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1-ethyl-3,5-dimethyl-N-[2-(4-phenylpiperidin-1-yl)ethyl]-1H-pyrazole-4-carboxamide
4-{[(1R,3S,3aS,6aR)-1-(hydroxymethyl)-3-(2-methoxypyridin-3-yl)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-1-yl]methyl}phenol
N-{1-[1-(5-fluoropyrimidin-2-yl)piperidin-4-yl]-1H-pyrazol-5-yl}-2-methylbenzamide
3-(1-methylpiperidin-3-yl)-1-[3-(pyridin-3-yl)azetidin-1-yl]propan-1-one
N-cyclopropyl-N-[(2-methoxyphenyl)methyl]-2-(phenylamino)pyrimidine-5-carboxamide
2-(4-{[4-(methylsulfanyl)phenyl]methyl}piperazin-1-yl)-1-(piperidin-1-yl)ethan-1-one
5-(1-cyclohexyl-3-methyl-1H-1,2,4-triazol-5-yl)-4-oxo-1-(propan-2-yl)-1,4-dihydropyridine-3-carboxylic acid
2-[4-(dimethylamino)phenyl]-1-[(3R,4R)-3-(hydroxymethyl)-4-[(4-methylpiperazin-1-yl)methyl]pyrrolidin-1-yl]ethan-1-one
4-({2-[4-(2,6-dimethylpyridin-3-yl)pyrimidin-2-yl]phenyl}methyl)morpholine
6-{3-[(3,4-difluorophenyl)amino]piperidine-1-carbonyl}-2-methyl-2,3,4,5-tetrahydropyridazin-3-one
5-[4-(azonane-1-carbonyl)quinolin-2-yl]pyrimidin-2-amine
5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-(thiophen-2-ylmethyl)-1,2-oxazole-3-carboxamide
methyl 3-(furan-3-amido)-5-{[(2E)-2-methylbut-2-en-1-yl]amino}-1-(2-methylpropyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
N-[(2R,3R)-2-methoxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-1,3-dimethyl-1H-pyrazole-4-carboxamide
6-methoxy-N-(5-{[({8-methylimidazo[1,2-a]pyridin-3-yl}methyl)amino]methyl}-1,3-thiazol-2-yl)pyridin-3-amine
1-[4-(2H-1,3-benzodioxol-5-yl)pyrimidin-2-yl]-N-benzyl-5-cyclopropyl-1H-pyrazole-4-carboxamide
N3-(3-{[(2-fluorophenyl)methyl]sulfanyl}propyl)piperidine-1,3-dicarboxamide
N-cyclopropyl-1-{1-[(2,4,5-trimethylphenyl)methyl]piperidin-4-yl}piperidine-3-carboxamide
1-(4-chlorophenyl)-N-{[(3S,4S)-3-hydroxypiperidin-4-yl]methyl}cyclohexane-1-carboxamide
2-{[4-(2-chlorophenyl)-5-[1-(1H-imidazol-1-yl)ethyl]-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
7-methyl-N-[2-(4-sulfamoylphenyl)ethyl]pyrazolo[1,5-a]pyrimidine-6-carboxamide
3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}propanamide
2-(1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}piperidin-2-yl)-5-fluoro-1H-1,3-benzodiazole
N-[(5-{[6-(dimethylamino)pyridin-3-yl]methyl}-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl)methyl]-2-methoxyacetamide
(3aS,6aS)-2-(dimethylcarbamoyl)-5-[(4-hydroxy-5-methoxypyridin-2-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-(4-{[(adamantan-2-ylmethyl)amino]methyl}phenoxy)-3-(4-methylpiperazin-1-yl)propan-2-ol
9-hydroxy-4-oxo-N-[2-(pyridin-2-yl)ethyl]-4H-pyrido[1,2-a]pyrimidine-3-carboxamide
1-(2-methoxyphenyl)-2,2-dimethyl-4-(pyridine-2-carbonyl)piperazine
4-{[1-(1-cyclopentylpiperidine-3-carbonyl)azetidin-3-yl]oxy}benzoic acid
5-(morpholin-4-ylmethyl)-N-[5-oxo-1-(propan-2-yl)pyrrolidin-3-yl]-1,2-oxazole-3-carboxamide
(2S,4R)-4-amino-1-[2-(azocan-1-yl)acetyl]-N-ethylpyrrolidine-2-carboxamide
3-{1-[4-(1H-imidazol-1-yl)benzoyl]piperidin-2-yl}pyridine
1-(1-cyclopropanecarbonylpiperidin-4-yl)-N-[2-(5-methylfuran-2-yl)ethyl]piperidine-3-carboxamide
3-{1-[(3-acetylphenyl)methyl]piperidin-3-yl}-N-[(5-methylfuran-2-yl)methyl]propanamide
1-{3-[(dimethylamino)methyl]-3-hydroxypyrrolidin-1-yl}-3-(1H-indol-3-yl)propan-1-one
8-(3-methoxypyrazin-2-yl)-2-(pyridin-4-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
(4aR,7aS)-1-(2-{2H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}pyrimidin-4-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
2-{[(4aS,7aR)-4-(2-methylpropyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]sulfonyl}benzonitrile
4-(2-{1-[4-(trifluoromethyl)benzoyl]piperidin-2-yl}ethyl)morpholine
4-{8-thia-4,6,11-triazatricyclo[7.4.0.02,7]trideca-1(9),2,4,6-tetraen-3-yl}piperazine-1-carboxamide
3-[1-(cyclohex-3-en-1-ylmethyl)-1H-pyrazol-5-yl]-1-[2-(4,6-dimethyl-2-oxo-1,2-dihydropyrimidin-1-yl)ethyl]urea
7-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-3-methyl-3,4-dihydroquinazolin-4-one
2-[1-cyclopentyl-4-({5-[(4-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]furan-2-yl}methyl)piperazin-2-yl]ethan-1-ol
8-(4-methyl-1H-imidazole-2-carbonyl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-{4-[(1-propyl-1H-imidazol-2-yl)methyl]morpholin-2-yl}ethan-1-amine
7-(1H-imidazol-2-ylmethyl)-N-[2-(3-methyl-1H-pyrazol-1-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-(2-methyl-1-{4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-1-oxopropan-2-yl)acetamide
3-[(3R,7S,8aS)-3-methyl-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-(5-fluoro-2-methylphenyl)urea
N-(2-methoxypropyl)-3-{[3-(piperidin-1-yl)azetidin-1-yl]sulfonyl}benzamide
(5-{1-[(2-ethyl-1,3-thiazol-4-yl)methyl]-4-phenyl-1H-imidazol-5-yl}furan-2-yl)methanol