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N-[2-(4-fluorophenyl)ethyl]-1-methyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-fluoro-N,3-dimethyl-N-[(1-phenylpyrrolidin-3-yl)methyl]-1H-indole-2-carboxamide
5-[1-(6-methanesulfonamidopyridin-3-yl)-1H-imidazol-2-yl]thiophene-2-carboxylic acid
1-(4-{[(2,3-dihydro-1H-inden-2-yl)amino]methyl}-2-methoxyphenoxy)-3-(morpholin-4-yl)propan-2-ol
2-[4-(dimethylamino)-6-oxo-1,6-dihydropyridazin-1-yl]-N-(2,4,6-trimethylphenyl)acetamide
(4aS,7aR)-1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-[4-(2-amino-6-methylpyrimidin-4-yl)-1H-pyrazol-1-yl]-N-(3-methyl-1-phenyl-1H-pyrazol-5-yl)acetamide
4-phenyl-2-{[3-(2-phenylethyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2-dihydrophthalazin-1-one
3-[3-(4-methylpiperazin-1-yl)propyl]-1-{3-[(E)-2-(pyridin-2-yl)ethenyl]phenyl}urea
5-{[4-(benzyloxy)piperidin-1-yl]methyl}quinoxaline
4-{1-[2-(4-ethoxyphenyl)-1H-imidazol-1-yl]-2-methylpropan-2-yl}morpholine
N-[1-(2,3-dihydro-1,4-benzodioxin-6-yl)ethyl]-N-methyl-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
N-[(2,3-dimethoxyphenyl)methyl]-4-methyl-5-[1-(pyridin-4-ylmethyl)-1H-pyrazol-3-yl]-1,3-thiazol-2-amine
1-(3-{[5-methyl-6-(2-methylpiperidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-yl]amino}propyl)pyrrolidin-2-one
3-(furan-2-yl)-N-[(5-methyl-1H-1,2,4-triazol-3-yl)methyl]-3-phenylpropanamide
N,N-dimethyl-5-[({[2-(propan-2-ylsulfanyl)phenyl]carbamoyl}amino)methyl]furan-2-carboxamide
1-cyclohexyl-N3-methyl-4-oxo-N5-{[4-(trifluoromethoxy)phenyl]methyl}-1,4-dihydropyridine-3,5-dicarboxamide
4-(1H-1,3-benzodiazol-1-yl)-1-(dimethylsulfamoyl)piperidine-4-carboxylic acid
2-(3-fluoro-2,4-dimethylphenyl)-1-[2-(1H-imidazol-4-yl)ethyl]-1H-imidazole
2-(dimethyl-1,3-thiazol-5-yl)-1-[4-(1H-imidazol-2-yl)piperidin-1-yl]ethan-1-one
N-(1,4-dimethyl-3-phenyl-1H-pyrazol-5-yl)-4-methyl-1,2,3,6-tetrahydropyridine-1-carboxamide
N-{[2-(diethylamino)pyridin-3-yl]methyl}-2-(pyridin-4-yl)acetamide
(3R,5S)-5-{4-[2-(3-methoxyphenoxy)ethyl]piperazine-1-carbonyl}pyrrolidin-3-amine
4-[1-(2-fluorophenyl)-1H-pyrazol-4-yl]-N-(furan-2-ylmethyl)pyrimidin-2-amine
(3aR,6aR)-2-methanesulfonyl-5-(3-phenoxypropyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-{[3-(pyridin-3-yl)-1,2,4-oxadiazol-5-yl]methyl}-1-(pyrrolidin-1-yl)cyclopentane-1-carboxamide
(2E)-N-({3-[(2-chloroprop-2-en-1-yl)oxy]-4-methoxyphenyl}methyl)-N-cyclopropyl-3-(thiophen-2-yl)prop-2-enamide
N-(5-oxo-1-{[2-(trifluoromethyl)phenyl]methyl}pyrrolidin-3-yl)-2-(piperidin-1-yl)acetamide
{1-[(6-ethoxyquinolin-2-yl)methyl]pyrrolidin-3-yl}methanamine
5-methyl-N-(oxolan-3-yl)-6-[4-(1,2,3,4-tetrahydroisoquinolin-2-yl)piperidine-1-carbonyl]thieno[2,3-d]pyrimidin-4-amine
(2R,3R)-1'-(2-ethoxyethyl)-3-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
2-{4-[(2,5-dimethoxyphenyl)methyl]-1-[(4-methoxy-2,3-dimethylphenyl)methyl]piperazin-2-yl}ethan-1-ol
8-{[3-(pyridin-2-yl)phenyl]methyl}-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
2-{[4-(3-chloro-4-hydroxy-5-methoxyphenyl)-2-oxo-1,2,3,4-tetrahydroquinolin-7-yl]oxy}acetic acid
2,4-dimethyl-5-{octahydro-1H-pyrido[1,2-a]piperazine-2-carbonyl}pyrimidine
3-(4-hydroxyphenyl)-N-{[1-(methoxymethyl)cyclopentyl]methyl}-1H-pyrazole-5-carboxamide
1-{imidazo[1,2-a]pyridine-2-carbonyl}-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
N-cyclopropyl-2-[(E)-2-phenylethenyl]pyridine-4-carboxamide
2-{1-[(3-fluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-hydroxyethyl)-N-methylacetamide
2-[(1-cyclohexylpiperidin-4-yl)formamido]-2-(3-hydroxyphenyl)acetic acid
ethyl 4-(2-phenoxyethyl)-1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-ylmethyl)piperidine-4-carboxylate
6-chloro-2-{2-[7-(2,2-dimethylpropyl)-2,7-diazaspiro[4.5]decan-2-yl]-2-oxoethyl}-2,3-dihydropyridazin-3-one
[1-(1H-1,3-benzodiazol-2-yl)ethyl]({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)amine
2-(4-ethyl-3,5-dimethyl-1H-pyrazol-1-yl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
[4-({1-[(6-ethoxyquinolin-2-yl)methyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-[(5-cyclobutyl-1,2,4-oxadiazol-3-yl)methyl]-N-ethyl-2-fluoro-5-sulfamoylbenzamide
methyl 2-(4-{1-[N-methyl-1-(2-methylfuran-3-yl)formamido]-2-phenylethyl}piperidine-1-carbonyl)benzoate
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-3-(4-methyl-1,3-thiazol-5-yl)propanamide
7-(2-methoxyacetamido)-1-methyl-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]-2-phenyl-1H-1,3-benzodiazole-5-carboxamide
3-[({[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}carbamoyl)amino]-N-(propan-2-yl)benzamide