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2-(3-{[4-(hydroxymethyl)piperidin-1-yl]methyl}phenyl)-6-(pyridin-3-yl)-3,4-dihydropyrimidin-4-one
(2,1,3-benzoxadiazol-5-ylmethyl)(methyl)({2-methylimidazo[1,2-a]pyridin-3-yl}methyl)amine
3-(1-benzofuran-2-yl)-1-benzyl-4-{[(2S)-2-(methoxymethyl)pyrrolidin-1-yl]methyl}-1H-pyrazole
3-chloro-6-[2-chloro-4-(pyrrolidin-1-ylmethyl)phenoxy]pyridazine
N-methyl-4-{1-methyl-1H-pyrrolo[2,3-b]pyridin-4-yl}benzamide
2-{[5-(1-ethyl-1H-pyrazol-4-yl)-4-(2-methoxyphenyl)-4H-1,2,4-triazol-3-yl]sulfanyl}acetic acid
(3aS,7aR)-2-(5-acetylthiophene-2-carbonyl)-5-methyl-octahydro-1H-pyrrolo[3,4-c]pyridine-3a-carboxylic acid
1-[(2-fluorophenyl)methyl]-N-(3-hydroxy-2,2-dimethylpropyl)-6-oxopiperidine-3-carboxamide
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-[(2-methoxyphenyl)methyl]piperazine
3-{[(2-methoxy-4,6-dimethylpyridin-3-yl)methyl]sulfamoyl}-N,N-dimethylbenzamide
2-[(5-methyl-1,3,4-oxadiazol-2-yl)sulfanyl]-1-{3-[2-(2-methylphenyl)ethyl]piperidin-1-yl}ethan-1-one
N-(cyclohexylmethyl)-2-{1-[(4-ethoxyphenyl)methyl]-3-oxopiperazin-2-yl}acetamide
N-methyl-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}-N-(1,3-thiazol-2-ylmethyl)acetamide
3-{6-hydroxy-4-[(4-methyl-1H-imidazol-5-yl)methyl]-1,4-diazepan-1-yl}-N,N-dimethylpropanamide
5-{[2-(3-methoxyphenyl)ethyl]amino}-N,N-dimethyl-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
N-[(5-{[(2-fluorophenyl)methyl]sulfanyl}-4-(2-methylpropyl)-4H-1,2,4-triazol-3-yl)methyl]cyclohexanecarboxamide
4-{7-methyl-6-oxo-2,7-diazaspiro[4.5]decan-2-yl}-4-oxobutane-1-sulfonamide
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-(pentan-3-yl)piperidine-3-carboxamide
[(1-ethylpyrrolidin-2-yl)methyl]({[8-methyl-2-(thiophen-2-yl)quinolin-3-yl]methyl})amine
5-(2-{2-[2-(4-hydroxyphenyl)ethyl]piperidin-1-yl}-2-oxoethyl)-2,6-dimethyl-3,4-dihydropyrimidin-4-one
1-benzyl-4-phenyl-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]piperidine-4-carboxamide
7-(2-methoxyphenyl)-2-[1-(2-methylpropyl)-1H-imidazol-5-yl]-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
2-(2-methoxyphenyl)-2-[methyl(pyrazin-2-ylmethyl)amino]acetic acid
1-[4-(hydroxymethyl)-4-{[2-(trifluoromethyl)phenyl]methyl}piperidin-1-yl]-3-phenoxypropan-1-one
N-methyl-2-(4-methyl-1-oxo-1,2-dihydrophthalazin-2-yl)-N-(pyrazin-2-ylmethyl)acetamide
N-[1-(3-chlorophenyl)cyclopropyl]-3-(6-methyl-2-oxo-1,2-dihydropyridin-1-yl)propanamide
5-oxo-1-[(4-phenyl-1,3-thiazol-5-yl)methyl]pyrrolidine-3-carboxylic acid
7-(1,3-benzothiazol-2-yl)-4-[(2,4-dimethoxy-3-methylphenyl)methyl]-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
5-acetyl-N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-[4-(benzyloxy)piperidin-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
N-{1,9-dioxaspiro[5.5]undecan-4-yl}-2-(5-oxo-2-phenylcyclopent-1-en-1-yl)acetamide
N-({3-[(3-fluorophenyl)methyl]-4,5-dihydro-1,2-oxazol-5-yl}methyl)-3-(2-oxo-2,3-dihydro-1H-1,3-benzodiazol-1-yl)propanamide
1-{3-[1-(cyclopropylmethyl)-1H-imidazol-2-yl]piperidine-1-carbonyl}naphthalen-2-ol
5-{4-[2-(4-chloro-2-methylphenoxy)ethyl]piperazine-1-carbonyl}-4-methylpyrimidine
2-(3-{[3-(5-fluoro-2-methoxybenzoyl)piperidin-1-yl]methyl}-1H-indol-1-yl)acetamide
N-[(1-{[5-(methoxymethyl)furan-2-yl]methyl}piperidin-3-yl)methyl]naphthalene-1-carboxamide
1-(4-methyl-1,3-oxazole-5-carbonyl)-4-[(2E)-3-phenylprop-2-en-1-yl]piperazine
N-[(4-methoxy-3,5-dimethylpyridin-2-yl)methyl]-N-methyl-7H-pyrrolo[2,3-d]pyrimidin-4-amine
1-(4-methoxybenzoyl)-N-[3-(5-methyl-1,3,4-thiadiazol-2-yl)phenyl]piperidine-2-carboxamide
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-5-methyl-N-(oxolan-2-ylmethyl)-1H-pyrazole-3-carboxamide
(2S)-2-(methoxymethyl)-1-{2-[(2-methylprop-2-en-1-yl)oxy]benzoyl}pyrrolidine
4-(3-hydroxy-6-methylpyridin-2-yl)-3-methyl-1-[(3-methylphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
4-phenyl-N-(1,3,4-thiadiazol-2-yl)-1,4-diazepane-1-carboxamide
2-ethyl-4-phenyl-9-(pyrrolidine-1-sulfonyl)-2,9-diazaspiro[5.5]undecane
4-chloro-N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-methyl-3-(trifluoromethyl)-1H-pyrazole-5-carboxamide
2-[4-(4-chlorophenoxy)piperidin-1-yl]-N-cyclopropylpyridine-4-carboxamide
[(3,4-dimethoxyphenyl)methyl]({[2-(2-ethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})methylamine
(3aR,6aR)-2-(2-hydroxyethyl)-5-[3-(methylsulfanyl)propanoyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N4-[1-(furan-2-carbonyl)piperidin-4-yl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-2,4-diamine
N5-[2-(4-chlorophenyl)ethyl]-1-(cyclohexylmethyl)-N3,N3-dimethyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide