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9-(cyclopropylmethyl)-4-(2,6-diaminopyrimidin-4-yl)-1-methyl-1,4,9-triazaspiro[5.6]dodecan-10-one
1-(1-{[4-(2-aminoethyl)phenyl]methyl}piperidin-3-yl)-3-phenylpropan-1-one
N-[(2R,4R,6S)-2-[2-(3,5-dimethyl-1H-pyrazol-1-yl)ethyl]-6-(2-phenylethyl)oxan-4-yl]acetamide
N-ethyl-1-(2-fluorophenyl)-N-(2-methylprop-2-en-1-yl)cyclopropane-1-carboxamide
N-(dicyclopropylmethyl)-3-[5-(2-phenylethyl)-1,3,4-oxadiazol-2-yl]propanamide
(4aR,7aS)-1-(2-methoxyacetyl)-4-[(3-methyl-1H-1,2,4-triazol-5-yl)methyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
6-[(3-methoxyphenyl)methyl]-3-propyl-[1,2,4]triazolo[3,4-b][1,3,4]thiadiazole
N-{[8-(2-amino-6-ethyl-5-methylpyrimidin-4-yl)-1-oxa-8-azaspiro[4.5]decan-2-yl]methyl}acetamide
3-(1-{2-[2-(propan-2-yl)-1H-imidazol-1-yl]propanoyl}piperidin-4-yl)-1,3-oxazolidin-2-one
1-{5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}-3-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
2-(benzyloxy)-N-{5H,6H,7H,8H-imidazo[1,2-a]pyridin-3-yl}benzamide
3-(4-chlorophenyl)-1-[4-(methoxymethyl)piperidin-1-yl]-3-phenylpropan-1-one
4-[4-(morpholin-4-ylmethyl)piperidine-1-carbonyl]benzene-1-sulfonamide
N3-(cyclopropylmethyl)-N5-[(4-methylphenyl)methyl]-4-oxo-1-[2-(pyridin-2-yl)ethyl]-1,4-dihydropyridine-3,5-dicarboxamide
1-[(3-{[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]oxy}phenyl)methyl]-4-(pyridin-3-ylmethyl)piperazine
3-(benzenesulfonyl)-1-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}propan-1-one
4-chloro-5-{1-[(3-ethyl-1,2-oxazol-5-yl)methyl]-1H-imidazol-2-yl}-N,N-dimethyl-1,3-thiazol-2-amine
2-methyl-4-{4-[3-(pyridin-3-yl)propanoyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
4-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidine-1-carbonyl)pyridin-1-ium-1-olate
1-[1-({1-[4-(pyrrolidin-1-yl)benzoyl]piperidin-4-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
N-[1-(2,3-dihydro-1H-inden-2-yl)-2-methylpropan-2-yl]-3-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}propanamide
(1S,9aR)-1-{[4-(3-phenyl-1,2,4-oxadiazol-5-yl)piperidin-1-yl]methyl}-octahydro-1H-quinolizine
N-({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)-N-(pyridin-3-ylmethyl)cyclobutanecarboxamide
2-[(2-hydroxyethyl)(3-{5-[2-(methylsulfanyl)propyl]-4-phenyl-1H-imidazol-1-yl}propyl)amino]ethan-1-ol
3-[1-(2-amino-4-methyl-1,3-benzothiazole-6-carbonyl)piperidin-3-yl]benzoic acid
1-[(2S,6S)-6-butyl-2-(prop-2-en-1-yl)-1,2,3,6-tetrahydropyridin-1-yl]-2-{[3-(pyridin-3-yl)-[1,2,4]triazolo[4,3-b]pyridazin-6-yl]sulfanyl}ethan-1-one
N-{[2-methanesulfonyl-1-(3-phenylpropyl)-1H-imidazol-5-yl]methyl}-N-methyloxolan-3-amine
2-cyclopropyl-5-{4-[(4-ethyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}-3,4-dihydropyrimidin-4-one
2-(3-benzyl-1-methyl-2-oxo-2,3-dihydro-1H-indol-3-yl)-N-[2-(pyrrolidin-1-yl)ethyl]acetamide
5-[(4-ethylpiperazin-1-yl)methyl]-N-methyl-N-[(5-methylfuran-2-yl)methyl]-1,2-oxazole-3-carboxamide
ethyl 1-(1H-imidazol-2-ylmethyl)-3-[(3-methoxyphenyl)methyl]piperidine-3-carboxylate
(3R,4S)-4-cyclopropyl-1-{[3-(methoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}-N,N-dimethylpyrrolidin-3-amine
5-(4-methylpiperidine-1-carbonyl)-4-oxo-1-(propan-2-yl)-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}-1,4-dihydropyridine-3-carboxamide
N-(1-cycloheptyl-5-oxopyrrolidin-3-yl)-6-(2-methylpropyl)-2-oxo-1,2-dihydropyrimidine-4-carboxamide
2-[4-(1,3-benzothiazol-2-yl)-2-[(dimethylamino)methyl]phenoxy]-N-(1,2,3,4-tetrahydronaphthalen-1-yl)acetamide
6-{4-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]piperazin-1-yl}pyrimidine-2,4-diamine
ethyl 4-(cyclopropylmethyl)-1-(4-methylbenzenesulfonyl)piperidine-4-carboxylate
ethyl (4aR,6R,8aS)-6-(morpholin-4-yl)-2-(pyridin-2-ylmethyl)-decahydroisoquinoline-8a-carboxylate
(3S,4R)-1-[2-(ethylamino)pyrimidine-5-carbonyl]-4-(3-fluorophenyl)pyrrolidine-3-carboxylic acid
5-butyl-1'-{[1-(propan-2-yl)-1H-imidazol-2-yl]methyl}-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-3-(3-hydroxy-3-methylbut-1-yn-1-yl)-N-methylbenzamide
(1S,9S)-11-[2-(4-acetyl-3,5-dimethyl-1H-pyrazol-1-yl)acetyl]-7,11-diazatricyclo[7.3.1.02,7]trideca-2,4-dien-6-one
3-(2,3-dihydro-1H-inden-2-yl)-1-(2-methylpropyl)-8-{[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
(5S,9aS,9bS)-5-(2-methylphenyl)-2-(2-phenylethyl)-octahydro-1H-pyrrolo[3,4-h]pyrrolizin-1-one
N-{2-[(5,8-dimethoxy-4-methylquinolin-2-yl)amino]ethyl}methanesulfonamide
1-ethyl-3-(2-methylpropyl)-N-(oxan-4-yl)-1H-pyrazole-5-carboxamide
(1R,3S)-7-{2-amino-5H,6H,7H-cyclopenta[d]pyrimidin-4-yl}-7-azaspiro[3.5]nonane-1,3-diol
1-{1,6-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl}-3-(1-methyl-1H-imidazole-2-carbonyl)piperidine
1-ethyl-3-methyl-5-(3-phenyl-1H-pyrazol-4-yl)-1H-1,2,4-triazole
3-{1-[(3-methyl-1-propyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl}-N-(oxolan-2-ylmethyl)propanamide