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3-[5-({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)-1,2,4-oxadiazol-3-yl]pyridazine
ethyl({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]amine
2-{[6-ethyl-2-(piperidin-1-yl)pyrimidin-4-yl]amino}acetamide
4-{[(1R,9aR)-1-hydroxy-octahydro-1H-quinolizin-1-yl]methyl}piperazin-2-one
N-[1-(azepan-1-yl)-2-methylpropan-2-yl]-2-chloro-5-(1H-pyrazol-1-yl)benzamide
4-{4-[(4-methanesulfonylphenyl)methyl]piperazin-1-yl}quinoline
1-{[3-(3-fluorophenyl)oxolan-3-yl]methyl}-4-[2-(1H-imidazol-1-yl)ethyl]piperazine
N-(cyclohexylmethyl)-2-{1-[(2-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
2-(dimethylamino)-N-(3-methoxypropyl)-6-(2-methylphenyl)-N-(1-methylpiperidin-4-yl)pyridine-3-carboxamide
5-[4-(adamantan-1-yl)piperazine-1-carbonyl]-4-methyl-1,3-thiazol-2-amine
1-[(3-fluorophenyl)methyl]-4-[5-(1H-imidazol-1-ylmethyl)pyridin-2-yl]piperazin-2-one
4,6-dimethyl-3-[4-(3-methylpyridin-4-yl)-1,4-diazepane-1-carbonyl]-1,2-dihydropyridin-2-one
1-{2-[2-(2-methyl-2,3-dihydro-1-benzofuran-5-yl)-1H-imidazol-1-yl]ethyl}imidazolidin-2-one
1-(2-methanesulfonylethyl)-4-[(4-methoxy-2,3,6-trimethylphenyl)methyl]piperazine
2,4-dimethyl-N-[4-(4-{[(2-phenyl-2H-1,2,3-triazol-4-yl)methyl]amino}piperidin-1-yl)phenyl]benzamide
(1S,5R)-6-[1-methyl-3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonane
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propan-1-one
5-methyl-1-(4-methylphenyl)-4-(3-phenyl-1,2-oxazole-5-carbonyl)piperazin-2-one
[(3R,4R)-4-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]methyl}-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)pyrrolidin-3-yl]methanol
1-[9-(1,3-dimethyl-1H-pyrazole-4-carbonyl)-1-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]ethan-1-one
5-(furan-2-yl)-3-[1-(pyridin-3-yl)propan-2-yl]-3H,4H-thieno[2,3-d]pyrimidin-4-one
3-benzyl-5-(prop-2-en-1-yl)-1H-1,2,4-triazole
(2R,3S,6R)-3-(3-methoxyphenyl)-5-(4-methyl-1,2,5-oxadiazole-3-carbonyl)-1,5-diazatricyclo[5.2.2.02,6]undecane
1-methyl-5-[4-(1H-pyrazol-3-yl)piperidine-1-carbonyl]-1,2,3,4-tetrahydropyrimidine-2,4-dione
N-(furan-2-ylmethyl)-6-oxo-N-(prop-2-yn-1-yl)-1-[2-(pyridin-2-yl)ethyl]piperidine-3-carboxamide
3-methyl-N-[2-(5-methyl-4-phenyl-1H-imidazol-1-yl)ethyl]pyridin-2-amine
2-[(1S,5R)-3-(4-fluoro-2-methylbenzoyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-6-yl]-N,N-dimethylacetamide
4-(2-{[3-(piperidine-1-carbonyl)-1-propyl-4,5,6,7-tetrahydro-1H-indazol-5-yl]amino}ethyl)benzene-1-sulfonamide
N-cyclohexyl-2-{1-[(4-methoxy-3-methylphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
methyl 4-{[5-(2-chloro-4-methoxyphenoxymethyl)-1,2-oxazol-3-yl]formamido}butanoate
1-[1-(1,3-benzoxazol-2-yl)piperidin-4-yl]-N-ethylpiperidine-4-carboxamide
2-[3-({cyclopropyl[(4-methoxyphenyl)methyl]amino}methyl)phenyl]-6-methyl-3,4-dihydropyrimidin-4-one
(2R,3S,6R)-3-phenyl-5-[(1-propyl-1H-imidazol-2-yl)methyl]-1,5-diazatricyclo[5.2.2.02,6]undecane
(2S,4R)-4-amino-1-(3,4-dimethylbenzoyl)-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[4-(benzyloxy)piperidin-1-yl]-4,4,4-trifluorobutan-1-one
8-[2-(difluoromethoxy)benzoyl]-1-methyl-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
1-ethyl-N-[2-(4-methyl-1H-imidazol-2-yl)ethyl]-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
3-{[(2S,4R)-4-amino-2-[(propan-2-yl)carbamoyl]pyrrolidin-1-yl]methyl}-5-methyl-1H-indole-2-carboxylic acid
2-(3-methoxypropyl)-9-(1-methyl-1H-indole-3-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl (2S)-1-{5-[(cyclohexylmethyl)carbamoyl]-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carbonyl}pyrrolidine-2-carboxylate
1-({[3-(4-cyclohexylphenyl)-1-methyl-1H-pyrazol-4-yl]methyl}(methyl)amino)propan-2-ol
2-{4-[(3,5-dichloropyridin-4-yl)methyl]piperazin-1-yl}pyridine-3-carbonitrile
N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]thian-4-amine
2-({4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-6-methylpyridine
2-methyl-5-(4-{[2-methyl-4-(1H-pyrazol-1-yl)phenyl]methyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
3,5-dichloro-4-{[3-(piperidin-1-yl)azetidin-1-yl]methyl}pyridine
3-(4-hydroxyphenyl)-4-[(3-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
[(4-phenyloxan-4-yl)methyl]({[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl})amine
(1S,5R)-3-benzoyl-6-(5-ethylthiophene-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
3-[(3S,4R)-4-(dimethylamino)-1-(naphthalen-2-ylmethyl)piperidin-3-yl]-1-[4-(4-fluorophenyl)piperazin-1-yl]propan-1-one