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6-[4-(2,7-dioxo-1,3-diazepane-4-carbonyl)piperazin-1-yl]pyridine-3-carbonitrile
2-methyl-4-oxo-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]-4,5,6,7-tetrahydro-1H-indole-3-carboxamide
2-[(3,5-difluorophenyl)methyl]-8-(pyrrolidine-1-carbonyl)-2,8-diazaspiro[4.5]decan-3-one
4-[3-(2-fluorophenyl)pyrrolidine-1-carbonyl]-3-methyl-1-propyl-1H-pyrazole
1-{3-[2-(2,4-difluorophenyl)ethyl]piperidin-1-yl}-3-(pyrazin-2-yl)propan-1-one
N-[(1-ethyl-1H-imidazol-5-yl)methyl]-2-(1H-indol-3-yl)-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
4-{4-[(3,5-dimethyl-1H-pyrazol-1-yl)methyl]benzoyl}-2,7-dimethyl-2,3,4,5-tetrahydro-1,4-benzoxazepine
8-fluoro-2-[(2R)-2-(hydroxymethyl)pyrrolidine-1-carbonyl]-1,4-dihydroquinolin-4-one
3-(5-chloro-2-methoxyphenyl)-N-cyclohexyl-N-methyl-5-(1H-1,2,3,4-tetrazol-1-yl)benzamide
1-(cyclohexylmethyl)-N-[(4-ethyl-4H-1,2,4-triazol-3-yl)methyl]-N-methyl-6-oxopiperidine-3-carboxamide
N-[(5-ethyl-1,3,4-thiadiazol-2-yl)methyl]-2-propyl-1,3-thiazole-4-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-1-ethyl-3-(4-methyl-1,4-diazepane-1-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-methyl-2-{4-[2-(pyridin-2-yl)-1H-imidazol-1-yl]phenyl}acetamide
5-[1-(ethanesulfonyl)piperidin-4-yl]-5-(pyridin-3-yl)imidazolidine-2,4-dione
2,6-dimethyl-4-(4-phenyl-1H-imidazol-5-yl)phenol
3-methoxy-1-[2-(3-methoxypyrrolidin-1-yl)-2-oxoethyl]-1,2-dihydropyridin-2-one
2-(1-cyclohexyl-2,6,6-trimethyl-4-oxo-4,5,6,7-tetrahydro-1H-indol-3-yl)-N-(2-acetamidoethyl)acetamide
N-[(2,4-dimethoxyphenyl)methyl]-3-{1-[(2,5-dimethylphenyl)methyl]piperidin-3-yl}propanamide
1-[2-(4-fluorophenyl)piperidin-1-yl]-2-(3-hydroxyphenyl)ethan-1-one
1-{3-[(4-fluorophenyl)amino]piperidin-1-yl}-2-(2,2,3,3-tetrafluoropropoxy)ethan-1-one
(3R,4R)-4-ethyl-1-(1-ethyl-2,5-dimethyl-1H-pyrrole-3-carbonyl)piperidine-3,4-diol
1-[2-ethyl-5-(4H-1,2,4-triazol-4-yl)phenyl]-3-[2-(2-oxoimidazolidin-1-yl)ethyl]urea
1-(5-methyl-2-phenyl-1H-imidazole-4-carbonyl)-3-[(methylsulfanyl)methyl]piperidine
3-fluoro-4-methoxy-N-[1-(1-methylpiperidin-4-yl)piperidin-3-yl]benzamide
1-[5-(2-chloro-4-methoxyphenoxymethyl)-1H-pyrazole-3-carbonyl]-3-methoxypiperidine
N-{[2-(4-chlorophenyl)-7-(methylsulfanyl)quinolin-3-yl]methyl}-2-(3-methyl-1H-pyrazol-1-yl)-N-(oxolan-2-ylmethyl)acetamide
3-[4-hydroxy-4-(5-methylpyridin-2-yl)piperidine-1-carbonyl]-6-phenyl-1,2-dihydropyridin-2-one
N-({1-[(2,4-dimethylphenyl)methyl]pyrrolidin-3-yl}methyl)-2-(1H-1,2,4-triazol-1-yl)acetamide
2-methyl-9-[(1-methyl-1H-1,2,3-benzotriazol-4-yl)sulfonyl]-2,9-diazaspiro[5.5]undecan-3-one
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-(pyrazin-2-yl)-2,7-diazaspiro[4.5]decane
2-(3-{3-[5-(pyrrolidine-1-carbonyl)furan-2-yl]phenyl}-1H-pyrazol-1-yl)acetamide
(2R,3R,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(3,6-dimethylpyrazin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane
3-(3-cyclohexylpyrrolidin-1-yl)-1-ethylpiperidine
3-(2-hydroxyphenyl)-3-(4-hydroxyphenyl)-1-[4-(pyrazin-2-yl)piperazin-1-yl]propan-1-one
3-(2H-1,3-benzodioxol-5-yl)-5-(cyclohex-3-en-1-ylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
methyl 3-(2-chloro-6-fluorobenzamido)-6-(piperidin-1-ylmethyl)thieno[2,3-b]pyridine-2-carboxylate
N-[(3-chlorophenyl)methyl]-N-cyclopropyl-5-methyl-1,3-oxazole-4-carboxamide
N-(2,1,3-benzothiadiazol-5-ylmethyl)-8-fluoro-N-methylquinoline-2-carboxamide
[(6-chloro-2H-1,3-benzodioxol-5-yl)methyl](methyl)(oxan-2-ylmethyl)amine
N-[(4-ethylphenyl)methyl]-N-methyl-3-{2-[(4-methylphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
4-[2-(ethylamino)-4-methyl-1,3-thiazole-5-carbonyl]piperazine-2-carboxylic acid
4-{1-[3-(1-methylpiperidin-4-yl)propanoyl]piperidin-3-yl}benzoic acid
1-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-4-(3-methylphenoxy)piperidine
3-hydroxy-N-[3-(1H-imidazol-1-yl)propyl]-N-(pyridin-4-ylmethyl)pyridine-2-carboxamide
N-[2-(ethylsulfanyl)ethyl]-3-phenyladamantane-1-carboxamide
2-{4-[(4-methylphenyl)methyl]-1-(2-methylpropyl)piperazin-2-yl}ethan-1-ol
2-[5-methanesulfonyl-4-(piperidin-3-yl)pyrimidin-2-yl]-1,2,3,4-tetrahydroisoquinoline
ethyl 2-[2-(dimethylamino)-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl]acetate
3-benzyl-5-(1-benzyl-1H-pyrazol-4-yl)-1H-1,2,4-triazole
1-[5-(trifluoromethyl)pyridin-2-yl]-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one