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9-[(3-hydroxyphenyl)methyl]-6-(4-methoxyphenyl)-6,9-diazaspiro[4.5]decan-7-one
8-{[3-(1H-pyrazol-1-ylmethyl)phenyl]methyl}-1,3-dioxa-8-azaspiro[4.5]decan-2-one
2-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-2-(furan-3-yl)acetic acid
5-fluoro-2-[1-({3-methylimidazo[1,5-a]pyridin-1-yl}methyl)piperidin-4-yl]-1H-1,3-benzodiazole
[2-(4-methoxyphenyl)ethyl][(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl][(1-methylpiperidin-4-yl)methyl]amine
6-cyclopentyl-2-methoxy-3-{[(1-methoxypropan-2-yl)amino]methyl}-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
methyl (2S)-1-{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidine-2-carboxylate
4-{4-[(4aR,8aR)-octahydro-2H-1,4-benzoxazine-4-carbonyl]phenyl}-2-methylbutan-2-ol
5-(2-chloro-4-methoxyphenoxymethyl)-N-(1,3-dihydroxypropan-2-yl)-1H-pyrazole-3-carboxamide
1-[(2R,3R)-2-hydroxy-3-(thiomorpholin-4-yl)-2,3-dihydrospiro[indene-1,4'-piperidine]-1'-yl]propan-2-one
1-(2-fluorophenyl)-4-[(4-{[1-(furan-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]piperazine
2-cyclobutyl-N-[(3R,4S)-1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propyl]-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
[(2-fluoro-5-methoxyphenyl)methyl][(1-methylpiperidin-3-yl)methyl](2-phenylethyl)amine
2,8-dimethyl-4-(2-phenylazetidine-1-carbonyl)quinoline
3-[(3-methoxyphenyl)methyl]-1-(3-methylbutyl)-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
8-(1-methyl-5-phenyl-1H-pyrazole-3-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
N-[(3S,4R)-1-[(3-methyl-1-benzofuran-2-yl)methyl]-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
1-[(3,4-difluorophenyl)methyl]-3-hydroxy-3-({methyl[2-(1H-pyrazol-4-yl)ethyl]amino}methyl)piperidin-2-one
5-ethyl-4-({5-[(N-methylacetamido)methyl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)furan-2-carboxamide
4-(methoxymethyl)-6-[4-(pyridin-2-ylmethoxy)piperidin-1-yl]pyrimidine
2-(2-{[3-(4-chlorobenzoyl)piperidin-1-yl]methyl}-1H-pyrrol-1-yl)pyridine
2-(3-phenylpropyl)-N-{[3-(propan-2-yl)-1,2-oxazol-5-yl]methyl}-1,3-benzoxazole-5-carboxamide
1-(cyclopropylmethyl)-3-hydroxy-3-({[(2-methyl-1,3-thiazol-4-yl)methyl]amino}methyl)piperidin-2-one
{4-[(4-chlorophenyl)methyl]-1-[2-(1H-imidazol-2-yl)benzoyl]piperidin-4-yl}methanol
4-fluoro-N-({3-[2-(2-fluorophenyl)ethoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)benzamide
5-cyclopropanecarbonyl-1'-(2-ethylpyridine-4-carbonyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
3-(pyrrolidin-1-yl)-1-{[3-(trifluoromethyl)phenyl]methyl}pyrrolidine
3-[1-(1,3-dihydroxypropan-2-yl)piperidin-3-yl]propanamide
N-[4-(4-{[(2,3-dimethoxyphenyl)methyl]amino}piperidin-1-yl)phenyl]-2,4-dimethylbenzamide
N-(1-cycloheptylpiperidin-3-yl)-2-(2,6-difluorophenyl)acetamide
7-(5-methylthiophen-2-yl)-4-(oxolane-2-carbonyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
4-[4-(dimethylamino)azepane-1-carbonyl]benzene-1-sulfonamide
2-[2-(1H-imidazol-1-yl)ethyl]-1-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperidine
4-[(1-{[3-(propan-2-yl)-1H-pyrazol-5-yl]methyl}piperidin-2-yl)methyl]morpholine
2-methoxy-N-methyl-N-[(5-methylfuran-2-yl)methyl]-2-phenylacetamide
3-benzyl-7-[(2Z)-2-chloro-3-phenylprop-2-en-1-yl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine
3-[(3S,7S,8aS)-3-[(4-methoxyphenyl)methyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(naphthalen-1-yl)urea
N-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-(prop-2-yn-1-yl)cyclohexanamine
N-{4-chloro-1H-pyrrolo[2,3-b]pyridin-6-yl}-1-(pyridin-3-ylmethyl)piperidin-3-amine
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-[(2-methoxyphenyl)methyl]-N-[(3-methylphenyl)methyl]acetamide
N-[5-(2-phenylethyl)-1,3,4-thiadiazol-2-yl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
2,3-dimethyl-6-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]quinoxaline
2-(4-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidin-1-yl)pyridine-4-carbonitrile
N-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carboxamide
N-[2-(azepan-1-yl)ethyl]-3-hydroxy-N-(propan-2-yl)pyridine-2-carboxamide
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2,2-dimethyloxane-4-carboxamide
2-(dimethyl-1,2-oxazol-4-yl)-1-[1-(2-fluorophenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]ethan-1-one
N-[(1-ethyl-1H-pyrazol-4-yl)methyl]-8-fluoro-N-methylquinoline-2-carboxamide
N-[(3-benzyl-1,2,4-oxadiazol-5-yl)methyl]-3-(2-hydroxyphenyl)-1H-pyrazole-5-carboxamide
(3aS,6aS)-5-(6-methyl-2-propylpyrimidin-4-yl)-1-oxo-2-(prop-2-en-1-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid