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(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(thiophene-3-carbonyl)-decahydro-1,6-naphthyridin-2-one
(3S,4R)-1-(1-benzoylpiperidin-4-yl)-3-benzyl-4-methylpiperidin-4-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-3-ol
4-{[2-fluoro-3-(trifluoromethyl)phenyl]methyl}-1,3λ6,4-oxathiazinane-3,3-dione
2-{1-tert-butyl-3-[2-(methylsulfanyl)ethyl]-1H-1,2,4-triazol-5-yl}ethan-1-ol
N-benzyl-N-{[(2S)-5-oxopyrrolidin-2-yl]methyl}-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
(3S,9aR)-3-[(benzyloxy)methyl]-8-{[4-(4-fluorophenyl)-1,3-thiazol-2-yl]methyl}-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
N-(adamantan-1-yl)-6-{[benzyl(ethyl)amino]methyl}-2-oxo-1,2-dihydropyridine-3-carboxamide
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](4-phenylbutan-2-yl)amine
2-({[(3R,4R)-1-(3,5-dichlorobenzoyl)-4-(hydroxymethyl)pyrrolidin-3-yl]methyl}(methyl)amino)ethan-1-ol
6-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-9H-purin-2-amine
[(5-{[(2-chlorophenyl)methyl]sulfanyl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl](methyl)[(2E)-3-phenylprop-2-en-1-yl]amine
2-[4-fluoro-3-(trifluoromethyl)phenyl]-2-{methyl[2-(1-methyl-1H-pyrazol-4-yl)ethyl]amino}acetic acid
1-{3-[2-(morpholin-4-ylmethyl)piperidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
2-(dimethyl-1,2-oxazol-4-yl)-N-[1-(dimethyl-1,3-thiazol-2-yl)propyl]acetamide
2-{ethyl[3-(morpholin-4-yl)propyl]amino}-2-(2-methoxy-5-methylphenyl)acetic acid
2-methyl-5-{[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]methyl}pyrazine
N-{4-[2-(2-acetamidoethyl)piperidine-1-carbonyl]phenyl}pentanamide
N-(3-phenylpropyl)-5-[(quinolin-6-yloxy)methyl]-1,2-oxazole-3-carboxamide
1-{[4-(dimethylamino)phenyl]methyl}-4-(2-methylpropyl)-1,4-diazepan-5-one
3-(4-cyclopentylpiperazin-1-yl)-5-(2-methylphenyl)-1,2,4-triazine
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)-1H-pyrazole-4-carboxamide
1-methyl-3-propyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H-pyrazole-5-carboxamide
3-chloro-N-[2-(dimethylamino)ethyl]-4-({1-[(1-ethyl-1H-imidazol-2-yl)methyl]piperidin-4-yl}oxy)benzamide
N-ethyl-3-(3-methoxyphenyl)-N-[(5-methylfuran-2-yl)methyl]-1H-pyrazole-4-carboxamide
2-[(4-methyl-1,2,5-oxadiazol-3-yl)methyl]-4-[3-(2-methylpiperidine-1-carbonyl)piperidin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N,1,4,6-tetramethyl-2-oxo-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,2-dihydropyridine-3-carboxamide
N-[1-(cyclopropylmethyl)-1H-indazol-3-yl]-2-{1H-pyrazolo[3,4-b]pyridin-1-yl}acetamide
methyl({5-[(oxolan-2-ylmethyl)sulfanyl]-4-(prop-2-en-1-yl)-4H-1,2,4-triazol-3-yl}methyl){[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}amine
1-methyl-4-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]-4-phenylpiperidine
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}-2-(4-methylphenoxy)ethan-1-one
1-{2-methyl-5-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]phenyl}imidazolidin-2-one
methyl 9-(benzyloxy)-3-(oxan-4-yl)-7-oxo-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
5-(1,3-thiazol-4-yl)-3-(thiophen-2-ylmethyl)-1,2,4-oxadiazole
1-{3,9-diazaspiro[5.5]undecan-3-yl}-4-(1H-imidazol-1-yl)butan-1-one
5-[4-(4-cyclohexyl-1H-1,2,3-triazol-1-yl)piperidine-1-carbonyl]-1H-indole
(3aR,6aS)-5-(2,3-dihydro-1-benzofuran-5-carbonyl)-2-ethyl-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{2-[3-(dimethylamino)pyrrolidin-1-yl]ethyl}-8-(furan-2-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
3-[(1,1-dioxo-1λ6-thiolan-3-yl)(methyl)amino]-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)propanamide
1-{[6-chloro-2-(1,2,3,4-tetrahydroisoquinoline-2-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}azetidin-3-ol
3-{1-[(2E)-3-(1,3-benzothiazol-2-yl)prop-2-enoyl]piperidin-3-yl}-N-cyclopropylpropanamide
8-(1H-imidazol-2-ylmethyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-amino-6-methyl-4-[5-methyl-2-(1H-pyrazol-1-yl)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-{2-[3-(naphthalene-2-carbonyl)piperidin-1-yl]-2-oxoethyl}methanesulfonamide
3-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-1,2-dihydroquinoxalin-2-one
N-({5-cyclohexyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}methyl)-1H-1,3-benzodiazole-5-carboxamide
4-(4-{5-[(dimethylamino)methyl]-4-ethyl-4H-1,2,4-triazol-3-yl}piperidine-1-carbonyl)phenol
N-cyclopropyl-4-fluoro-N-{[3-(oxolan-2-ylmethoxy)phenyl]methyl}benzamide
(4aS,8aR)-6-(1,3-benzoxazol-2-yl)-1-[3-(1H-imidazol-1-yl)propyl]-decahydro-1,6-naphthyridin-2-one
3-ethyl-8-(2-methoxyquinoline-4-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one