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N-[2-(3,5-dimethylphenoxy)ethyl]-N-methyl-2-(2-oxo-1,3-oxazolidin-3-yl)acetamide
7-[(2-fluoro-5-methoxyphenyl)methyl]-2-{[5-(methoxymethyl)furan-2-yl]methyl}-2,7-diazaspiro[4.5]decane
(3R,5S)-5-(7-chloro-2,3,4,5-tetrahydro-1,4-benzoxazepine-4-carbonyl)pyrrolidin-3-amine
1-methyl-N-[2-(morpholin-4-yl)ethyl]-5-[2-(propan-2-yl)-1,3-thiazole-4-carbonyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxamide
4-(2-{1-[(4,6-dimethylpyrimidin-2-yl)methyl]piperidin-2-yl}ethyl)morpholine
4-[3-(hydroxymethyl)-3-(2-phenoxyethyl)piperidin-1-yl]-2-methoxypyridine-3-carbonitrile
2-[4-(1,3-benzothiazol-2-yl)piperazin-1-yl]-N-ethylpyridine-3-carboxamide
4-{3-carbamoyl-5H,6H,7H-cyclopenta[b]pyridin-2-yl}morpholine-2-carboxylic acid
2-(azepan-1-yl)-N-{[5-(2-methylpropyl)-1,2-oxazol-3-yl]methyl}acetamide
N-{1-methyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-1-(pyridin-3-ylmethyl)piperidin-4-amine
[(2S,4R)-4-(dimethylamino)-1-(pyridine-2-carbonyl)pyrrolidin-2-yl]methanol
N-(1-{1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)-2-phenylacetamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-(4H-1,2,4-triazol-4-yl)pyridine-4-carboxamide
1-[(2-chloro-6-fluoro-3-methylphenyl)methyl]-4-(2-methylquinolin-6-yl)piperidin-4-ol
8-{[2-(furan-2-yl)phenyl]methyl}-3-phenyl-1,8-diazaspiro[4.5]decan-2-one
1-(2-ethoxyethyl)-4-(1,2,3,4-tetrahydronaphthalen-2-yl)piperazine
4-(4-{[(3R,5S)-3-[(dimethylamino)methyl]-5-(hydroxymethyl)piperidin-1-yl]methyl}phenyl)-2-methylbut-3-yn-2-ol
1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}-3-[4-(dimethylamino)phenyl]propan-1-one
(2S,4R)-N-methyl-1-(2-phenylethyl)-4-[3-(1H-1,2,3,4-tetrazol-1-yl)propanamido]pyrrolidine-2-carboxamide
1-benzyl-4-(1-methyl-1H-pyrrole-2-carbonyl)-1,4-diazepan-6-ol
1-(2-chloropyridine-4-carbonyl)-N-(4-fluorophenyl)piperidin-3-amine
{[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}(methyl)(oxolan-3-ylmethyl)amine
1-[4-({ethyl[2-(1H-pyrazol-1-yl)ethyl]amino}methyl)-2-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
N,N-bis(2-hydroxyethyl)-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
[(3R,5R)-1-[3-(dimethylamino)benzoyl]-5-(pyrrolidin-1-ylmethyl)piperidin-3-yl]methanol
2-{2-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-1-yl}-6-methylpyridine
methyl 1-({4-[(2H-1,3-benzodioxol-5-yl)amino]-8-methylquinazolin-2-yl}methyl)piperidine-2-carboxylate
2-[2-(2-oxo-1,3-oxazolidin-3-yl)acetyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
N-(1,3-dimethyl-4-phenyl-1H-pyrazol-5-yl)-4-oxo-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepine-7-carboxamide
2-{[5-(2-methylphenyl)-1,2,4-triazin-3-yl](propan-2-yl)amino}ethan-1-ol
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
N-[(2,5-dimethylphenyl)methyl]-2-[3-oxo-1-(pyridin-3-ylmethyl)piperazin-2-yl]acetamide
N-{[5-(2-amino-2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}cyclobutanecarboxamide
1-(4-ethenylphenyl)-3-methyl-3-[2-(2-oxopiperidin-1-yl)ethyl]urea
3-{[8-(quinoxalin-2-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}phenol
methyl({[5-methyl-2-(1H-pyrazol-1-yl)phenyl]methyl})(pyrazin-2-ylmethyl)amine
2-[4-(4-fluorophenyl)-2-[(4-methylpiperazin-1-yl)methyl]phenoxy]-1-(4-phenyl-1,2,3,6-tetrahydropyridin-1-yl)ethan-1-one
(3S)-1-{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}pyrrolidin-3-ol
2-[(1H-imidazol-2-ylmethyl)[(2-methylphenyl)methyl]amino]butan-1-ol
1-(2-methylphenyl)-4-(pyridine-4-carbonyl)-1,4-diazepane
(4aS,7aR)-1-(3-aminopropanoyl)-4-(pyridin-3-ylmethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-(2-{1-[6-(azepan-1-yl)-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-yl]piperidin-4-yl}ethyl)acetamide
2-(methylamino)-N-[1-(3-methylpyridin-2-yl)propan-2-yl]acetamide
N-({3-[2-(morpholin-4-yl)ethoxy]phenyl}methyl)-N-(pyridin-2-ylmethyl)-4-(trifluoromethyl)benzamide
N-ethyl-2-(2-oxo-1,3-oxazolidin-3-yl)-N-{[4-(propan-2-yl)phenyl]methyl}acetamide
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-{[2-(1H-1,2,4-triazol-1-yl)phenyl]methyl}acetamide
N-[(2R,4R,6S)-2-(3,5-difluorophenyl)-6-(2,6-dimethylphenyl)oxan-4-yl]acetamide
1-(4-methylpyridin-2-yl)-1H-1,3-benzodiazole
1-[(2S,4R)-1-[(4-fluorophenyl)methyl]-4-[(1-methyl-1H-imidazol-2-yl)sulfanyl]pyrrolidine-2-carbonyl]-4-methyl-1,4-diazepane
1-cyclopentyl-N3-[furan-2-yl(phenyl)methyl]-4-oxo-N5-(propan-2-yl)-1,4-dihydropyridine-3,5-dicarboxamide