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1-[1-(6-methylpyridine-2-carbonyl)piperidin-3-yl]-2-phenylethan-1-one
1-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)-2-(pyrrolidin-1-ylmethyl)piperidine
2-{[(5-fluoro-2,3-dimethyl-1H-indol-7-yl)methyl]amino}pyridine-3-carboxamide
ethyl 1-{2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]ethyl}-1H-imidazole-2-carboxylate
2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]-N-({2-[(methylsulfanyl)methyl]-1,3-thiazol-4-yl}methyl)acetamide
2,6-dihydroxy-N-[2-(propylsulfanyl)ethyl]benzamide
N-[2-(1H-imidazol-4-yl)ethyl]-2-[(6-methyl-1H-1,3-benzodiazol-2-yl)methoxy]acetamide
3-(4-methyl-1H-pyrazol-1-yl)-1-{2-methyl-4-phenyl-2,9-diazaspiro[5.5]undecan-9-yl}propan-1-one
N-({2-[(dimethylamino)methyl]phenyl}methyl)-N,1,3-trimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
(3aS,6aS)-2-[2-(4-hydroxyphenyl)ethyl]-5-(oxan-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{5-[(2,5-dimethoxyphenyl)methyl]-1,3,4-oxadiazol-2-yl}-1-[2-(methoxymethyl)piperidin-1-yl]propan-1-one
3-[(4aR,7aS)-4-[(1-methyl-1H-imidazol-2-yl)methyl]-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]propanoic acid
N-{2-[2-(pyridin-3-yl)-1,3-thiazol-4-yl]ethyl}-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
N-cyclopropyl-2-fluoro-N-{[3-(oxolan-2-ylmethoxy)phenyl]methyl}benzamide
1-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-3-carbonyl}-4-(4-methoxyphenyl)-2-methylpiperazine
{7-methyl-2-[4-(2-phenoxyethyl)piperazin-1-yl]quinolin-3-yl}methanol
3-[1-(1H-1,3-benzodiazole-5-carbonyl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
2-methyl-5-[2-(1H-pyrazol-4-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-5-carbonyl]pyrazine
1-{4-[4-methyl-5-(1H-1,2,4-triazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-pyrazol-1-yl)propan-1-one
4-{4-[(1-phenyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}quinazoline
2-methyl-4-{4-[3-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine-1-carbonyl]phenyl}butan-2-ol
(1S,2R)-2-({[2-(furan-2-yl)phenyl]methyl}(methyl)amino)cyclohexan-1-ol
2-ethyl-N-(2-methylphenyl)-3-oxo-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-(2-methylphenyl)-3-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}formamido)propanamide
1-(1-{2-phenyl-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}piperidine-4-carbonyl)-1,4-diazepane
N-[(4-acetamidophenyl)methyl]-2-{[2-(1H-imidazol-4-yl)ethyl]amino}acetamide
1-{1-[(4,5-dimethylfuran-2-yl)methyl]piperidin-3-yl}-4-phenylpiperazine
1-(methoxymethyl)-N-{2-methyl-1,1-dioxo-2H,3H,4H-1λ6-thieno[2,3-e][1,2]thiazin-4-yl}cyclobutane-1-carboxamide
5-cyclopropyl-N-[2-methyl-4-(5-methyl-1,3-benzoxazol-2-yl)phenyl]-1,2-oxazole-4-carboxamide
1-methyl-4-{[8-methyl-2-(piperidine-1-carbonyl)imidazo[1,2-a]pyridin-3-yl]methyl}piperazine
N-(2H-1,3-benzodioxol-5-ylmethyl)-4-cyclobutaneamidobenzamide
1-[2-(dimethyl-1,3-thiazol-5-yl)acetyl]-4-methyl-1,4-diazepan-5-one
5-oxo-1-phenyl-N-[(4-phenyloxan-4-yl)methyl]-2,5-dihydro-1H-pyrazole-3-carboxamide
1-(4-acetylphenyl)-3-[3-methyl-1-(1-methyl-1H-1,2,4-triazol-5-yl)butyl]urea
(2S,4S)-4-amino-N,N-diethyl-1-(6-methyl-2-oxo-1,2-dihydropyridine-3-carbonyl)pyrrolidine-2-carboxamide
N-[(1-benzylpiperidin-3-yl)methyl]pyrimidin-4-amine
3-(3-fluorophenyl)-N-[(1-phenyl-1H-pyrazol-4-yl)methyl]-1H-pyrazole-4-carboxamide
7-hydroxy-6-methyl-4-[2-(2-methylphenyl)-1,3-thiazol-5-yl]-1,2,3,4-tetrahydroquinolin-2-one
6-(4-cyclohexylpiperazine-1-carbonyl)-3-ethyl-3H-imidazo[4,5-b]pyridin-2-amine
[1-(dimethyl-1,3-thiazol-4-yl)ethyl]({[4-methoxy-3-(1H-pyrazol-1-ylmethyl)phenyl]methyl})methylamine
3-ethyl-5-{3-[2-(oxolan-3-yl)-1H-imidazol-1-yl]phenyl}-1,2,4-oxadiazole
2-(cyclopropylmethyl)-9-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
3-(2-oxo-2-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}ethyl)-1,3-diazinane-2,4-dione
methyl 2-[4-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)piperidin-1-yl]acetate
3-({[1-(hydroxymethyl)cyclohexyl]carbamoyl}methyl)-N,N,4-trimethyl-3,4-dihydro-2H-1,4-benzoxazine-6-carboxamide
N-{2-[cyclopentyl(methyl)amino]ethyl}-N-methylquinoxaline-5-carboxamide
(2S,4R)-4-{[(9-ethyl-9H-carbazol-3-yl)methyl]amino}-N-(propan-2-yl)-1-(1-propylpiperidin-4-yl)pyrrolidine-2-carboxamide
1-(cyclohexylmethyl)-N-[(3,4-difluorophenyl)methyl]-6-oxopiperidine-3-carboxamide
N-(pyridin-3-ylmethyl)-4-[3-(4H-1,2,4-triazol-4-yl)phenyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
4-(5-chloro-2-ethoxy-4-methylbenzenesulfonyl)piperazine-2-carboxylic acid