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4-(1-benzyl-1H-imidazol-2-yl)-1-[1-(1H-pyrazol-1-ylmethyl)cyclopropanecarbonyl]piperidine
methyl({[3-(1H-pyrazol-1-yl)phenyl]methyl}){[3-(thiophen-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amine
methyl({[5-methyl-2-(naphthalen-1-yl)-1,3-oxazol-4-yl]methyl})[1-(1,2-oxazol-3-yl)ethyl]amine
1-(naphthalene-1-carbonyl)-4-[2-(pyrrolidin-1-yl)ethyl]-1,4-diazepan-5-one
2-[4-(cyclopropylmethyl)-1-[1-(propan-2-yl)piperidin-4-yl]piperazin-2-yl]ethan-1-ol
N-[1-(dimethyl-1,3-thiazol-4-yl)ethyl]-N-methyl-1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carboxamide
2-(4-chloro-3,5-dimethyl-1H-pyrazol-1-yl)-N-[(3-ethyl-1,2-oxazol-5-yl)methyl]-N-methylacetamide
5-[3-(2-chlorophenoxy)azetidine-1-carbonyl]-2,4-dimethylpyridine
methyl (2S)-2-phenyl-2-{[3-(2-phenylethyl)-1,2-oxazol-5-yl]formamido}acetate
9-[(2S)-2-hydroxy-3-phenylpropanoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
2-benzyl-N-(2-oxooxolan-3-yl)-1,3-thiazole-4-carboxamide
4-({5-ethylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-N,N-dimethylbutanamide
1-{4-[(3-fluorophenyl)methyl]piperazin-1-yl}-3-(1H-1,2,3,4-tetrazol-1-yl)propan-1-one
2-{4-[2-amino-3-cyano-5-ethyl-6-(propan-2-yl)pyridin-4-yl]-2-methoxyphenoxy}acetamide
4-(5-{[ethyl({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amino]methyl}thiophen-2-yl)-2-methylbut-3-yn-2-ol
1-(2-methoxyethyl)-3-(naphthalen-1-ylmethyl)-8-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
[1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidin-4-yl](1-methyl-1H-imidazol-2-yl)methanol
6-(methoxymethyl)-N-[2-(2-methyl-1H-indol-1-yl)ethyl]pyrimidin-4-amine
1-{dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}-4-(3-methoxybenzoyl)piperazine
2-({[2-methoxy-1-(pyridin-2-yl)ethyl](methyl)amino}methyl)-6,8-dimethylquinolin-4-ol
N-[(3R,4S)-1-(carbamoylmethyl)-4-cyclopropylpyrrolidin-3-yl]-4-(pyrrolidin-1-yl)benzamide
N-(1-cycloheptylpiperidin-3-yl)-4-methyl-1,2,5-oxadiazole-3-carboxamide
N-[4-(1-ethyl-1H-1,2,4-triazol-5-yl)-7-methoxy-2-oxo-1,2,3,4-tetrahydroquinolin-6-yl]-3-methylbutanamide
4-[(1-methanesulfonylpiperidin-4-yl)oxy]-N-(2-phenylethyl)benzamide
9-(2-ethoxypropanoyl)-2-[2-(1H-imidazol-4-yl)ethyl]-2,9-diazaspiro[5.5]undecan-3-one
3-(1-{2-[4-(methylsulfanyl)phenyl]acetyl}piperidin-3-yl)-1-(pyrrolidin-1-yl)propan-1-one
1-(2-methoxyethyl)-3-[(3-methoxyphenyl)methyl]-8-(quinoxalin-5-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{2-[9-(2-hydroxyethyl)-7-(hydroxymethyl)-3,9-diazaspiro[5.5]undecan-3-yl]-2-oxoethyl}acetamide
1-[(1-{[2-(ethanesulfonyl)-1-(2-methoxyethyl)-1H-imidazol-5-yl]methyl}piperidin-3-yl)methyl]pyrrolidin-2-one
1-(3-{[1-(3-hydroxyphenyl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenyl)ethan-1-one
N-[(1-methyl-4-phenylpiperidin-4-yl)methyl]-2,3,4,5-tetrahydro-1-benzoxepine-4-carboxamide
dimethyl(2-{2-[1-(2-methylpyrimidine-5-carbonyl)piperidin-3-yl]-1H-imidazol-1-yl}ethyl)amine
N-[(3R,4S)-1-methanesulfonyl-4-propylpyrrolidin-3-yl]-3-(1H-pyrazol-4-yl)propanamide
2-[4-(5-tert-butyl-1,3,4-oxadiazol-2-yl)piperazin-1-yl]benzonitrile
2-hydroxy-5-{[(3-phenylprop-2-yn-1-yl)(propyl)amino]methyl}benzoic acid
N-(cyclohexylmethyl)-5-(2-methylphenyl)-1,2,4-triazin-3-amine
N-[(2S)-4-(methylsulfanyl)-1-oxo-1-{4-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidin-1-yl}butan-2-yl]acetamide
(1R,2R,6S,7S)-4-(2,3-dihydro-1H-isoindole-1-carbonyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
(4aS,8aR)-1-[2-(pyridin-2-yl)ethyl]-6-(pyridin-4-yl)-decahydro-1,6-naphthyridin-2-one
2-({[2-(2-fluorophenyl)ethyl]amino}methyl)-4-(6-methoxypyridin-2-yl)phenol
1-[(3R,4S)-3-amino-4-cyclopropylpyrrolidin-1-yl]-3-(4-hydroxyphenyl)propan-1-one
1-methyl-4-{[3-(2-phenylethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-7-yl]methyl}-1H-pyrazole
N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}-1H-pyrrolo[2,3-b]pyridin-6-amine
(4aS,8aR)-6-[4-(trifluoromethyl)benzoyl]-decahydro-1,6-naphthyridine-4a-carboxylic acid
4-phenyl-3-[1-(pyridin-4-ylmethyl)piperidin-3-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(3-{[4-(hydroxymethyl)phenyl]methyl}pyrrolidine-1-carbonyl)-6-methyl-4H-pyran-4-one
N-[(3R,5S)-5-(hydroxymethyl)-1-methylpyrrolidin-3-yl]-4-phenoxybenzamide
(3R,4S)-1-(4-chloro-1-ethyl-1H-pyrazole-5-carbonyl)-4-cyclopropylpyrrolidin-3-amine
N-ethyl-2-[2-(1H-imidazol-1-yl)acetamido]-4,5,6,7-tetrahydro-1-benzothiophene-3-carboxamide
N-cyclopentyl-2-({2-[2-(pyrimidin-2-yl)-1,3-thiazol-4-yl]ethyl}amino)propanamide