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3-[4-(1-ethoxyethyl)phenyl]-N,N-dimethyl-1H-1,2,4-triazol-5-amine
5-{4-[(3-methoxyphenyl)methyl]piperazine-1-carbonyl}-1-(3-methylbutyl)-N-(2-methylpropyl)-4-oxo-1,4-dihydropyridine-3-carboxamide
2-{4-[4-(methylamino)pyrimidin-2-yl]-1H-pyrazol-1-yl}-N-[1-(thiophen-2-ylmethyl)-1H-pyrazol-5-yl]acetamide
5-{3-[4-(1,3-benzoxazol-2-yl)-1,4-diazepan-1-yl]-3-oxopropyl}-5-ethylpyrrolidin-2-one
2-{4-[(3,5-difluorophenyl)methyl]-1-[(2-ethoxyphenyl)methyl]piperazin-2-yl}ethan-1-ol
1-(2-methylpyrimidin-4-yl)-4-(morpholine-4-carbonyl)-1,4-diazepane-6-carboxylic acid
6-(5-chloro-2-methoxypyridin-4-yl)-N-methylpyridine-2-carboxamide
N-({1-[2-(dimethylamino)benzoyl]piperidin-3-yl}methyl)-4-methoxybenzene-1-sulfonamide
3-(4-methoxy-2-methylbenzoyl)-1-(thiophene-3-sulfonyl)piperidine
N-{[2-(3-hydroxypiperidin-1-yl)pyridin-3-yl]methyl}-4-methyl-2-(propan-2-yl)pyrimidine-5-carboxamide
1-[(3-methoxyphenyl)methyl]-5-{[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]methyl}-1H-1,2,4-triazole
N-{2-[4-(1-methylpiperidin-4-yl)morpholin-2-yl]ethyl}cyclohexanecarboxamide
2-(3-ethoxypropanoyl)-7-methyl-2,7-diazaspiro[4.5]decan-6-one
1-[2-({[3-(furan-2-yl)-1,2,4-oxadiazol-5-yl]methyl}amino)ethyl]imidazolidin-2-one
4-hydroxy-N-[3-hydroxy-1-(4-methylphenyl)propyl]-2-(3-methylphenyl)pyrimidine-5-carboxamide
{[3-(2H-1,3-benzodioxol-5-yl)-1,2,4-oxadiazol-5-yl]methyl}(methyl)[4-(morpholin-4-yl)butyl]amine
2-methyl-5-(2-{2-[4-(1,3-thiazol-2-yl)-1H-1,2,3-triazol-1-yl]ethyl}morpholin-4-yl)-2,3-dihydropyridazin-3-one
1-{1-[(6-ethyl-2-oxo-2H-chromen-4-yl)methyl]piperidin-3-yl}pyrrolidin-2-one
2-({[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)amino)-N-methylacetamide
1-[(4S,4aS,8aS)-4-hydroxy-4-phenyl-decahydroquinolin-1-yl]-4-(1H-imidazol-1-yl)butan-1-one
1-[(3S)-3-(dimethylamino)azepan-1-yl]-2-[(1-methyl-1H-indol-3-yl)sulfanyl]ethan-1-one
3-butyl-1-methyl-4-{[3-(trifluoromethyl)-1,2,4-oxadiazol-5-yl]methyl}piperazin-2-one
N-(prop-2-en-1-yl)-N-(prop-2-yn-1-yl)-4-{[1-(pyridine-3-carbonyl)piperidin-4-yl]oxy}benzamide
N-[cyclopropyl(6-methylpyridin-2-yl)methyl]-4-(3-hydroxy-3-methylbutyl)benzamide
2-(dimethyl-1,2-oxazol-4-yl)-1-[(3S,4S)-3-hydroxy-4-[methyl(pyridin-3-ylmethyl)amino]pyrrolidin-1-yl]ethan-1-one
methyl[(6-methylquinolin-5-yl)methyl][2-(methylsulfanyl)ethyl]amine
(3R,4R)-4-(2-ethyl-4-methyl-1H-imidazol-5-yl)-1-methyl-N-{pyrazolo[1,5-a]pyrimidin-3-ylmethyl}pyrrolidine-3-carboxamide
1-ethyl-N-{[2-(morpholin-4-yl)-1,3-thiazol-4-yl]methyl}-6-oxopiperidine-3-carboxamide
3-{[(2,3-dihydroxypropyl)(methyl)amino]methyl}-6,7-dimethoxy-1,2-dihydroquinolin-2-one
3-[(3R,4S)-3-amino-4-(propan-2-yl)pyrrolidin-1-yl]-N,N-dimethylpropanamide
5-(8-methoxy-2-methylquinolin-5-yl)furan-2-carboxamide
2-(cyclopropylmethyl)-8-[2-(2-oxo-2,3-dihydro-1,3-benzoxazol-3-yl)ethyl]-2,8-diazaspiro[5.5]undecan-3-one
2-(2H-1,2,3-benzotriazol-2-yl)-1-{4-[(dimethylamino)methyl]-4-hydroxyazepan-1-yl}ethan-1-one
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-4-methoxy-2-methylbenzamide
methyl 4-({[2-(propan-2-yl)-1,3-benzoxazol-5-yl]formamido}methyl)benzoate
2-ethyl-8-[2-(pyridin-3-yl)acetyl]-2,8-diazaspiro[4.5]decan-3-one
4-[5-(methoxymethyl)thiophene-2-carbonyl]-1-[(4-methoxyphenyl)methyl]piperazin-2-one
2-(2,3-dihydro-1H-isoindol-2-yl)-1-[(3S,4R)-3,4-dihydroxy-4-methylpiperidin-1-yl]ethan-1-one
1-(1-methyl-1H-1,2,4-triazol-3-yl)-3-[1-(2-methylpropyl)cyclopropyl]urea
methyl 5-(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-carbonyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxylate
1-[3-(3-ethyl-1,2,4-oxadiazol-5-yl)phenyl]-3-[(3-ethyl-4,5-dihydro-1,2-oxazol-5-yl)methyl]urea
N-[(3,4-difluorophenyl)methyl]-3-[4-(3-methylphenyl)piperazin-1-yl]propanamide
(4aR,7aS)-1-[(4-methyl-1H-imidazol-5-yl)methyl]-4-[2-(3-methyl-1H-pyrazol-1-yl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
3-[1-(5-ethyl-1,3-oxazole-4-carbonyl)piperidin-4-yl]-N-(3-methylphenyl)propanamide
2-[(2H-1,3-benzodioxol-5-yloxy)methyl]-4-{4H,5H,6H,7H-thieno[3,2-c]pyridine-5-carbonyl}-1,3-oxazole
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-methyl-N-[1-(2-phenylethyl)piperidin-3-yl]acetamide
1-[(1S,5R)-3-benzyl-3,6-diazabicyclo[3.2.2]nonan-6-yl]-3-(4-methyl-1H-pyrazol-1-yl)propan-1-one
ethyl 5-[2-(5-carbamoylthiophen-2-yl)pyrrolidine-1-carbonyl]-2,4-dimethyl-1H-pyrrole-3-carboxylate
2-methoxy-1-{4-[(6-methylquinolin-5-yl)methyl]-1,4-diazepan-1-yl}ethan-1-one
5-(4-fluorophenyl)-N-{2-[(3-methyl-1H-1,2,4-triazol-5-yl)sulfanyl]ethyl}-1,2,4-triazin-3-amine