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2-[(3R,4R)-3-({[2-(dimethylamino)ethyl](methyl)amino}methyl)-4-(hydroxymethyl)pyrrolidine-1-carbonyl]-5-methylphenol
N-(2-methoxyethyl)-N-[(4-methylphenyl)methyl]-1-(pyrimidin-2-yl)piperidine-4-carboxamide
N-[3-(5-methyl-2H-1,2,3,4-tetrazol-2-yl)adamantan-1-yl]pyrazin-2-amine
2-(adamantan-1-yl)-N-[(2-chloropyridin-3-yl)methyl]-N-methylacetamide
1-(methoxymethyl)-N-{3-[methyl(phenyl)amino]propyl}cyclopropane-1-carboxamide
[4-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-1,4-oxazepan-6-yl]methanol
4-(hydroxymethyl)-1-{[5-(1H-pyrazol-3-yl)thiophen-2-yl]methyl}azepan-4-ol
1-cyclopentyl-N-[2-(4-fluorobenzenesulfonyl)ethyl]-5-oxopyrrolidine-3-carboxamide
N-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]-2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-amine
6-{3-[1-(pyrrolidin-1-yl)ethyl]phenyl}-2H-1,3-benzodioxole-5-carboxamide
N,N-diethyl-1-[1-(furan-3-ylmethyl)piperidin-3-yl]-1H-1,2,3-triazole-4-carboxamide
2-amino-4-(3-fluoro-2-methylphenyl)-6-(oxolane-2-carbonyl)-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
2-({methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]amino}methyl)quinolin-8-ol
3-methoxy-1-[3-(2-methoxyphenoxy)propyl]-1,2-dihydropyridin-2-one
2-(2-hydroxypropyl)-9-(1-methyl-1H-pyrazole-4-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
1-[2-(2-methoxyphenyl)ethyl]-2,6-dimethyl-4-oxo-N-[1-(thiophen-2-yl)propyl]-1,4-dihydropyridine-3-carboxamide
N-(2-methoxyethyl)-5-(methoxymethyl)-1-[4-(2-methoxyphenyl)pyrimidin-2-yl]-N-(propan-2-yl)-1H-pyrazole-4-carboxamide
N-(1-phenylbutyl)-5-(pyrrolidin-1-ylmethyl)furan-2-carboxamide
5-(2-chlorophenyl)-N-[cyclopropyl(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]furan-2-carboxamide
N-[2-hydroxy-2-(pyridin-3-yl)ethyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
3-(5-fluoro-1H-1,3-benzodiazol-2-yl)-1-(2-methylpyrrolidin-1-yl)propan-1-one
N-{2-[4-(2H-1,3-benzodioxol-5-ylmethyl)-3-oxopiperazin-1-yl]-2-oxoethyl}acetamide
(1R,5R)-6-{[4-(1H-imidazol-1-yl)phenyl]methyl}-3-(pyrimidin-2-yl)-3,6-diazabicyclo[3.2.2]nonane
1-ethyl-4-{2-[4-(methoxymethyl)piperidine-1-carbonyl]-2,3-dihydro-1H-inden-2-yl}piperazine
2-(1-benzyl-2-methyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(propan-2-yl)acetamide
N-(2-hydroxyethyl)-N-[(1-methyl-1H-imidazol-2-yl)methyl]-3-(2-methyl-1H-indol-1-yl)propanamide
4-chloro-N-[2-({5-methylpyrazolo[1,5-a]pyrimidin-7-yl}amino)ethyl]benzene-1-sulfonamide
3-(2-oxoazepan-1-yl)-N-[(2-phenoxypyridin-3-yl)methyl]propanamide
methyl 3-[7-(1,3-benzothiazol-2-yl)-9-hydroxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]propanoate
4-{5,7-dimethylpyrazolo[1,5-a]pyrimidine-2-carbonyl}-6-(pyrrolidin-1-ylmethyl)-1,4-oxazepan-6-ol
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-{[1-(pyridin-4-yl)-1H-pyrrol-2-yl]methyl}piperidin-3-ol
(4S)-1-[(4-methoxypyridin-2-yl)methyl]-3,3,4-trimethylpiperidin-4-ol
2-{2,7-diazaspiro[4.5]decane-7-sulfonyl}benzonitrile
1-(diethylsulfamoyl)-4-(4-methyl-1H-pyrazol-1-yl)piperidine-4-carboxylic acid
8-chloro-2-{4-[1-(morpholin-4-yl)ethyl]piperidin-1-yl}quinoline
2-methyl-5-{2-[(3E)-4-methylhex-3-en-1-yl]phenyl}-1,3,4-oxadiazole
3-[2-(morpholin-4-ylmethyl)piperidine-1-carbonyl]-4H-pyrido[1,2-a]pyrimidin-4-one
methyl 4-methoxy-3-({4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carbonyl}amino)benzoate
{[2-(2,4-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
4-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2,2-dimethylmorpholine
3-(4-phenyl-1H-pyrazol-5-yl)-1-[4-(propan-2-yl)-1,2,3-thiadiazole-5-carbonyl]piperidine
1-[3-(furan-2-yl)benzoyl]-4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine
N-({4-[(3-fluorophenyl)methoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)thiophene-2-sulfonamide
(3S)-1-(2-{[(2E)-3-phenylprop-2-en-1-yl]sulfanyl}pyridine-3-carbonyl)pyrrolidin-3-ol
1-{1-[(5-methylfuran-2-yl)methyl]piperidin-4-yl}-N-(2-phenylethyl)piperidine-4-carboxamide
1-(2-fluorophenyl)-4-{1-[1-(pyridin-2-ylmethyl)piperidin-4-yl]piperidin-3-yl}piperazine
N-{2-[ethyl(methyl)amino]ethyl}-3-{[(2S)-2-(hydroxymethyl)pyrrolidin-1-yl]sulfonyl}-N-methylbenzamide
4-{1-[(2-phenyl-1,3-thiazol-5-yl)methyl]piperidin-4-yl}pyridine
3-{[(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)(methyl)amino]methyl}pyridin-2-ol
N-methyl-5-(2-methylphenyl)-N-[(1-methylpiperidin-4-yl)methyl]-1,2,4-triazin-3-amine