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4-(3-hydroxy-3-methylbutyl)-N-[(3-hydroxyphenyl)methyl]-N-methylbenzamide
6-(2-chlorophenyl)-N-(1-methoxypropan-2-yl)-8-oxo-7-(prop-2-en-1-yl)-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
2-(2-hydroxyethyl)-N-(3-methyl-1,2,4-thiadiazol-5-yl)piperidine-1-carboxamide
(4aS,7aR)-1-(1H-imidazol-4-ylmethyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(4-methyl-4H-1,2,4-triazol-3-yl)ethyl]-5-oxo-1-[4-(propan-2-yl)phenyl]pyrrolidine-3-carboxamide
N-cyclopropyl-3-({[2-(3,5-dimethyl-1H-pyrazol-4-yl)ethyl](methyl)carbamoyl}amino)-4-methoxybenzamide
3-cyclopropyl-5-(3,6,7-trimethyl-1-benzofuran-2-carbonyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
(3R,4R)-4-(hydroxymethyl)-1-[5-(1H-imidazol-1-ylmethyl)furan-2-carbonyl]piperidin-3-ol
(2S,4S)-1-[(3-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-({[3-(trifluoromethyl)phenyl]methyl}amino)pyrrolidine-2-carboxamide
5-methyl-N-{2-[4-methyl-6-(trifluoromethyl)pyrimidin-2-yl]ethyl}-1-propyl-1H-pyrazole-4-carboxamide
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(3-methylphenyl)ethan-1-one
1-{4-[(4-butyl-1H-1,2,3-triazol-1-yl)methyl]piperidin-1-yl}ethan-1-one
1-cyclohexyl-N-(1H-imidazol-2-ylmethyl)-N-methylpiperidine-4-carboxamide
N-{2-[1-(furan-2-ylmethyl)piperidin-3-yl]ethyl}-2-oxo-2-(pyrrolidin-1-yl)acetamide
N-[3-(5-amino-1,3,4-thiadiazol-2-yl)propyl]-5-methyl-4,5,6,7-tetrahydro-1-benzothiophene-2-carboxamide
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)acetamide
2-cyclopropanecarbonyl-N-methyl-N-(1,3-thiazol-2-ylmethyl)-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
2-[(2,6-dichlorophenyl)methyl]-5-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl}pyrimidin-4-ol
N-{4-methyl-2-[2-(5-methyl-3-oxo-2,3-dihydro-1H-pyrazol-4-yl)acetamido]phenyl}cyclohexanecarboxamide
1-{2-[(oxan-4-ylmethyl)amino]pyrimidin-4-yl}piperidin-3-ol
N-[1-(3,5-difluorophenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-3-hydroxypropanamide
3-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-8-{[4-(furan-2-yl)phenyl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
6-{1-[2-(2,3-dihydro-1H-inden-1-yl)acetyl]piperidin-4-yl}-3,4-dihydropyrimidin-4-one
2-({4-[5-(1H-imidazol-1-ylmethyl)-4-methyl-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)benzonitrile
N-[(3S,4R)-1-{2-[(2-methoxyethyl)(methyl)amino]acetyl}-4-(4-methylphenyl)pyrrolidin-3-yl]cyclopropanecarboxamide
4-[3-(1H-1,3-benzodiazol-2-ylmethyl)piperidin-1-yl]-6-methylpyrimidin-2-amine
2-(2-hydroxyphenyl)-1-{4-[1-(pyridin-3-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
N-methyl-N-[(3-phenyl-1,2-oxazol-5-yl)methyl]-4-(thiophen-2-yl)butanamide
1-[4-(3-hydroxypiperidin-1-yl)piperidin-1-yl]-2-[methyl(phenyl)amino]ethan-1-one
N-cyclopentyl-3-{[2-(1,3-thiazol-2-yl)ethyl]sulfamoyl}benzamide
N-{[1-(3-methoxypropyl)pyrrolidin-3-yl]methyl}-5,7-dimethylpyrido[2,3-d]pyrimidin-4-amine
1-(3-{1-[2-(dimethylamino)ethyl]-1H-imidazol-2-yl}piperidin-1-yl)-2-(2-methyl-1,3-thiazol-4-yl)ethan-1-one
3-(1-{2-[4-hydroxy-3-methoxy-5-(prop-2-en-1-yl)phenyl]-1H-imidazol-1-yl}ethyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[1-(hydroxymethyl)cyclopentyl]-2-[3-oxo-1-(thiophen-2-ylmethyl)piperazin-2-yl]acetamide
1-[1-(cyclohex-1-en-1-yl)ethyl]-3-[3-(2-oxo-1,3-oxazolidin-3-yl)phenyl]urea
(2S,4S)-4-{[(2,4-difluorophenyl)methyl]amino}-N-ethyl-1-(2-methylpropyl)pyrrolidine-2-carboxamide
(3R,4R)-4-(2-methoxyethyl)-3-methyl-1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]piperidin-4-ol
5-[4-(2-phenylethyl)piperidine-1-carbonyl]-N-(piperidin-3-yl)pyridin-2-amine
3-{2-[(4-methoxyphenyl)methyl]morpholine-4-carbonyl}-4,5,6,7-tetrahydro-1,2-benzoxazole
2-(3,4-dimethoxyphenyl)-1-{3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
methyl 1-{3-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]benzoyl}piperidine-2-carboxylate
2-[2-(5-ethylpyridin-2-yl)-1H-imidazol-1-yl]-N-methylethane-1-sulfonamide
2-{2-[3-(4-fluorophenyl)pyrrolidin-1-yl]-2-oxoethyl}-4-methyl-1,2-dihydrophthalazin-1-one
5-(1-ethyl-1H-1,2,4-triazol-5-yl)-1H,5H,6H,7H,8H-pyrido[3,2-f]indazol-7-one
4-(2-ethyl-4-methyl-1,3-thiazole-5-carbonyl)-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-[(3S,4R)-4-amino-1-(6-ethyl-2-methylquinoline-4-carbonyl)pyrrolidin-3-yl]ethan-1-ol
3-[methyl({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)amino]propane-1,2-diol
{[3-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]methyl}({1-[1-(4-methoxyphenyl)-5-methyl-1H-pyrazol-4-yl]ethyl})amine
1-{2-[4-(2-amino-1,3-thiazol-4-yl)phenyl]-4-fluorophenyl}ethan-1-one
2-[1-(2,2-diphenylethyl)-3-oxopiperazin-2-yl]-N-[(5-methylfuran-2-yl)methyl]acetamide