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N-[(3S,4R)-4-hydroxyoxolan-3-yl]-N,2,8-trimethylquinoline-4-carboxamide
(2R,3S,6R)-3-(3,5-difluorophenyl)-5-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]-1,5-diazatricyclo[5.2.2.02,6]undecane
{[2-(ethanesulfonyl)-1-(2-phenylethyl)-1H-imidazol-5-yl]methyl}(methyl)[(4-methylphenyl)methyl]amine
2-[(4aS,7aS)-octahydro-1H-pyrrolo[3,4-b]pyridin-6-ylmethyl]-6-fluoroquinolin-4-ol
4-[(1R,2R,6S,7S)-4-azatricyclo[5.2.1.02,6]decan-4-yl]-6-methoxypyrimidin-2-amine
5-{1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-4-yl}-2-phenoxypyridine
8-methyl-3-{2-methyl-2,8-diazaspiro[4.5]decane-8-carbonyl}-1,4-dihydroquinolin-4-one
2-[3-benzyl-1-(4-chlorophenyl)-5-oxo-4,5-dihydro-1H-1,2,4-triazol-4-yl]-N-(carbamoylmethyl)acetamide
1-(2-amino-6-methylpyrimidin-4-yl)-N-[4-(3-methylphenyl)phenyl]piperidine-4-carboxamide
1-{2-ethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-yl}-3-(3-methylphenyl)piperidine
N-methyl-3-(5-methyl-1H-1,2,4-triazol-3-yl)-N-[(1-phenylpyrrolidin-3-yl)methyl]propanamide
2-[2-(4-methylpiperazine-1-carbonyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-5-yl]-2-oxo-N-(propan-2-yl)acetamide
2-(2,5-dioxoimidazolidin-1-yl)-N-[(3R,4S)-1-(2-hydroxyethyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
3-(5-tert-butyl-1,3,4-thiadiazol-2-yl)-1-{[1-(propan-2-yl)-1H-pyrazol-4-yl]methyl}urea
2-{[(dimethylsulfamoyl)amino]methyl}-N-(3-phenylpropyl)quinazolin-4-amine
(3aR,6aR)-2-cyclopropanecarbonyl-5-(1,3-thiazol-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
[(2-butyl-1H-imidazol-4-yl)methyl][(1-ethylpyrrolidin-2-yl)methyl]{[1-(2-methoxyethyl)piperidin-4-yl]methyl}amine
(2R,3R)-3-methoxy-1'-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]-2,3-dihydrospiro[indene-1,4'-piperidine]-2-ol
4-{4-[(2,5-difluorophenyl)methyl]piperazin-1-yl}-2-[(4-methoxyphenyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
3-[(3R,4S)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(morpholin-4-yl)piperidin-3-yl]propanoic acid
4,5-dimethyl-6-[3-(thiophene-2-carbonyl)piperidin-1-yl]pyrimidin-2-amine
1-cyclopropyl-5-oxo-N-[(3-phenoxyphenyl)methyl]pyrrolidine-3-carboxamide
N-[2-(5-amino-1,3,4-thiadiazol-2-yl)ethyl]-2-(1H-1,3-benzodiazol-1-yl)propanamide
1-[2-({[2-(4-chlorophenyl)pyrimidin-5-yl]methyl}(methyl)amino)ethyl]piperidin-2-one
2-{1-[(4-methanesulfonylphenyl)methyl]pyrrolidin-2-yl}pyridine
6-[(3R,4R)-3-hydroxy-4-[4-(pyridin-2-yl)piperazin-1-yl]piperidin-1-yl]pyridine-2-carbonitrile
N-(9H-fluoren-9-yl)-2-oxo-6-({1,3,3-trimethyl-6-azabicyclo[3.2.1]octan-6-yl}methyl)-1,2-dihydropyridine-3-carboxamide
2-[(2R,6S)-2,6-dimethylmorpholine-4-carbonyl]-N-[(3-methylthiophen-2-yl)methyl]aniline
5-acetyl-N-[(4-phenyloxan-4-yl)methyl]-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
2-{3-[2-methyl-6-(pyrrolidin-1-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-ol
2-{5-[(4-methylpiperidin-1-yl)methyl]-1H-1,2,3,4-tetrazol-1-yl}-1-{2-[2-(morpholin-4-yl)ethyl]piperidin-1-yl}ethan-1-one
2-[4-(dimethylamino)phenyl]-N-(oxolan-3-yl)acetamide
methyl 4-({3-[(2H-1,3-benzodioxol-5-yl)amino]piperidin-1-yl}methyl)benzoate
N-[2-(1H-indol-1-yl)ethyl]-5-methylpyrazolo[1,5-a]pyrimidin-7-amine
(2R,3R,6R)-3-phenyl-5-{pyrazolo[1,5-a]pyrimidine-2-carbonyl}-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[1-(1H-imidazol-1-yl)-3,3-dimethylbutan-2-yl]-2-(thiophen-2-yl)-1,3-thiazole-4-carboxamide
2-[ethyl(methyl)amino]-1-{4-[2-methyl-6-(morpholin-4-yl)pyrimidin-4-yl]piperidin-1-yl}ethan-1-one
(2R,6R)-4-(2-hydroxypyridine-3-carbonyl)-10-methoxy-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
1-(2-methoxy-4-methyl-1,3-thiazole-5-carbonyl)-3-(2-methylphenoxymethyl)piperidine
4-fluoro-1-(5-{1-[(3-methylthiophen-2-yl)methyl]pyrrolidin-2-yl}thiophene-2-carbonyl)piperidine
2-(2-methyl-1H-1,3-benzodiazol-5-yl)-N-[(3R)-pyrrolidin-3-yl]acetamide
N-(1-{2-[4-(2H-1,3-benzodioxol-5-ylmethyl)piperazin-1-yl]-2-oxoethyl}-1H-pyrazol-4-yl)-2-fluorobenzamide
7-(1-ethyl-1H-pyrazole-4-carbonyl)-N,N-dimethyl-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-[7-(3-chlorophenyl)-9-(oxan-2-ylmethoxy)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-ethylbutan-1-one
(1,4-dioxan-2-ylmethyl)({[3-(3-fluoro-4-methoxyphenyl)-1H-pyrazol-4-yl]methyl})methylamine
N-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-N-methyl-5-(phenoxymethyl)-1H-pyrazole-3-carboxamide
5-(1,4-oxazepane-4-carbonyl)-1-(3-phenylpropyl)piperidin-2-one
3-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-cyclopropylpropanamide
N-[(2-fluorophenyl)methyl]-1-methyl-5-(morpholin-4-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(2S)-1-methoxy-3-phenylpropan-2-yl]-2-(1H-1,2,4-triazol-3-yl)benzamide