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2-(2-hydroxyethyl)-9-[2-(3-methylphenyl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
N-{[2-(2-methoxyphenoxy)pyridin-3-yl]methyl}-1H-pyrrole-2-carboxamide
2-[(methylsulfanyl)methyl]-4-[(2-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}-1H-imidazol-1-yl)methyl]-1,3-thiazole
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-[2-(1H-pyrazol-1-yl)acetyl]-decahydro-1,6-naphthyridin-2-one
3-methoxy-N-(4-methyl-3-propanamidophenyl)pyrrolidine-1-carboxamide
2-cyclopentyl-9-[2-(2-oxo-1,2-dihydropyrimidin-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
6-ethyl-N-[(4-methoxyphenyl)(pyridin-4-yl)methyl]pyrimidin-4-amine
[(3-tert-butyl-1H-pyrazol-5-yl)methyl](methyl)(3,3,3-trifluoropropyl)amine
1-{2-[3-(propan-2-yl)-1-(pyridin-2-yl)-1H-1,2,4-triazol-5-yl]phenyl}-1,3-diazinane-2,4-dione
2,3,5-trimethyl-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}pyrazolo[1,5-a]pyrimidin-7-amine
3-[5-(2-hydroxypyridin-3-yl)-3-(2-methyl-1,3-thiazol-4-yl)-1H-1,2,4-triazol-1-yl]-1λ6-thiolane-1,1-dione
N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4-(pyrrolidin-1-ylmethyl)benzamide
(2S,4S)-N,N-diethyl-1-[(4-fluoro-2-methylphenyl)methyl]-4-(2-hydroxyacetamido)pyrrolidine-2-carboxamide
1-(3-acetylphenyl)-3-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-(2-methoxyethyl)urea
N-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-5-propyl-1,2-oxazole-3-carboxamide
N-[5-(2-fluorophenyl)-4H-1,2,4-triazol-3-yl]-1,2,3,4-tetrahydroisoquinoline-2-carboxamide
N-[3-(5-chloro-1H-1,3-benzodiazol-2-yl)propyl]-3-methyl-[1,2]oxazolo[5,4-d]pyrimidin-4-amine
{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}[(3-methoxyphenyl)methyl]methylamine
2-[(2-propyl-1,3-thiazol-4-yl)formamido]-N-(2,3,4-trifluorophenyl)acetamide
2-(6-aminopyridin-3-yl)-2-[4-(2-phenoxyethyl)piperazin-1-yl]acetic acid
5-(1-ethyl-1H-pyrazole-4-carbonyl)-N-(3-phenylpropyl)-1-(pyridin-4-ylmethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
6-cyano-N-{[2-(2,4-difluorophenoxy)pyridin-3-yl]methyl}pyridine-3-carboxamide
methyl 6-cyclobutanecarbonyl-2-[(2,3-dimethylphenyl)sulfamoyl]-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
4-(butan-2-yl)-3-[(4-methoxyphenyl)methyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
1-[5-(oxolan-2-yl)thiophene-2-amido]cyclopentane-1-carboxylic acid
5-chloro-N-[(trimethylpyrazin-2-yl)methyl]pyridin-2-amine
N-[(2-ethoxy-3-methoxyphenyl)methyl]-N,2-dimethyl-2,8-diazaspiro[4.5]decane-3-carboxamide
4-[5-(methoxymethyl)furan-2-carbonyl]-6-[(3-methoxyphenyl)methoxy]-1-(pyridin-2-ylmethyl)-1,4-diazepan-2-one
1-[(2-phenyl-1,3-thiazol-5-yl)methyl]-3-(pyrrolidin-1-ylmethyl)piperidin-3-ol
methyl 5-(4-methanesulfonylbenzoyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxylate
2-{1-[(2-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-[2-(methylsulfanyl)ethyl]acetamide
1-[1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidin-3-yl]pyrrolidin-2-one
1-{3-[(1S,5R)-3-(2,3-dihydro-1H-inden-2-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-oxopropyl}pyrrolidin-2-one
2-(2-amino-4,6-dimethylpyrimidin-5-yl)-N-[(2,3,5-trimethyl-1H-indol-7-yl)methyl]acetamide
N-methyl-3-(6-oxo-1,6-dihydropyridazin-3-yl)-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]propanamide
2-[(1-acetylpiperidin-4-yl)oxy]-5-chloro-N-(1H-1,2,3,4-tetrazol-5-ylmethyl)benzamide
N-[3-(3-ethylphenoxy)propyl]-3-hydroxy-N-methylpropanamide
3-(4-fluoro-3-methylphenyl)-6-(oxolane-2-carbonyl)-1-(pyridin-3-ylmethyl)-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
N-methyl-N-[(1-{2-[3-(trifluoromethyl)phenyl]ethyl}piperidin-3-yl)methyl]-1H-imidazole-2-carboxamide
N-(prop-2-en-1-yl)-N-(pyridin-2-ylmethyl)-2-(pyridin-3-yl)acetamide
3-[1-methyl-3-(pyridin-3-yl)-1H-pyrazol-5-yl]-1-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}urea
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)methanesulfonamide
2-(4-{[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}piperazin-1-yl)pyrazine
2-(dimethylamino)-2-(3-methylphenyl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}acetamide
4-[2-(1-{3-fluoro-6-methylimidazo[1,2-a]pyridine-2-carbonyl}piperidin-2-yl)ethyl]morpholine
N-[2-(dimethylamino)ethyl]-3-{1-[(1-methyl-3-phenyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}propanamide
1-(2-hydroxyethyl)-5-(2-methoxy-4-methylbenzoyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylic acid
(1S,5R)-N-benzyl-6-(cyclobutylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonane-3-carboxamide
1-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-2-[4-(hydroxymethyl)phenyl]ethan-1-one
(1R,5R)-6-(2-methoxyethyl)-3-{7-methylthieno[3,2-d]pyrimidin-4-yl}-3,6-diazabicyclo[3.2.2]nonane