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3-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}-N-[(2-fluorophenyl)methyl]propanamide
1-{5H,6H-benzo[h]quinazolin-2-yl}-5-methyl-N,N-bis(prop-2-en-1-yl)-1H-pyrazole-4-carboxamide
6-{4-[(2R,6S)-2,6-dimethylmorpholin-4-yl]piperidin-1-yl}-N-(2-methoxyethyl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}acetamide
1-(3-cyano-4-methylphenyl)-3-[2-(2-methylpropanesulfonyl)ethyl]urea
5-{7-[(3,4-difluorophenyl)methyl]-2,7-diazaspiro[4.5]decane-2-carbonyl}pyridin-2-ol
N-ethyl-2-(4-fluorophenoxymethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-1,3-oxazole-4-carboxamide
N-[2-methoxy-1-(pyridin-2-yl)ethyl]-N-methyl-2-(1-methylpiperidin-4-yl)acetamide
5-{[(2,1,3-benzothiadiazol-5-ylmethyl)(methyl)amino]methyl}-N-(oxolan-2-ylmethyl)pyrimidin-2-amine
5-{[3-(1,2-dihydroacenaphthylene-5-carbonyl)piperidin-1-yl]methyl}-2-(methylsulfanyl)pyrimidine
4-{6-[(pyridin-3-ylmethyl)amino]-1H-pyrrolo[2,3-b]pyridin-4-yl}thiophene-2-carboxamide
N-[1-(5-propyl-1,2-oxazole-3-carbonyl)pyrrolidin-3-yl]acetamide
2-[3-(hydroxymethyl)-3-(2-phenylethyl)piperidin-1-yl]pyridine-3-carboxamide
methyl 2-{[5-(4-fluorophenyl)-4-[1-(2-phenoxyacetyl)piperidin-3-yl]pyrimidin-2-yl]sulfanyl}acetate
N-{2-[4-(acetamidomethyl)-1,2,3,6-tetrahydropyridin-1-yl]ethyl}benzamide
N-[(3,4-difluorophenyl)methyl]-4-[5-(morpholin-4-ylmethyl)-1H-1,2,3,4-tetrazol-1-yl]butanamide
8-[5-(morpholin-4-ylmethyl)furan-3-carbonyl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
N-ethyl-4-(hydroxymethyl)-N-[2-(1H-pyrazol-1-yl)ethyl]pyridine-2-carboxamide
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carbonyl}-10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocine
methyl 6-(but-3-enoyl)-2-[(3,5-dimethylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-ethyl-1-(1-ethyl-4,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carbonyl)piperidine-3-carboxylic acid
2-[3-(5-methoxy-1-benzofuran-3-yl)-1H-pyrazol-1-yl]-N-(2-methyl-2H-1,2,3-triazol-4-yl)acetamide
N-methyl-4-oxo-N-{[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]methyl}-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-(1H-pyrrole-2-carbonyl)-3-{2-[2-(trifluoromethyl)phenyl]ethyl}piperidine
N-[(1R,3R)-3-aminocyclopentyl]-2,4-dioxo-1,2,3,4-tetrahydropyrimidine-5-sulfonamide
5-{[5-(2-methoxyacetyl)-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl]carbonyl}-3,4-dihydropyrimidin-4-one
4-[(1-acetylpiperidin-4-yl)amino]-1-(cyclohexylmethyl)pyrrolidin-2-one
1-(cyclohexylmethyl)-5-[4-(3-methoxypropyl)piperidine-1-carbonyl]piperidin-2-one
7-chloro-4-{2-methyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-yl}-2,3,4,5-tetrahydro-1,4-benzoxazepine
9-(3-chloro-2-methylbenzoyl)-2-(2-hydroxyethyl)-2,9-diazaspiro[5.5]undecan-3-one
(2S,4S)-N-ethyl-1-(3-methoxypropyl)-4-[2-(2-methylphenyl)acetamido]pyrrolidine-2-carboxamide
4-(2,4-difluorophenyl)-3-[(4-methoxyphenyl)methyl]-4H-1,2,4-triazole
4-(8-chloroquinoline-2-carbonyl)-1-phenylpiperazin-2-one
5-ethyl-N-[2-(3-methylpiperidin-1-yl)ethyl]pyrimidin-2-amine
(4aS,8aR)-1-propyl-6-(quinoxaline-6-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-methyl-6-{4-[4-(2-phenylethyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}-1H-1,3-benzodiazole
2-amino-4-(3-cyclohexyl-1H-pyrazol-4-yl)-5H,7H,8H-pyrano[4,3-b]pyridine-3-carbonitrile
7-(2-methoxypyridine-3-carbonyl)-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
N-{2-[(1-methyl-1H-imidazol-2-yl)sulfanyl]ethyl}-1-(oxan-4-yl)piperidine-3-carboxamide
3-{1-[(3-acetylphenyl)methyl]piperidin-4-yl}-N-[2-(dimethylamino)ethyl]propanamide
(2S,4S)-N-[2-(2H-1,3-benzodioxol-5-yl)ethyl]-1-benzyl-4-{[(2-chlorophenyl)methyl]amino}pyrrolidine-2-carboxamide
4-{5-[(dimethylamino)methyl]-4-methyl-4H-1,2,4-triazol-3-yl}-N-(4-fluorophenyl)piperidine-1-carboxamide
N-{[5-(2,6-difluorophenyl)-1,2,4-oxadiazol-3-yl]methyl}-4-(pyridin-3-yl)pyrimidin-2-amine
N,N,4-trimethyl-3-({[(propylcarbamoyl)methyl]carbamoyl}methyl)-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
3-(3,5-dimethyl-1H-pyrazol-4-yl)-1-[4-(2-phenylethyl)piperazin-1-yl]propan-1-one
1-[(2-fluorophenyl)methyl]-3-hydroxy-3-(thiomorpholin-4-ylmethyl)piperidin-2-one
1-(1-methyl-1H-pyrrole-2-carbonyl)-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
7-(3,5-dichloro-4-methoxybenzoyl)-5H,6H,7H,8H-imidazo[1,2-a]pyrazine-3-carboxamide
N-benzyl{[4-(2-methoxyphenoxy)phenyl]amino}sulfonamide
5-({methyl[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]amino}methyl)-N-(oxolan-2-ylmethyl)pyrimidin-2-amine