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4-{4-[(2-fluorophenyl)methyl]piperazin-1-yl}-2-(thiophen-3-ylmethyl)-2,3-dihydro-1H-isoindole-1,3-dione
1-(4-methoxyphenyl)-2,2-dimethyl-N-[3-(2-oxopyrrolidin-1-yl)propyl]cyclopropane-1-carboxamide
N-[3-(azepane-1-carbonyl)phenyl]-6-(hydroxymethyl)-1,4-oxazepane-4-carboxamide
({3-[1-(4-methylphenyl)cyclopentyl]-1,2,4-oxadiazol-5-yl}methyl)(oxolan-2-ylmethyl)(pyridin-2-ylmethyl)amine
7-(1-phenyl-1H-1,2,3,4-tetrazol-5-yl)-2-oxa-7-azaspiro[4.5]decane
N-(2-{7-[(2-methylphenyl)methyl]-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl}ethyl)furan-3-carboxamide
5-(1H-imidazol-1-ylmethyl)-2-[3-(1H-pyrazol-5-yl)phenyl]pyridine
N-{2H,3H-imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-5-phenyl-5H,6H,7H-pyrrolo[3,2-d]pyrimidin-2-amine
(1R,5R)-N,N-dimethyl-6-{[5-(1H-pyrazol-3-yl)furan-2-yl]methyl}-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
3-(5-{[(2-ethyl-6-methylpyridin-3-yl)oxy]methyl}-1,2,4-oxadiazol-3-yl)-6-methylpyridazine
6-(6-hydroxy-1,4-diazepane-1-carbonyl)-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
N-[1-(3-ethyl-1,2,4-oxadiazol-5-yl)ethyl]-1-[5-(trifluoromethyl)pyridin-2-yl]piperidin-4-amine
1-[(5-tert-butyl-1H-pyrazol-3-yl)methyl]-4-(1H-pyrazol-1-yl)piperidine-4-carboxylic acid
2-(2-{1-[2-(2H-indazol-2-yl)acetyl]piperidin-3-yl}-1H-imidazol-1-yl)acetamide
1-[(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
1-[4-({[(3-hydroxypyrrolidin-3-yl)methyl]amino}methyl)phenyl]pyrrolidin-2-one
1-{[2-(propan-2-yl)-1,3-oxazol-4-yl]methyl}-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
1-[1-(3-phenylprop-2-yn-1-yl)piperidin-4-yl]-N-(pyridin-2-ylmethyl)piperidine-4-carboxamide
2-{2-[1-(6,8-dimethylquinolin-4-yl)piperidin-3-yl]-1H-imidazol-1-yl}acetamide
N-[(1-benzyl-1H-imidazol-2-yl)methyl]-N-methyl-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxamide
1-(2-methoxyphenyl)-N-[2-(pyridin-3-yl)ethyl]-1H-pyrazole-4-carboxamide
4-{[3-(furan-2-yl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-1-azatricyclo[7.3.1.05,13]trideca-3,5,7,9(13)-tetraen-2-one
5-methyl-N,N-bis(1,3-oxazol-4-ylmethyl)-2-phenyl-1H-imidazole-4-carboxamide
3-(1-methylpiperidin-3-yl)-1-[4-(1H-1,2,4-triazole-3-carbonyl)piperazin-1-yl]propan-1-one
methyl 3-propanamido-5-({[3-(1H-pyrazol-1-yl)phenyl]formamido}methyl)benzoate
(2R,6S)-4-{2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-1,3-oxazole-4-carbonyl}-2,6-dimethylmorpholine
(1S,5R)-6-(5-ethylthiophene-2-carbonyl)-3-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonane
dimethyl(2-{2-[1-(morpholine-4-sulfonyl)piperidin-4-yl]-1H-imidazol-1-yl}ethyl)amine
1-{4-[(3-methylphenyl)sulfanyl]piperidin-1-yl}-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
2-(2-fluorophenoxymethyl)-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}-1,3-oxazole-4-carboxamide
7-chloro-3-[2-(oxan-2-yl)ethyl]-3,4-dihydroquinazolin-4-one
2,3,5-trimethyl-N-[(2-methyl-1,2,3,4-tetrahydroisoquinolin-3-yl)methyl]pyrazolo[1,5-a]pyrimidin-7-amine
2-(2-{[methyl(oxan-4-yl)amino]methyl}-4-(pyrazin-2-yl)phenoxy)acetic acid
2,5-dioxo-6-{[2-(piperidin-1-yl)phenyl]methyl}-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
ethyl 5-({[1-cyclopentyl-4-oxo-5-(piperidine-1-carbonyl)-1,4-dihydropyridin-3-yl]formamido}methyl)furan-2-carboxylate
2-(4-methylpentanoyl)-N-[2-(pyridin-2-yl)ethyl]-1,2,3,4-tetrahydroisoquinoline-7-sulfonamide
4-[({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl}amino)methyl]benzene-1,3-diol
4-methyl-2-{4-[4-methyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine-1-carbonyl}phenol
2-{5-[1-(3-methoxyphenoxy)ethyl]-1-(2-methylphenyl)-1H-1,2,4-triazol-3-yl}acetamide
1-(2,2-dimethyloxan-4-yl)-1-ethyl-3-(2-methoxy-5-methylphenyl)urea
(2S,4R)-N,N-diethyl-1-(4-hydroxybenzoyl)-4-propanamidopyrrolidine-2-carboxamide
1-[(1R,5R)-6-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-3,6-diazabicyclo[3.2.2]nonan-3-yl]ethan-1-one
7,8-dimethyl-4-(2-methylpyrrolidine-1-carbonyl)-2-[2-(propan-2-yl)pyrimidin-5-yl]quinoline
2-(2H-1,3-benzodioxol-5-yl)-1-(4-{2-[2-(4-methoxyphenyl)ethyl]-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)ethan-1-one
3-[2-(3,4-difluorophenyl)ethyl]-N,N-dimethylpiperidine-1-sulfonamide
7-(cyclopropylmethyl)-2-{[4-(3-hydroxy-3-methylbutyl)phenyl]methyl}-2,7-diazaspiro[4.5]decan-6-one
N-[2-(4,5-dimethyl-1H-1,3-benzodiazol-2-yl)ethyl]-2-(4-oxo-3,4-dihydroquinazolin-3-yl)acetamide
3-{imidazo[1,2-a]pyridin-2-yl}-N-{[1-(1-methyl-6-oxo-1,6-dihydropyridazin-4-yl)pyrrolidin-3-yl]methyl}propanamide
1-{3-[3-(4-methylphenoxymethyl)piperidine-1-carbonyl]phenyl}pyrrolidin-2-one
3-(3-methoxyphenyl)-N-{3-[(5-methylpyridin-2-yl)amino]propyl}-1H-pyrazole-4-carboxamide