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(3S,4S)-3,4-dihydroxy-N-pentylpiperidine-1-carboxamide
(3aS,6aS)-3a-(hydroxymethyl)-N-(4-methyl-2-oxo-2H-chromen-7-yl)-octahydrocyclopenta[c]pyrrole-2-carboxamide
1-methyl-4-{4-[1-(naphthalen-2-yl)-1H-1,2,4-triazol-5-yl]butan-2-yl}piperazine
1-(2-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl}-2-oxoethyl)-5-methyl-1,2,3,4-tetrahydropyrimidine-2,4-dione
(2R)-N-[2-(7-methyl-1H-indol-3-yl)ethyl]oxolane-2-carboxamide
(3S,4S)-1-({3-[(2-methylprop-2-en-1-yl)oxy]phenyl}methyl)-4-(pyrrolidin-1-yl)pyrrolidin-3-ol
N-[1-phenyl-3-(1H-1,2,4-triazol-1-yl)propyl]thian-4-amine
8-[3-(propan-2-yl)-4,5-dihydro-1,2-oxazole-5-carbonyl]-2,8-diazaspiro[4.5]decan-3-one
N-(oxolan-3-yl)-3-(thiomorpholine-4-carbonyl)benzene-1-sulfonamide
ethyl 2-{1-[(2-fluorophenyl)carbamoyl]piperidin-2-yl}acetate
1-(3-methylpyridin-4-yl)-4-(1H-pyrazole-4-carbonyl)piperazine
2-amino-4-ethyl-N-[(4-methyl-1,4-oxazepan-6-yl)methyl]-1,3-thiazole-5-carboxamide
3-[(1R)-2,3-dihydro-1H-inden-1-yl]-1-(4-ethyl-3-oxo-3,4-dihydro-2H-1,4-benzoxazin-6-yl)urea
1-{4-[3-({[2-(3-chlorophenyl)ethyl]amino}methyl)-7-(methylsulfanyl)quinolin-2-yl]piperazin-1-yl}ethan-1-one
3,6-dimethyl-N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-[1,2]oxazolo[5,4-b]pyridine-4-carboxamide
N-ethyl-9-oxo-8-(pyridin-2-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxamide
N-{1H,4H,5H,6H-cyclopenta[c]pyrazol-3-ylmethyl}-3-(1H-1,2,3,4-tetrazol-1-yl)-1H-pyrazole-4-carboxamide
N-{[2-(propan-2-yl)-1,3-thiazol-4-yl]methyl}-5-[(quinolin-8-yloxy)methyl]-1,2-oxazole-3-carboxamide
[(4-ethoxyphenyl)methyl]({1-[2-(4-methoxyphenyl)ethyl]piperidin-4-yl}methyl)methylamine
N-{5-[2-(hydroxymethyl)phenyl]quinolin-8-yl}acetamide
(4S)-4-(propan-2-yl)-3-{[1,2,4]triazolo[1,5-a]pyrimidin-2-ylmethyl}-1,3-oxazolidin-2-one
1-(6-methoxy-2,3-dihydro-1H-indene-5-carbonyl)-1,4-diazepan-6-ol
N-[3-({[3-(4H-1,2,4-triazol-4-yl)propyl]carbamoyl}amino)phenyl]cyclopentanecarboxamide
1-[(3R,4R)-3-{[(2-hydroxyethyl)(methyl)amino]methyl}-4-(hydroxymethyl)pyrrolidin-1-yl]-2-(4-phenylpiperidin-1-yl)ethan-1-one
2-methyl-N-[4-(pyridin-2-yl)butyl]-3-[(pyridin-2-ylmethyl)amino]benzamide
2-(2-methylphenyl)-1-{3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidin-1-yl}ethan-1-one
2-(3-{2-[2-(thiophen-2-yl)ethyl]piperidine-1-carbonyl}phenoxy)acetamide
2-(2-{5H,6H,7H,8H,9H-imidazo[1,5-a][1,4]diazepin-8-ylmethyl}-1H-pyrrol-1-yl)-1,3-thiazole
1-[(3aS,6aS)-octahydropyrrolo[2,3-c]pyrrol-1-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
ethyl 2-{methyl[5-({[(3R)-oxolan-3-yl]amino}methyl)pyrimidin-2-yl]amino}acetate
5-cyclobutyl-N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N-methyl-1,3,4-oxadiazol-2-amine
1-[(2,2-dimethyloxan-4-yl)methyl]-4-(3-methylpyridin-4-yl)-1,4-diazepane
1-methyl-3-{1-[(2-methyl-1,3-oxazol-4-yl)methyl]piperidin-3-yl}-4-phenyl-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[3-(1H-imidazol-1-yl)propyl]-2-methyl-1-benzofuran-5-carboxamide
4-(1-{[1-(propan-2-yl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)benzoic acid
2-(2-{[(3aR,6aS)-5-methyl-octahydropyrrolo[3,4-c]pyrrol-2-yl]methyl}phenoxy)ethan-1-ol
2-(dimethylamino)-N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-methylpyrimidine-5-carboxamide
1-{5-[(6-methoxypyrimidin-4-yl)amino]-7,7-dimethyl-5,6,7,8-tetrahydroquinazolin-2-yl}piperidin-4-ol
N-[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]-2-(1H-1,2,3,4-tetrazol-5-yl)benzamide
3-butanamido-N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-N,4-dimethylbenzamide
5-{[2-(1-ethylpiperidin-4-yl)acetamido]methyl}-N,N-dimethylfuran-2-carboxamide
N-methyl-N-[2-(pyridin-2-yl)ethyl]-3-[1-(4,4,4-trifluorobutanoyl)piperidin-3-yl]propanamide
7-oxo-2-(pyridine-4-amido)-N-{[2-(trifluoromethoxy)phenyl]methyl}-4,5,6,7-tetrahydro-1,3-benzothiazole-5-carboxamide
5-({3-[4-(4-fluorophenyl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-N,N-dimethylpyrimidin-2-amine
5-[(2-methyl-1H-1,3-benzodiazol-1-yl)methyl]-N-[2-(pyridin-3-yloxy)ethyl]-1H-pyrazole-3-carboxamide
4-(1H-1,3-benzodiazol-1-yl)-1-(2,1,3-benzoxadiazol-4-ylmethyl)piperidine-4-carboxylic acid
3-methyl-1-{4-[(1-methylpiperidin-4-yl)oxy]phenyl}-3-[(3-propyl-1,2,4-oxadiazol-5-yl)methyl]urea
3-(2H-1,3-benzodioxol-5-ylmethyl)-1-[1-(2-methoxyethyl)piperidine-4-carbonyl]-3-methylpiperidine
3-methyl-8-[2-(methylsulfanyl)pyrimidin-4-yl]-1-oxa-3,8-diazaspiro[4.6]undecan-2-one
6-(1-acetylpiperidine-3-carbonyl)-N,N,1-trimethyl-1H,4H,5H,6H,7H-pyrrolo[2,3-c]pyridine-2-carboxamide