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N-[3-({5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}carbamoyl)-2-methylphenyl]oxolane-2-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-(3-ethyl-1H-pyrazole-5-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
1-cyclopropanecarbonyl-4-[2-(4-phenylazepane-1-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N-methyl-6-(pyridin-3-yl)pyridine-3-carboxamide
4-{[(1S,5R)-6-(cyclopropylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzamide
(2E)-3-(3,4-dimethoxyphenyl)-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]prop-2-enamide
2-[3-({3'-oxo-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-1-yl}carbonyl)piperidin-1-yl]acetamide
6-methyl-2-(pyrazin-2-yl)-5-[5-(thiophen-3-yl)-1,2,4-oxadiazol-3-yl]-1,2,3,4-tetrahydro-2,7-naphthyridine
({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)[(4-methoxyphenyl)methyl]methylamine
5-{3-[(2,3-dihydro-1,4-benzodioxin-6-yl)amino]piperidine-1-carbonyl}-2-methyl-2,3-dihydro-1H-isoindole-1,3-dione
3-oxo-N-[1-(pyrazin-2-yl)propan-2-yl]-3,4-dihydroquinoxaline-2-carboxamide
(2S,4S)-N-ethyl-1-(naphthalen-1-ylmethyl)-4-{[(4-phenylphenyl)methyl]amino}pyrrolidine-2-carboxamide
5-[3-(2-ethylphenoxy)azetidine-1-carbonyl]-2-methoxyphenol
2-{4-[1-(2-methoxyethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}-6-(methoxymethyl)pyridine
2-(dimethylamino)-2-(3-fluorophenyl)-N-[3-(4-methylpiperidin-1-yl)-3-oxopropyl]acetamide
2-(4-cyclohexyl-4H-1,2,4-triazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[2-(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)ethyl]-2-propyl-1,3-thiazole-4-carboxamide
3-chloro-N-[cyclopropyl(4-methylpyridin-2-yl)methyl]-4-hydroxybenzamide
1-[(3R,4R)-3-[(dimethylamino)methyl]-4-(hydroxymethyl)pyrrolidin-1-yl]-3-(4-methylphenyl)propan-1-one
1-{[4-(2,3-dihydro-1,4-benzodioxin-6-yl)phenyl]methyl}pyrrolidine
N-[(1,5-dimethyl-1H-indazol-3-yl)methyl]-1-(oxolane-2-carbonyl)piperidin-4-amine
5-(3-benzyl-1,2,4-oxadiazol-5-yl)-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]pyridin-2-amine
3-[(4-{[(3S,4S)-4-ethoxy-1-methylpyrrolidin-3-yl]amino}-6-methylpyrimidin-2-yl)amino]phenol
4-[2-(methylamino)benzoyl]-7-(pyridin-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(3S,4S)-1-(piperidine-1-sulfonyl)-4-(pyridin-2-yl)pyrrolidine-3-carboxylic acid
1-{2-[(2S)-2-(morpholine-4-carbonyl)pyrrolidin-1-yl]-2-oxoethyl}-1,2,3,4-tetrahydroquinolin-2-one
ethyl 5-(2-benzyl-1,3-thiazole-4-carbonyl)-1-(2-methylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
3-[4-(dimethylamino)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-6-fluoroquinolin-4-ol
6-[3-(1-methyl-1H-imidazol-2-yl)piperidine-1-carbonyl]quinoxaline
1-[3-(pyridin-2-yl)azetidin-1-yl]-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propan-1-one
2-cyclopropyl-9-[(2,5-dimethylphenyl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
1-[1-(adamantan-2-yl)piperidin-3-yl]-4-(4-methoxyphenyl)piperazine
3-{2-[(1R,5R)-6-(2-methoxyethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-2-oxoethyl}-2,3-dihydro-1,3-benzoxazol-2-one
2-(pyridin-3-yl)-N-{2-[2-(pyridin-4-yl)-1,3-thiazol-4-yl]ethyl}pyrimidine-5-carboxamide
(4aR,7aS)-1-methyl-4-(2,3,6-trimethylquinoline-4-carbonyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-(3-fluorophenyl)-N-[2-(1H-imidazol-1-yl)ethyl]-N-methylimidazo[2,1-b][1,3]thiazole-3-carboxamide
[(3R,4R)-4-[(4-methyl-1,4-diazepan-1-yl)methyl]-1-[(4-methyl-1H-imidazol-2-yl)methyl]pyrrolidin-3-yl]methanol
N,N-diethyl-1-{1-[4-(2-fluorophenyl)pyrimidin-2-yl]-5-(propan-2-yl)-1H-pyrazole-4-carbonyl}pyrrolidin-3-amine
N-(2-methoxyethyl)-N-[(4-methylphenyl)methyl]-2-(propan-2-yloxy)propanamide
methyl 2-{[5-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)-1,3,4-thiadiazol-2-yl]sulfanyl}acetate
[(3-{[1-(3,4-dimethoxybenzenesulfonyl)piperidin-4-yl]oxy}phenyl)methyl](methyl)(thiophen-3-ylmethyl)amine
1-methyl-4-(quinoxaline-5-carbonyl)piperazin-2-one
3-{2-[(4-chlorophenyl)methyl]-5-oxopyrrolidin-2-yl}-N-[1-(thiophen-3-yl)propan-2-yl]propanamide
4-(3,4-dimethoxyphenyl)-1H-pyrrolo[2,3-b]pyridine
2-[3,5-dimethyl-4-(7-methyl-1H-1,3-benzodiazol-2-yl)-1H-pyrazol-1-yl]ethan-1-ol
cyclopentyl 4-({[(5-amino-1,3,4-thiadiazol-2-yl)methyl]carbamoyl}amino)benzoate
4-[(5-chlorothiophen-2-yl)sulfonyl]-9-methoxy-7-(6-methoxypyridin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
3-{1-[5-(4-fluorophenyl)pyrazolo[1,5-a]pyrimidin-7-yl]piperidin-3-yl}propanamide
1-(4-aminopyrimidin-2-yl)-3-(2-phenoxyethyl)piperidine-3-carboxylic acid
3-(dimethyl-1,2-oxazol-4-yl)-1-[(1S,5R)-3-(pyridine-3-carbonyl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]propan-1-one