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4-[4-(ethanesulfonyl)piperazin-1-yl]-2-methyl-6-(piperidin-4-yl)pyrimidine
N-(4-fluoro-3-methoxyphenyl)-3-(methoxymethyl)pyrrolidine-1-carboxamide
(2,1,3-benzothiadiazol-5-ylmethyl)(methyl){4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-ylmethyl}amine
2-(4-{6-amino-1H-pyrrolo[2,3-b]pyridin-4-yl}-1H-pyrazol-1-yl)propanoic acid
N-(4,7-dimethyl-2-oxo-2H-chromen-6-yl)-2-(1H-indol-3-yl)acetamide
2-(3-methoxypropyl)-N-methyl-3-oxo-N-phenyl-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-(isoquinolin-5-ylmethyl)-N-methyl-2-[1-(3-methylbutyl)-3-oxopiperazin-2-yl]acetamide
2-{[3-(azepane-1-carbonyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}-2-methylpropan-1-ol
5-methyl-4-(1-methyl-1H-pyrazole-4-carbonyl)-1-(2-phenylphenyl)piperazin-2-one
N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
N-ethyl-1-methyl-N-[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]-1H-indole-3-carboxamide
4-[(2,3-difluoro-6-methoxyphenyl)methyl]morpholine-2-carboxylic acid
[(3R,4R)-4-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-1-[1-(4-methylphenyl)cyclopropanecarbonyl]pyrrolidin-3-yl]methanol
N-(1,3-benzothiazol-2-ylmethyl)-N-methyl-3-(1H-pyrazol-1-yl)benzamide
1-[2-(naphthalen-1-ylmethyl)morpholin-4-yl]-3-(pyrazin-2-yl)propan-1-one
3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]-N-[(5-methylthiophen-2-yl)methyl]propanamide
4-benzyl-3-ethyl-1-(1-methyl-1H-pyrazole-4-carbonyl)-1,4-diazepan-5-one
(2S,4S)-4-amino-1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
N-(1-{[4-(2-methylpropyl)phenyl]methyl}piperidin-3-yl)-1H-imidazole-5-carboxamide
1-{2-[2-(1-methyl-1H-pyrrol-3-yl)acetamido]ethyl}-N-[1-(thiophen-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
5-methanesulfonyl-4-[3-(2-methoxyphenoxy)azetidin-1-yl]-2-methylpyrimidine
N-cyclopropyl-2-(7-methyl-3-oxo-3,4-dihydro-2H-1,4-benzothiazin-4-yl)-N-(1,3-thiazol-2-ylmethyl)acetamide
(1R,2R,6S,7S)-4-(1-benzyl-1H-pyrazole-4-carbonyl)-4-azatricyclo[5.2.1.02,6]decane
2-[4-(2H-1,3-benzodioxol-5-yl)-2-[(3-methylpiperidin-1-yl)methyl]phenoxy]-N-[(3-fluorophenyl)methyl]acetamide
3-hydroxy-1-(3-phenylpropyl)-3-{[(propan-2-yl)amino]methyl}piperidin-2-one
2-(dimethylamino)-2-(3-fluorophenyl)-N-{2-[(3-methylpyridin-2-yl)amino]ethyl}acetamide
2-(4-butyl-2,3-dioxopiperazin-1-yl)-2-phenyl-N-(pyrimidin-4-ylmethyl)acetamide
2-{[1-(furan-2-ylmethyl)piperidin-4-yl]oxy}-4-methoxy-N-(2-methoxyethyl)benzamide
4-[2-(4-fluorophenyl)azetidine-1-carbonyl]-5-methyl-1-propyl-1H-pyrazole
N-{2-[7-(thiophen-3-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]ethyl}oxolane-2-carboxamide
1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]-2-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine
8-(8-fluoroquinoline-2-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
1-methyl-3-[3-(pyridin-4-yl)propyl]-8-(quinolin-6-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-(4-{2-[(1R,4R)-2-azabicyclo[2.2.1]heptan-2-yl]acetamido}-2-methoxyphenyl)-3-methylbutanamide
[(3R,4R)-1-{[4-methoxy-2-methyl-5-(propan-2-yl)phenyl]methyl}-4-(piperidin-1-ylmethyl)pyrrolidin-3-yl]methanol
N-[2-(4-ethoxyphenyl)ethyl]-2,8-diazaspiro[4.5]decane-3-carboxamide
(4aR,8aR)-1-[(1R,2R,4R)-bicyclo[2.2.1]hept-5-ene-2-carbonyl]-6-(propane-2-sulfonyl)-decahydro-1,6-naphthyridine
1-{1-[1-(methylsulfanyl)propan-2-yl]piperidin-4-yl}-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
dimethyl[(4-{1-[2-(methylsulfanyl)pyrimidine-5-carbonyl]piperidin-2-yl}phenyl)methyl]amine
[(3-chloropyridin-4-yl)methyl](methyl)(quinolin-6-ylmethyl)amine
N-benzyl-1-(2-hydroxyethyl)-5-(quinoxalin-5-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
{[2-cyclopropylmethanesulfonyl-1-(oxolan-2-ylmethyl)-1H-imidazol-5-yl]methyl}(methyl)[(5-methylfuran-2-yl)methyl]amine
1-[1,3-dioxo-2-(thiophen-2-ylmethyl)-2,3-dihydro-1H-isoindol-4-yl]-N-methyl-N-(1,3-thiazol-4-ylmethyl)piperidine-4-carboxamide
3,4-dimethoxy-N-methyl-N-[1-(3-phenylpropyl)piperidin-3-yl]benzamide
N-methyl-N-(1,2-oxazol-3-ylmethyl)-5-[3-(3-phenylpropyl)-1,2,4-oxadiazol-5-yl]pyridin-2-amine
N-[(2E)-3-phenylprop-2-en-1-yl]-N-propyl-2-(pyrrolidin-1-ylmethyl)-1,3-thiazole-5-carboxamide
4-(pyrimidin-5-yl)-2-({1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}methyl)phenol
N,2-dimethyl-N-{1-[1-(5-methyl-1H-indole-2-carbonyl)piperidin-4-yl]-2-phenylethyl}furan-3-carboxamide
(2S,4S)-4-amino-1-(2,3-dimethyl-1H-indole-7-carbonyl)-N,N-diethylpyrrolidine-2-carboxamide
4-[(2-hydroxy-4-methylquinolin-6-yl)sulfonyl]piperazine-2-carboxylic acid