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[(1-benzylpiperidin-4-yl)methyl]({3-[(3-fluorophenyl)methyl]-1,2,4-oxadiazol-5-yl}methyl)methylamine
1-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-1-yl]-2-(4-hydroxyphenyl)ethan-1-one
3-({1-[(5-methylthiophen-2-yl)methyl]piperidin-4-yl}oxy)-N-(pyridin-2-ylmethyl)benzamide
3-(2H-1,3-benzodioxol-5-ylmethyl)-N-(2,3-dihydro-1H-inden-1-yl)-4,5-dihydro-1,2-oxazole-5-carboxamide
1-[3-(2-methoxyethyl)-5-[4-(2-methyl-2H-1,2,3,4-tetrazol-5-yl)phenyl]-1H-1,2,4-triazol-1-yl]butan-2-ol
N-{4-chloro-3-[(propan-2-yl)carbamoyl]phenyl}-2-(ethoxymethyl)pyrrolidine-1-carboxamide
(2S,4S)-4-[2-(3-chlorophenyl)acetamido]-1-cyclopentyl-N-ethylpyrrolidine-2-carboxamide
N-({4-methoxy-3-[(3-methyloxetan-3-yl)methoxy]phenyl}methyl)-N-(oxolan-2-ylmethyl)-3-(2-oxopyrrolidin-1-yl)benzamide
5-(5-chloro-2-methoxypyridin-4-yl)-4-methylpyridin-2-amine
N-{[(3S,4S)-3-hydroxy-1-[2-(4-methyl-1,2,5-oxadiazol-3-yl)acetyl]piperidin-4-yl]methyl}furan-2-carboxamide
3-{5H,6H,7H,8H,9H-[1,2,3,4]tetrazolo[1,5-a]azepin-9-ylformamido}-N-(1,3-thiazol-2-yl)propanamide
5-{4-[1-(pyrrolidin-1-yl)ethyl]phenyl}pyrimidin-2-amine
N-[2-(2-methoxyphenyl)ethyl]-[1,2,4]triazolo[4,3-a]pyridine-7-carboxamide
(2R,6R)-6-methyl-2-(prop-2-en-1-yl)-1-{[3-(3,4,5-trimethoxyphenyl)-1H-pyrazol-4-yl]methyl}-1,2,3,6-tetrahydropyridine
4-(1H-1,3-benzodiazol-2-yl)-N-[(2-methylpyrimidin-5-yl)methyl]aniline
1-{1-azabicyclo[2.2.2]octan-3-yl}-3-(7-methyl-2,3-dihydro-1,4-benzodioxin-6-yl)urea
2-(2-butylpyrimidin-5-yl)-4-(4-methylpiperazine-1-carbonyl)quinoline
(3S,4R)-1-[(2-butyl-1H-imidazol-4-yl)methyl]-N,N-dimethyl-4-propylpyrrolidin-3-amine
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-1-[4-methyl-6-(methylamino)pyrimidin-2-yl]piperidin-3-ol
1-{[2-(furan-3-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-4-phenyl-1,4-diazepane
1-phenyl-N-({1-[2-(pyrrolidin-1-yl)acetyl]piperidin-3-yl}methyl)methanesulfonamide
N-benzyl-5-(2-chloro-4-fluorophenoxymethyl)-N-methyl-1,2-oxazole-3-carboxamide
5-(4-acetylphenoxymethyl)-N-(pyrrolidin-3-ylmethyl)-1,2-oxazole-3-carboxamide
2-(5-cyano-1H-indol-1-yl)-N-(1-methyl-4-phenyl-1H-pyrazol-5-yl)acetamide
9-ethyl-1-methyl-10-oxo-N-(2-phenylethyl)-1,4,9-triazaspiro[5.6]dodecane-4-carboxamide
1-{5-[(2,6-difluorophenyl)methyl]-1-(2-phenylethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carbonyl}piperidin-4-ol
2-propyl-N-{[2-(pyrrolidin-1-yl)-1,3-thiazol-4-yl]methyl}-1,3-thiazole-4-carboxamide
6-(2-chlorophenyl)-N-[2-(diethylamino)ethyl]-N-ethylimidazo[2,1-b][1,3]thiazole-3-carboxamide
N-[3-(2-amino-1,3-thiazol-4-yl)propyl]-3-(1H-pyrazol-1-yl)benzamide
N-[2-(4,6-dimethylpyrimidin-2-yl)ethyl]-1-methyl-3-(2-methylpropyl)-1H-pyrazole-5-carboxamide
1-(3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4-(thiophen-2-ylmethyl)piperazine
1-(1-{[5-(4-chlorophenyl)furan-2-yl]methyl}piperidin-4-yl)-N-(2-hydroxyethyl)-1H-1,2,3-triazole-4-carboxamide
5-[(4-hydroxypiperidin-1-yl)methyl]-N-[(2-methoxyphenyl)methyl]-N-methyl-1,2-oxazole-3-carboxamide
N-[1-(cyclohexylmethyl)-5-oxopyrrolidin-3-yl]-3-(methylsulfanyl)propanamide
(4aS,7aR)-1-[3-(propan-2-yl)-1H-pyrazole-5-carbonyl]-4-propanoyl-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[2-(5-methyl-1,3,4-thiadiazol-2-yl)ethyl]-3-(5-methylthiophen-2-yl)-1H-pyrazole-5-carboxamide
1-cyclopentyl-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
3-{[3-(2-ethylphenoxy)azetidin-1-yl]methyl}pyridine
2-{1-[(2,3-dimethoxyphenyl)methyl]-3-oxopiperazin-2-yl}-N-(2-methylpropyl)acetamide
N-(4-{[(3R,4R)-3-hydroxy-4-{methyl[2-(pyridin-2-yl)ethyl]amino}piperidin-1-yl]methyl}phenyl)acetamide
2-(1H-indol-3-yl)-N-[2-(pyrrolidin-1-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-4-amine
7-chloro-N-(2-methoxyethyl)-2-methyl-N-(pyridin-4-ylmethyl)quinoline-4-carboxamide
8-(3-cyano-5,6,7,8-tetrahydroquinolin-2-yl)-2-oxo-1,8-diazaspiro[4.5]decane-4-carboxylic acid
ethyl 2-[(3-{[1-(cyclohex-1-en-1-yl)ethyl]carbamoyl}phenyl)amino]acetate
2-(ethylamino)-N-[1-(1-methyl-1H-pyrazol-5-yl)propyl]pyrimidine-5-carboxamide
N-(5-chloro-2-{8-methyl-octahydro-1H-pyrazino[1,2-a]piperazine-2-carbonyl}phenyl)propanamide
1-[(3-phenyloxolan-3-yl)methyl]-4-(pyridin-3-yl)piperazine
3-(3-fluoro-4-methoxyphenyl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
N,N-diethyl-4-[(4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}piperidin-1-yl)methyl]aniline
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-2-(pyridin-4-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine