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2-(1-{[1-(1-methyl-1H-pyrrole-2-carbonyl)piperidin-4-yl]methyl}-1H-1,2,3-triazol-4-yl)pyridine
(1S,5R)-3-[(2-aminopyridin-3-yl)methyl]-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonan-7-one
5-cyclohexaneamido-1-(2-methoxyethyl)-N-({5-methylimidazo[1,2-a]pyridin-2-yl}methyl)-1H-1,3-benzodiazole-7-carboxamide
2-(4-ethylpiperazin-1-yl)-N-(2-methoxyethyl)-N-methyl-2,3-dihydro-1H-indene-2-carboxamide
(1S,5R)-3-[(4-methoxyphenyl)methyl]-6-(pyridine-2-carbonyl)-3,6-diazabicyclo[3.2.2]nonane
N-(2,5-dimethylphenyl)-N'-{3-[2-(hydroxymethyl)piperidin-1-yl]propyl}propanediamide
N-(2-fluoroethyl)-1-[1-(3-phenylpropyl)piperidin-4-yl]piperidine-4-carboxamide
2-(pyridin-3-yl)-N-[2-(4H-1,2,4-triazol-4-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
2-cyclopropyl-5-[4-(pyridin-3-ylmethoxy)piperidine-1-carbonyl]pyrimidin-4-ol
(2S,4R)-4-[4-(2-methoxyphenyl)-1H-1,2,3-triazol-1-yl]-N-(propan-2-yl)pyrrolidine-2-carboxamide
1-[(3-methyl-1-phenyl-1H-pyrazol-4-yl)methyl]-4-(pyridin-4-ylmethyl)-1,4-diazepane
3-[(3-cyclopentaneamidophenyl)formamido]-4,4,4-trifluorobutanoic acid
1-{2-amino-4-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-3-(1H-indol-3-yl)propan-1-one
1-{[3-(2-methylpropyl)-1H-1,2,4-triazol-5-yl]methyl}-1,2,3,6-tetrahydropyridazine-3,6-dione
1-{[4-(benzyloxy)phenyl]methyl}-3-(methanesulfonylmethyl)piperidine
2-cyclopropanecarbonyl-8-[(2E)-3-phenylprop-2-enoyl]-2,8-diazaspiro[4.5]decane-3-carboxylic acid
2-[1-(2-chlorophenyl)-5-[1-(4-methyl-1H-pyrazol-1-yl)ethyl]-1H-1,2,4-triazol-3-yl]acetamide
(3S,4R)-1-(1-methyl-1H-indole-3-carbonyl)-4-(pyridin-4-yl)pyrrolidine-3-carboxylic acid
({3-[(4-ethylpiperazin-1-yl)methyl]-2,5-dimethylphenyl}methyl)[2-(1H-imidazol-1-yl)ethyl]methylamine
N-[(2-chloropyridin-3-yl)methyl]-N,2-dimethyl-6-(piperidin-3-yl)pyrimidin-4-amine
3-[(3S,4R)-1-(pyridin-3-ylmethyl)-4-{4-[3-(trifluoromethyl)phenyl]piperazin-1-yl}piperidin-3-yl]-1-(1,2,3,4-tetrahydroisoquinolin-2-yl)propan-1-one
3-{[1-(2-{imidazo[2,1-b][1,3]thiazol-6-yl}acetyl)pyrrolidin-3-yl]methyl}benzamide
1-[3-(3-fluoro-4-phenylbenzoyl)piperidin-1-yl]-2-methoxyethan-1-one
4-(4-fluorophenoxy)-1-(thiophene-3-carbonyl)piperidine-4-carboxylic acid
N-[(4-hydroxy-1-methylpiperidin-4-yl)methyl]-5-[(5,6,7,8-tetrahydronaphthalen-2-yloxy)methyl]-1,2-oxazole-3-carboxamide
2-[2-(1H-1,3-benzodiazol-1-yl)ethyl]-5-(4-methyl-1,4-diazepan-1-yl)-2,3-dihydropyridazin-3-one
N-[(1-hydroxycyclohexyl)methyl]-5-[(4-hydroxypiperidin-1-yl)methyl]-1,2-oxazole-3-carboxamide
2-amino-4-(2,2-difluoro-2H-1,3-benzodioxol-4-yl)-6-(2-hydroxypropan-2-yl)pyridine-3-carbonitrile
1-(5,6-dimethylpyrimidin-4-yl)-3',4'-dihydro-1'H-spiro[piperidine-4,2'-quinoxaline]-3'-one
N-ethyl-N-(2-hydroxyethyl)-2-{3-oxo-1-[(2E)-3-phenylprop-2-en-1-yl]piperazin-2-yl}acetamide
N-[(3S,4S)-4-hydroxy-1,1-dioxo-1λ6-thiolan-3-yl]-N-methyl-1-benzothiophene-2-carboxamide
1-[4-(4-methoxyphenyl)-2-methylpiperazin-1-yl]-3-(5-methyl-1H-pyrazol-1-yl)propan-1-one
5-{[9-(cyclopropylmethyl)-1-methyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl]methyl}-1,2,4-oxadiazole-3-carboxamide
9-(4-chloro-2-methylbenzoyl)-2-(propan-2-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-(3-fluorophenyl)-N-[2-(4-methoxyphenyl)ethyl]-1,3-benzoxazole-5-carboxamide
(3S,4S)-1-{5-ethyl-2,3-dimethylpyrazolo[1,5-a]pyrimidin-7-yl}-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
2-amino-6-(3,4-dimethylphenyl)-4-[1-(2-hydroxyethyl)-3-methyl-1H-pyrazol-4-yl]pyridine-3-carbonitrile
5-ethoxy-N-methyl-N-[(4-methyl-1H-imidazol-2-yl)methyl]furan-2-carboxamide
2-(2-hydroxyethyl)-9-[(6-methyl-1H-1,3-benzodiazol-2-yl)methyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(3-hydroxy-3-methylbutyl)-N-methyl-N-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]benzamide
1-[2-(4-methoxyphenyl)ethyl]-5-(3-methyl-1,2,4-oxadiazol-5-yl)piperidin-2-one
N-[(2,3-dimethyl-1H-indol-5-yl)methyl]-2,4-dimethoxybenzamide
3-(2-fluorophenyl)-5-{spiro[2.5]octane-1-carbonyl}-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine
7-(cyclopropylmethyl)-2-(pyrimidin-2-yl)-2,7-diazaspiro[4.5]decane
(4aS,8aS)-2-cyclopentanecarbonyl-7-(1-methyl-1H-pyrazole-3-carbonyl)-decahydro-2,7-naphthyridin-4a-ol
1-tert-butyl-N-[3-(4-chlorophenyl)propyl]-5-oxopyrrolidine-3-carboxamide
4-[4-(2,6-dimethylpyridin-4-yl)piperazine-1-carbonyl]-5,6,7,8-tetrahydroquinazolin-2-amine
N-[2-(1-methylpiperidin-3-yl)ethyl]-5-phenyl-1H-pyrrole-2-carboxamide
methyl(1,2-oxazol-3-ylmethyl)[(4-{[1-(1,3-thiazole-5-carbonyl)piperidin-3-yl]methoxy}phenyl)methyl]amine
4-[(1-acetylpiperidin-4-yl)amino]-1-[2-(4-fluorophenyl)ethyl]pyrrolidin-2-one