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N-(propan-2-yl)-3-[5-(3,3,4,4-tetrafluorobutyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl]propanamide
N-[4-(4-{[(1,3-dimethyl-1H-pyrazol-4-yl)methyl](methyl)amino}piperidin-1-yl)phenyl]-2,4-dimethylbenzamide
N-[(1,2-dimethyl-1H-1,3-benzodiazol-5-yl)methyl]-3-[(4S)-2,5-dioxoimidazolidin-4-yl]propanamide
2-[4-(1-benzyl-1H-imidazol-2-yl)piperidin-1-yl]-4-methylpyrimidine
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}-3-(4,5,6,7-tetrahydro-1H-indazol-3-yl)propanamide
N-({2-[cyclohexyl(methyl)amino]pyridin-3-yl}methyl)-5,6-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
2-[(4aR,8aR)-octahydro-2H-1,4-benzoxazin-4-ylmethyl]-3,5-dimethoxybenzoic acid
1'-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-5-methyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
(3aS,6aS)-2-[3-(dimethylamino)benzoyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
3-{[8-(2-methylquinolin-4-yl)-1,8-diazaspiro[4.5]decan-1-yl]methyl}pyridin-2-amine
8-(4-methylpyridin-2-yl)-2-[2-(pyridin-2-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
3-(4-fluoro-3-methylphenyl)-1-methyl-6-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
1-{4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}-2-phenylethan-1-one
methyl[(5-methyl-1H-pyrazol-3-yl)methyl]{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}amine
1-[3-(2-methylphenyl)-3-phenylpropanoyl]piperidine-4-carboxamide
2-{2-[2-(2-aminoethyl)morpholin-4-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
(3R,4S)-1-(1-methyl-4,5,6,7-tetrahydro-1H-indazole-3-carbonyl)-4-(propan-2-yl)pyrrolidin-3-amine
(4aS,8aS)-2-(3-fluoropyridin-2-yl)-decahydro-2,7-naphthyridin-4a-ol
4-(difluoromethoxy)-N-methyl-N-{[3-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
1-[3-(5-methyl-4H-1,2,4-triazol-3-yl)phenyl]-3-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}urea
N-(3-methyl-1,2-thiazol-5-yl)-3-({methyl[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]amino}methyl)benzamide
6-[7-(cyclohexylmethyl)-2,7-diazaspiro[4.5]decane-2-carbonyl]-2,3-dihydropyridazin-3-one
3-[1-(2-methoxyphenyl)-3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]-6-methyl-1,2-dihydropyridin-2-one
7-chloro-3-{[(6-hydroxy-6-methylheptan-2-yl)amino]methyl}-1-(2-phenoxyethyl)-1,2-dihydroquinolin-2-one
2-(4-{[1-benzyl-2-(ethanesulfonyl)-1H-imidazol-5-yl]methyl}piperazin-1-yl)pyrazine
5-ethyl-N-[1-(1-ethyl-1H-1,2,4-triazol-5-yl)ethyl]-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-amine
3-(2-ethylbutyl)-8-(2-methoxypyridine-3-carbonyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
6-({[1,3-dimethyl-6-(pyridin-2-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]amino}methyl)pyrimidin-4-ol
N-[(5-methylpyrazin-2-yl)methyl]-5-phenyl-1,2-oxazole-3-carboxamide
N-[(1-ethylpyrrolidin-2-yl)methyl]-2-[3-(trifluoromethyl)phenoxymethyl]-1,3-oxazole-4-carboxamide
1-{4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-1-yl}-4-(1H-pyrazol-1-yl)butan-1-one
2-{[(2,2-dimethyloxan-4-yl)(methyl)amino]methyl}-3,5-dimethoxybenzoic acid
methyl 7-oxo-9-[2-(thiophen-2-yl)ethoxy]-3-[2-(1H-1,2,4-triazol-1-yl)acetyl]-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxylate
2-[(dimethylcarbamoyl)amino]-N-[2-(1H-1,2,4-triazol-5-ylsulfanyl)ethyl]acetamide
N-({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)-N-(2-methoxyethyl)-2-(1H-pyrazol-1-yl)acetamide
3-(1H-indol-3-yl)-1-[3-(naphthalene-2-carbonyl)piperidin-1-yl]propan-1-one
2-[1-({1-[2-(methylsulfanyl)pyrimidin-4-yl]piperidin-3-yl}methyl)-1H-1,2,3-triazol-4-yl]ethan-1-ol
(4aS,8aR)-1-[2-(1H-imidazol-4-yl)ethyl]-6-(2-phenoxyacetyl)-decahydro-1,6-naphthyridin-2-one
1-(methoxymethyl)-N-[(3R,4S)-1-(3-methylpyrazin-2-yl)-4-propylpyrrolidin-3-yl]cyclopropane-1-carboxamide
3-[(diethylamino)methyl]-N-(1,3,4-thiadiazol-2-yl)benzamide
7-(cyclopropylmethyl)-2-(5-methoxy-4-oxo-4H-pyran-2-carbonyl)-2,7-diazaspiro[4.5]decan-6-one
4-(hydroxymethyl)-1-{[2-(3-methoxyphenyl)-1,3-thiazol-5-yl]methyl}piperidin-4-ol
5-[(2R)-2-(methoxymethyl)pyrrolidine-1-carbonyl]-1H-imidazole-4-carboxylic acid
propan-2-yl 3-{[2-(2-aminoethyl)morpholine-4-carbonyl]amino}-4-chlorobenzoate
2-[methyl(2-phenylethyl)amino]-N-[(5-methyl-1,2-oxazol-3-yl)methyl]-2,3-dihydro-1H-indene-2-carboxamide
N-[1-(4-methyl-5-{[(2-methylphenyl)methyl]sulfanyl}-4H-1,2,4-triazol-3-yl)ethyl]-2-(thiophen-3-yl)acetamide
methyl 4-[4-(2-methyl-6-oxo-1,6-dihydropyrimidine-5-carbonyl)piperazin-1-yl]benzoate
(2S,4R)-4-(1H-1,3-benzodiazol-2-ylsulfanyl)-N-(1-benzothiophen-2-ylmethyl)-N-methyl-1-(pyridin-4-ylmethyl)pyrrolidine-2-carboxamide
methyl 4-{4-[3-oxo-3-(pyrrolidin-1-yl)propyl]piperidine-1-carbonyl}benzoate
{[2-(2-methylphenoxy)pyridin-3-yl]methyl}({[1-(pyridin-2-yl)-1H-pyrrol-2-yl]methyl})amine