(3-fluoropyridin-4-yl)-6-hydroxy-1,4-diazepan-1-yl]ethan-1-one
dimethyl[1-(1-{[4-(pyrrolidin-1-ylmethyl)thiophen-2-yl]methyl}piperidin-4-yl)ethyl]amine
N1-(pyridin-3-yl)-N3-[2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl]propane-1,3-diamine
2-ethyl-1-{2-[2-(pyrrolidine-1-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-5-yl]propyl}-1H-imidazole
1-[(2-chloro-6-fluorophenyl)methyl]-3-(2-methyl-1,3-thiazol-4-yl)-5-(pyrrolidin-3-yl)-1H-1,2,4-triazole
(4aR,8aR)-4a-hydroxy-N,N-dimethyl-7-(5,6,7,8-tetrahydroquinolin-2-yl)-decahydro-2,7-naphthyridine-2-carboxamide
(5S)-5-[3-oxo-3-(4-phenyl-1,4-diazepan-1-yl)propyl]imidazolidine-2,4-dione
N,N-diethyl-1-(prop-2-en-1-yl)-3-(pyrrolidine-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
1-[benzyl(methyl)amino]-3-(4-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}phenoxy)propan-2-ol
N-(1-{7-[(6-methylpyridin-2-yl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-2-carboxamide
N-{2-[(4-chlorophenyl)sulfanyl]ethyl}-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
1-[3-(azetidine-1-carbonyl)benzenesulfonyl]-2-(3-methoxypropyl)piperidine
3-[(3R,4S)-3-amino-4-propylpyrrolidine-1-carbonyl]-1-methyl-1,2-dihydroquinoxalin-2-one
2-[1-(1-ethylpiperidin-3-yl)piperidin-4-yl]ethan-1-ol