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2-{octahydropyrrolo[1,2-a]piperazin-2-ylmethyl}-1H-1,3-benzodiazole
3-(5-{[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]methyl}-1,2-oxazol-3-yl)pyridine
1-[2-(methylamino)pyridine-3-carbonyl]-4-(5-methylpyridin-2-yl)piperidin-4-ol
2-[(5-amino-1,3,4-thiadiazol-2-yl)sulfanyl]-N-[(2-ethoxypyridin-3-yl)methyl]acetamide
8-[3-(2-chlorophenyl)-5-methyl-1,2-oxazole-4-carbonyl]-1-oxa-8-azaspiro[4.5]decane
N-(2-{imidazo[1,2-a]pyridin-2-yl}ethyl)-1-(oxolan-2-ylmethyl)-1H-1,2,3-triazole-4-carboxamide
1-[(2R,3R,6R)-3-(3-hydroxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-4-(1H-pyrazol-4-yl)butan-1-one
methyl (2S)-1-{3-chloro-4-[(1-methanesulfonylpiperidin-4-yl)oxy]benzoyl}pyrrolidine-2-carboxylate
1-cyclopropyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}-6-oxopiperidine-3-carboxamide
1-benzyl-N3-[2-(4-fluorophenyl)ethyl]-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide
3-{[2-(1H-imidazol-4-yl)-1H-imidazol-1-yl]methyl}-4-propyl-4H-1,2,4-triazole
2-(5-aminopyrazin-2-yl)-N,N-bis(propan-2-yl)benzamide
3-{5-[5-(3-methyl-1,2,4-oxadiazol-5-yl)pyridin-2-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanoic acid
1-[4-ethoxy-3-(1H-pyrrol-1-yl)phenyl]-3-[3-(1-methyl-1H-pyrazol-4-yl)propyl]urea
1-methyl-2-(5-{[2-(pyridin-2-yl)pyrrolidin-1-yl]methyl}furan-2-yl)-1H-1,3-benzodiazole
5-{[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-4-(propan-2-yl)-1,2,3-thiadiazole
N-cyclopropyl-N-({4-methoxy-3-[2-(pyridin-2-yl)ethoxy]phenyl}methyl)-4-methylbenzamide
1-[3-(dimethyl-1,2-oxazol-4-yl)propyl]-3-[1-methyl-3-(pyridin-2-yl)-1H-pyrazol-5-yl]urea
5-[4-(2-phenylethyl)piperidine-1-carbonyl]-2-(pyridin-3-yl)pyrimidine
2-(3-{3-[(2-fluorophenyl)methoxy]azetidine-1-carbonyl}piperidin-1-yl)acetamide
5-acetyl-N-methyl-N-[(1-methylpiperidin-2-yl)methyl]thiophene-3-carboxamide
3-cyclobutyl-5-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazole
(3S,9aR)-3-benzyl-8-[(3,4-dimethylphenyl)methyl]-2-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
3-(2-fluorophenyl)-N-{5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-a]azepin-3-ylmethyl}-1H-pyrazole-5-carboxamide
methyl[(4-methyl-1H-imidazol-2-yl)methyl]{[2-(1H-pyrazol-1-yl)phenyl]methyl}amine
4-{[4-(1-hydroxy-2-phenylethyl)piperidin-1-yl]methyl}-1,5-dimethyl-1H-pyrrole-2-carbonitrile
1-(4-{3-[(4-fluorophenyl)methyl]-3-(hydroxymethyl)piperidine-1-carbonyl}phenyl)ethan-1-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-phenylethyl)cyclopropanamine
N-{[2-(2-fluorophenoxy)pyridin-3-yl]methyl}-3-(1,2-oxazinan-2-yl)propanamide
methyl (2S)-1-{[4-(1,3-thiazol-2-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}pyrrolidine-2-carboxylate
[2-({4-[(2-methoxypyrimidin-5-yl)methyl]piperazin-1-yl}methyl)phenyl]methanol
2-amino-N-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-N-methyl-1,3-benzothiazole-5-carboxamide
2-(2-methoxyethyl)-4-({3-phenylpyrazolo[1,5-a]pyrimidin-6-yl}methyl)morpholine
N-[(2-ethyl-5-fluoro-3-methyl-1H-indol-7-yl)methyl]-2-(ethylamino)pyrimidine-5-carboxamide
N1-{1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}hexane-1,6-diamine
N-(2-methylphenyl)-4-[4-(pyridin-2-yl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
2-cyclopropyl-8-(3-methoxybenzenesulfonyl)-2,8-diazaspiro[5.5]undecan-3-one
N-methyl-2-(1-methylpyrrolidin-2-yl)-N-[2-(1H-pyrazol-1-yl)ethyl]acetamide
1-ethyl-3-(propan-2-yl)-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1H-pyrazole-5-carboxamide
4-(2-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-2-oxoethyl)-1,2,3,6-tetrahydropyridazine-3,6-dione
2-(cyclopropylmethyl)-9-[(2S)-2-hydroxy-2-phenylacetyl]-2,9-diazaspiro[5.5]undecan-3-one
4-[1-(2-chloro-6-fluoro-3-methylbenzoyl)piperidin-3-yl]benzoic acid
N-[phenyl(pyridin-2-yl)methyl]-1-[(1s,4s)-4-aminocyclohexyl]-1H-1,2,3-triazole-4-carboxamide
3,4,7-trimethyl-2-[2-(1H-pyrazol-1-ylmethyl)-1,4-oxazepane-4-carbonyl]-1H-indole
2-[4-({2-[2-(1H-imidazol-1-yl)ethoxy]phenyl}methyl)morpholin-3-yl]acetic acid
1-[5-(1H-imidazol-2-yl)imidazo[2,1-b][1,3]thiazole-6-carbonyl]azocane
2-methyl-N-[(3-methyl-7-{[(4S)-4-(prop-1-en-2-yl)cyclohex-1-en-1-yl]methyl}-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]furan-3-carboxamide
4-[7-(1-ethyl-1H-pyrazole-4-carbonyl)-4-oxo-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
2-[1-(2-methylpropyl)-4-(quinolin-4-ylmethyl)piperazin-2-yl]ethan-1-ol
N,8-dimethyl-N-(2-phenylethyl)-3-{[4-(propan-2-yl)piperazin-1-yl]methyl}imidazo[1,2-a]pyridine-2-carboxamide