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N-[2-(3-phenylpropoxy)phenyl]-2-(1H-1,2,4-triazol-1-yl)acetamide
N-[3-(2,4-dimethylphenoxy)propyl]-N-methyl-1-phenyl-1H-1,2,3-triazole-4-carboxamide
2-{1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-3-oxopiperazin-2-yl}-N-methylacetamide
5-[4-(2-methanesulfonylethyl)piperazine-1-carbonyl]-1H-pyrrole-3-carbonitrile
9-[5-fluoro-2-(1H-pyrazol-1-yl)phenyl]-1H,2H,3H,6H,7H,8H,9H-[1,4]oxazino[3,2-g]quinoline-2,7-dione
1-(3-benzyl-4,5-dihydro-1,2-oxazole-5-carbonyl)-4-[(4-fluorophenyl)sulfanyl]piperidine
N-[(4-methoxyphenyl)methyl]-N-propyl-3-(1H-pyrazol-1-yl)butanamide
(3S,4S)-3-{[(2-butoxy-3-methoxyphenyl)methyl](methyl)amino}-4-hydroxy-1λ6-thiolane-1,1-dione
5-[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]-N-[1-(1H-pyrazol-1-yl)propan-2-yl]pyridin-2-amine
2-methoxy-5-methyl-N-{[1-(3,3,3-trifluoropropyl)pyrrolidin-3-yl]methyl}benzamide
1-[2-(dimethylamino)ethyl]-4-(5,6,7,8-tetrahydro-1,6-naphthyridine-6-carbonyl)pyrrolidin-2-one
(3S,4R)-4-(3-methylthiophen-2-yl)-1-[3-(1H-pyrazol-4-yl)benzoyl]piperidin-3-ol
3-[(4-tert-butyl-1H-1,2,3-triazol-1-yl)methyl]-1-{[1,2,4]triazolo[1,5-a]pyrimidine-2-carbonyl}piperidine
N-cyclopropyl-5-[4-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
4-(1-{1-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]piperidin-4-yl}-1H-1,2,3-triazole-4-carbonyl)morpholine
2-(dimethylamino)-2-(3-methylphenyl)-N-[3-(1H-1,2,3-triazol-1-yl)propyl]acetamide
1-ethyl-6-methyl-N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}-2-oxo-1,2-dihydropyridine-3-carboxamide
1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-(2,6-dimethylpyridin-4-yl)piperazine
N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}-3-(pyridin-3-yl)propanamide
1-ethyl-4,6-dimethyl-N-{[1-(2-methylpropyl)pyrrolidin-3-yl]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
N-[2-(benzyloxy)phenyl]-9-oxa-2-azaspiro[5.5]undecane-2-carboxamide
6-(2H-1,3-benzodioxol-5-yl)-N-{3-[2-(propan-2-yl)-1H-imidazol-1-yl]propyl}pyridine-3-carboxamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-5-ethyl-N-methylpyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(dimethylamino)ethyl]-3-(2-fluorophenyl)-N-(2-hydroxyethyl)-1H-pyrazole-4-carboxamide
5-methoxy-3-methyl-2-(thiomorpholine-4-carbonyl)-1H-indole
5-ethyl-N-[2-(pyridin-3-yloxy)propyl]pyrazolo[1,5-a]pyrimidin-7-amine
N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanamide
3-(4-fluorophenyl)-N-(2-{5-[(2-methoxyethyl)sulfanyl]-4-methyl-4H-1,2,4-triazol-3-yl}ethyl)benzamide
2-(1-{[3-(1H-pyrazol-1-yl)phenyl]methyl}pyrrolidin-3-yl)benzoic acid
4-{[7,7-dimethyl-2-(morpholin-4-yl)-5,6,7,8-tetrahydroquinazolin-5-yl]carbamoyl}pyridin-1-ium-1-olate
N4-[cyclopropyl(1-methyl-1H-imidazol-2-yl)methyl]-6-ethyl-N2,N2-dimethylpyrimidine-2,4-diamine
1-cyclohexyl-N-{[1-(2-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-1H-1,2,3-triazole-4-carboxamide
5-[2-(methylsulfanyl)phenoxymethyl]-N-[(3S)-2-oxoazepan-3-yl]-1,2-oxazole-3-carboxamide
N-[(3-propyl-1,2-oxazol-5-yl)methyl]-2-(pyridin-4-yl)pyrimidine-5-carboxamide
5-chloro-2-{7-methyl-3,7,11-triazaspiro[5.6]dodecane-11-carbonyl}phenol
2-benzyl-4-[2-(methylsulfanyl)benzoyl]morpholine
N-{5H,6H,7H-cyclopenta[b]pyridin-3-ylmethyl}-1-methyl-6-oxo-1,6-dihydropyridine-3-carboxamide
5-{2-[2-(2,2-dimethyloxan-4-yl)-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-{[2-(diethylamino)pyridin-3-yl]methyl}cyclobutanecarboxamide
2-ethyl-9-[(2-methyl-1,3-oxazol-4-yl)methyl]-4-phenyl-2,9-diazaspiro[5.5]undecan-3-one
2-{[2-(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-3-yl)-1H-imidazol-1-yl]methyl}pyridine
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-1,2-oxazole-5-carboxamide
2-{1-[1-ethyl-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-5-yl]propyl}-2,3-dihydro-1H-isoindol-1-one
1-{1-oxa-8-azaspiro[4.5]decan-8-yl}-2-[2-(propan-2-yl)-1H-imidazol-1-yl]propan-1-one
3-(propan-2-yl)-1-{[1-(2,2,6,6-tetramethylpiperidin-4-yl)pyrrolidin-3-yl]methyl}urea
N-[(1-benzyl-1H-pyrazol-4-yl)methyl]-2-(pyrazin-2-yl)acetamide
(2S)-1-[(2-butoxy-3-methoxyphenyl)methyl]-N,N-dimethylpyrrolidine-2-carboxamide
2-(4-{[4-(benzyloxy)phenyl]methyl}-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl)-1-(dimethylamino)propan-2-ol
(3S,4R)-1-[(5-ethylpyridin-2-yl)methyl]-4-(2-methylphenyl)pyrrolidine-3-carboxylic acid
1-{1-[1-(2H-1,3-benzodioxol-5-yl)-3-methyl-1H-1,2,4-triazol-5-yl]ethyl}-1H-1,3-benzodiazole