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N,1,3-trimethyl-2,6-dioxo-N-(4,5,6,7-tetrahydro-1,2-benzoxazol-3-ylmethyl)-1,2,3,6-tetrahydropyrimidine-4-carboxamide
[(3R,4R)-1-(dimethyl-1,3-oxazole-4-carbonyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-3-yl]methanol
(1R,7S)-N-ethyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-oxo-3-(pyridin-3-ylmethyl)-10-oxa-3-azatricyclo[5.2.1.01,5]dec-8-ene-6-carboxamide
2-(dimethylamino)-2-(2-fluorophenyl)-1-[4-(pyridin-3-ylmethyl)-1,4-diazepan-1-yl]ethan-1-one
1-[2-methyl-4-({2-[(1-methyl-1H-1,2,3,4-tetrazol-5-yl)sulfanyl]ethyl}amino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-7-yl]ethan-1-one
3,5-difluoro-N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]pyridine-2-carboxamide
5-[5-(2H-indazol-2-ylmethyl)-1,2,4-oxadiazol-3-yl]-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridine
methyl 2-(diethylsulfamoyl)-6-[(2-methylphenyl)methyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
N-[2-(3,4-dimethoxyphenyl)ethyl]-N-methyl-3-(2-methyl-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl)propanamide
1-[(3S,4R)-3-hydroxy-4-(hydroxymethyl)piperidin-1-yl]-2-[(3-methoxyphenyl)sulfanyl]ethan-1-one
1-{[4-(methylsulfanyl)phenyl]methyl}-N-[4-(1H-pyrazol-5-yl)phenyl]piperidine-3-carboxamide
1-{5-[3-(hydroxymethyl)-3-(3-phenylpropyl)piperidine-1-carbonyl]-1H-pyrazol-3-yl}ethan-1-one
{2-methyl-6-[2-(2-phenylethyl)pyrrolidin-1-yl]pyrimidin-4-yl}methanamine
N-methyl-2-(2-methyl-1,3-thiazol-4-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}acetamide
2-(5-methyl-1H-pyrazol-1-yl)-1-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]ethan-1-one
1-[1-(3-fluoro-4-methoxyphenyl)ethyl]-2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazole
(2S,4R)-4-[3-(4,5-dimethyl-1H-pyrazol-3-yl)propanamido]-N,N-diethyl-1-methylpyrrolidine-2-carboxamide
4-(4-cyclopentyl-1H-1,2,3-triazol-1-yl)-1-(2,2,3,3-tetramethylcyclopropanecarbonyl)piperidine
2-methoxy-N-methyl-5-({[1-(4,5,6,7-tetrahydro-1,3-benzothiazol-2-yl)ethyl]carbamoyl}amino)benzamide
1-(4-fluoro-3-methoxyphenyl)-2-(4,4,4-trifluorobutyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indole
6-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}pyridine-2-carboxylic acid
N-(2-hydroxyethyl)-N-(1,3-thiazol-2-ylmethyl)-2,3,4,9-tetrahydro-1H-carbazole-7-carboxamide
4-ethyl-1-methyl-3-[1-(1-phenylpiperidin-4-yl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
4-amino-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
1-[1-(2-hydroxyethyl)-1H-1,3-benzodiazol-2-yl]-3-(piperidin-1-ylmethyl)pyrrolidin-3-ol
(1R,2R,3R,4S)-N-cyclopropyl-3-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decane-8-carbonyl}bicyclo[2.2.1]hept-5-ene-2-carboxamide
2-[2-(2,5-dimethylfuran-3-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]-6-methylpyridine
7-(4-methylphenyl)-4-[5-(propan-2-yl)-1,3-oxazole-4-carbonyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2-[2-(propan-2-yloxy)acetyl]-1,2,3,4-tetrahydroisoquinoline-6-sulfonamide
2-[2-(3-methoxyphenyl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]-1,3-thiazole-4-carboxamide
2-{[2-(2,3-dimethoxyphenyl)-1H-imidazol-1-yl]methyl}-1,3-benzothiazole
N-methyl-2-(pyrrolidin-3-yl)-N-(quinolin-8-ylmethyl)benzamide
5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-(3-methylbutyl)-1,2-oxazole-3-carboxamide
[(3-fluorophenyl)methyl]({[6-(thiophen-3-yl)-2H-[1,3]dioxolo[4,5-g]quinolin-7-yl]methyl})amine
1-{1-[(3-chloro-5-fluoro-4-methoxyphenyl)methyl]piperidin-4-yl}piperidin-3-ol
2-[4-(4-phenyl-1H-pyrazol-5-yl)piperidin-1-yl]pyrimidin-4-amine
[(3-{2-[4-(2,1,3-benzothiadiazole-4-sulfonyl)piperazin-1-yl]ethoxy}phenyl)methyl](methyl)(thiophen-2-ylmethyl)amine
4-(4-methylpiperazin-1-yl)-6-[4-(methylsulfanyl)phenyl]pyrimidin-2-amine
2-methyl-6-[2-(4-methyl-1,3-oxazole-5-carbonyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl]pyridine
[1-(5-methyl-1-phenyl-1H-pyrazol-4-yl)ethyl]({[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl})amine
3-hydroxy-3-({[2-(morpholin-4-yl)ethyl]amino}methyl)-1-{[4-(propan-2-yl)phenyl]methyl}piperidin-2-one
N-{[3-(2-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-N-[(trimethyl-1H-pyrazol-4-yl)methyl]cyclopropanamine
1-(5-{[(dimethylsulfamoyl)amino]methyl}-6-methyl-1,2,3,4-tetrahydro-2,7-naphthyridin-2-yl)-2-(1H-indol-3-yl)ethan-1-one
N-({1-[(7-methoxy-2-oxo-1,2-dihydroquinolin-3-yl)methyl]piperidin-4-yl}methyl)acetamide
4-({2-[1-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-3-yl]-1H-imidazol-1-yl}methyl)pyridine
N-({3-[(dimethylamino)methyl]phenyl}methyl)-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
N,2-dimethyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
(1R,3S)-7-(5-chloropyridine-2-carbonyl)-3-(2-hydroxyethoxy)-7-azaspiro[3.5]nonan-1-ol
2-(3-oxo-2,3-dihydro-1H-isoindol-1-yl)-N-[2-(4-sulfamoylphenyl)ethyl]acetamide