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N-[(1S,3aS,6aS)-octahydropentalen-1-yl]-5-chloro-6-oxo-1,6-dihydropyridine-3-carboxamide
4-{[3-hydroxy-1-(2-methoxyethyl)-2-oxopiperidin-3-yl]methyl}-1-phenylpiperazin-2-one
(4aS,8aR)-1-(2-aminoethyl)-6-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-decahydro-1,6-naphthyridin-2-one
2-{2-[2-(4-methyl-1H-imidazol-5-yl)-1H-imidazol-1-yl]ethyl}-1,2,3,4-tetrahydrophthalazine-1,4-dione
4-(4-methoxy-2-methylphenyl)-3-[1-(propan-2-yloxy)ethyl]-4,5-dihydro-1H-1,2,4-triazol-5-one
6-methyl-N-{3-[(5-methyl-1,3,4-thiadiazol-2-yl)sulfanyl]propyl}pyrazolo[1,5-a]pyrimidine-3-carboxamide
3-(3-fluorophenyl)-6-(oxolane-2-carbonyl)-1-[2-(piperidin-1-yl)ethyl]-1,2,5,6,7,8-hexahydro-1,6-naphthyridin-2-one
(1-{1-[(2-fluoro-5-methoxyphenyl)methyl]piperidin-3-yl}piperidin-4-yl)methanol
N5-(butan-2-yl)-N3-butyl-1-cyclopentyl-N3-methyl-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
N-(2-methylphenyl)-4-[4-(thiomorpholin-4-ylmethyl)-1H-1,2,3-triazol-1-yl]piperidine-1-carboxamide
{5-[(4-methoxy-2,3-dimethylphenyl)methyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-3-yl}methanol
N-[(1-ethyl-3,5-dimethyl-1H-pyrazol-4-yl)methyl]-2-(3-methyl-4,5-dihydro-1H-pyrazol-1-yl)acetamide
3-{2-[4-(3-benzyl-1H-pyrazol-5-yl)piperidin-1-yl]-2-oxoethyl}-1,3-oxazolidin-2-one
4-(2-fluorophenoxy)-1-[(2,4,6-trimethoxyphenyl)methyl]piperidine
3-methyl-8-[3-oxo-3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]-1-oxa-3,8-diazaspiro[4.5]decan-2-one
9-{[3-(difluoromethoxy)phenyl]methyl}-2-ethyl-2,9-diazaspiro[5.5]undecan-3-one
1-(1-methyl-1H-pyrrole-2-carbonyl)-4-phenyl-1,4-diazepane
2-(2,2-dimethylpropanamido)-N-ethyl-5-methyl-N-(pyridin-4-ylmethyl)thiophene-3-carboxamide
7-fluoro-3-methyl-N-[2-(pyridin-3-yloxy)propyl]-1-benzofuran-2-carboxamide
3-[1-(2-methoxybenzoyl)piperidin-4-yl]-1-(4-phenylpiperazin-1-yl)propan-1-one
3-methoxy-2-[(8-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-6-methylpyridine
4-{6-cyclopropyl-3-methyl-[1,2]oxazolo[5,4-b]pyridine-4-carbonyl}piperazine-2-carboxylic acid
2-{1-[(3,4-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-(3-hydroxypropyl)acetamide
5-(2-chloro-4-methoxyphenoxy)-1-azabicyclo[3.2.1]octane
1-methyl-3-[3-(pyridin-4-yl)propyl]-8-(thiolan-3-yl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
methyl 4-{7-[(2-fluoro-5-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-2-yl}-4-oxobutanoate
3-[1-(5-methoxy-1H-indole-2-carbonyl)piperidin-3-yl]-1-(morpholin-4-yl)propan-1-one
1-(4-chlorophenyl)-4-(4-fluoro-2-methylbenzoyl)-5-methylpiperazin-2-one
4-(4-chlorophenyl)-N-[2-(1-oxo-1,2-dihydrophthalazin-2-yl)ethyl]butanamide
(1S,5R)-3-(5-propyl-1,2-oxazole-3-carbonyl)-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-(hydroxymethyl)-N-{[4-(propan-2-yl)-1,2,3-thiadiazol-5-yl]methyl}-1H-1,3-benzodiazole-5-carboxamide
(2S,4R)-N,N-diethyl-4-[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]pyrrolidine-2-carboxamide
2-(3-{1,9-dimethyl-1,4,9-triazaspiro[5.5]undecan-4-yl}-3-oxopropyl)-2,3-dihydro-1H-isoindol-1-one
5-{6-methylpyrazolo[1,5-a]pyrimidin-3-yl}-3-(oxolan-3-yl)-1,2,4-oxadiazole
1-(1-{imidazo[1,2-a]pyrimidine-2-carbonyl}piperidin-4-yl)-2-phenylethan-1-ol
N-[(1,1-dioxo-1λ6-thiolan-3-yl)methyl]-2-(propan-2-yl)-1,3-benzoxazole-5-carboxamide
{2-[3-(morpholin-4-ylmethyl)phenyl]pyridin-4-yl}methanol
2-amino-4-[3-methoxy-4-(pyrrolidin-1-yl)phenyl]-5,6,7,8-tetrahydro-1,6-naphthyridine-3-carbonitrile
N-({6-ethyl-2-methoxy-5-oxo-5H,6H,7H-pyrrolo[3,4-b]pyridin-3-yl}methyl)-1,1-dioxo-1λ6-thiane-4-carboxamide
N-methyl-N-[2-(4-methylphenoxy)ethyl]-3-[5-(5-methylthiophen-2-yl)-1,3,4-oxadiazol-2-yl]propanamide
1-{5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]-1'-yl}-2-(4-methyl-1,2,5-oxadiazol-3-yl)ethan-1-one
4-(2,4-dioxoimidazolidin-1-yl)-N-[2-oxo-2-(pyrrolidin-1-yl)ethyl]benzamide
5-(pyridin-4-yl)-N-[2-(pyridin-4-yl)ethyl]pyrazolo[1,5-a]pyrimidin-7-amine
({5-[(2E)-but-2-en-1-yl]-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)(methyl)[(7-methyl-1H-1,3-benzodiazol-2-yl)methyl]amine
dimethyl({1-[4-({4-[2-(methylsulfanyl)ethyl]piperazin-1-yl}methyl)phenyl]ethyl})amine
[(1-cyclopentylpiperidin-4-yl)methyl][(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl](oxolan-2-ylmethyl)amine
9-[(2-aminopyridin-3-yl)methyl]-2-(1-methylpyrrolidin-3-yl)-2,9-diazaspiro[5.5]undecan-3-one
N,N-dimethyl-5-({methyl[(1-phenyl-1H-pyrazol-4-yl)methyl]amino}methyl)pyridin-2-amine
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[3-(2-methyl-1H-imidazol-1-yl)propyl]benzamide
1-(5-phenyl-1,3,4-thiadiazol-2-yl)-N-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}piperidin-4-amine