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N-[2-(dimethylamino)ethyl]-N,1-dimethyl-6-propyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
2-[(2-chlorophenyl)methyl]-4-{4-[(3,5-dimethoxyphenyl)methyl]piperazin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
1-[3-(3-fluorophenyl)-1H-pyrazole-4-carbonyl]-4-(4-methyl-4H-1,2,4-triazol-3-yl)piperidine
3-(5-chloro-1-methyl-4-{[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]methyl}-1H-pyrazol-3-yl)-5-methyl-1,2-oxazole
methyl 3-{[2-(3,5-dimethyl-1H-pyrazol-1-yl)acetamido]methyl}-5-[3-(trifluoromethyl)benzamido]benzoate
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-2-oxoacetamide
N-(1-methyl-1H-pyrazol-5-yl)-2-(3-phenyl-1H-pyrazol-1-yl)acetamide
5-[(3aS,6aS)-octahydropyrrolo[3,4-b]pyrrol-5-ylmethyl]-2-(3-methylphenyl)pyrimidine
5-methyl-1-(4-methylphenyl)-4-{pyrazolo[1,5-a]pyridine-3-carbonyl}piperazin-2-one
5-[2-(ethylamino)ethyl]-1-[(3-methoxyphenyl)methyl]pyrrolidin-2-one
5-(3-cyclopropyl-1H-pyrazol-5-yl)-3-methyl-1H-1,2,4-triazole
4-{4H,5H,6H,7H-pyrazolo[1,5-a]pyridine-3-carbonyl}piperazine-2-carboxylic acid
2-{3-methyl-2-oxo-1-oxa-3,8-diazaspiro[4.6]undecan-8-yl}pyridine-3-carboxamide
N-[(3R,5S)-5-(ethylcarbamoyl)-1-(oxan-4-yl)pyrrolidin-3-yl]-2-(methylamino)pyrimidine-5-carboxamide
[(4-methyl-5,6,7,8-tetrahydroquinazolin-2-yl)methyl][1-(4-methylpiperazin-1-yl)propan-2-yl]amine
2-{4-[(4-cyclopropyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}-3,4-dihydroquinazolin-4-one
methyl 4-(5-{[(adamantan-1-ylmethyl)(2-hydroxyethyl)amino]methyl}-1,2,4-oxadiazol-3-yl)benzoate
4-(quinolin-2-ylmethyl)-1,4-oxazepan-5-one
2-{[4-(2-fluorophenyl)piperazin-1-yl]methyl}-N-(2-methylprop-2-en-1-yl)-1,3-oxazole-4-carboxamide
N-[3-(3-methoxyphenyl)phenyl]-1-[(methylcarbamoyl)methyl]piperidine-2-carboxamide
3-{4-[1-(3-fluoropropyl)-1,2,3,6-tetrahydropyridin-4-yl]-1H-pyrazol-1-yl}-3-methyl-1λ6-thiolane-1,1-dione
4-[2-(2-aminoethyl)phenyl]benzamide
methyl (2S,4S)-4-(4-ethyl-1,2,3-thiadiazole-5-amido)-1-methylpyrrolidine-2-carboxylate
N-[(3R,4R)-3-hydroxy-1-{[5-(2-methylpropyl)thiophen-2-yl]methyl}piperidin-4-yl]pyridine-4-carboxamide
1-[4-(2,3-dihydro-1H-isoindol-2-ylmethyl)-2-methoxyphenoxy]-3-(morpholin-4-yl)propan-2-ol
N-(1H-imidazol-2-ylmethyl)-N-[(3-methylthiophen-2-yl)methyl]cyclopropanamine
4-{2-propyl-3H-imidazo[4,5-b]pyridin-3-yl}-1-[4-(1H-pyrazol-1-yl)benzoyl]piperidine
1-[(2-ethylphenyl)methyl]-4-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidine
[2-({4-[(2E)-3-(furan-2-yl)-2-methylprop-2-en-1-yl]piperazin-1-yl}methyl)phenyl]methanol
N-[3-(2,3-dihydro-1H-isoindol-2-yl)propyl]-2-(1-ethylpiperidin-4-yl)acetamide
5-(4-{[4-(methoxymethyl)-1H-1,2,3-triazol-1-yl]methyl}piperidine-1-carbonyl)-1H-indole
5-methoxy-9-[4-(1H-pyrazol-1-yl)benzoyl]-1-oxa-9-azaspiro[5.5]undecane
2-(4-benzylmorpholin-2-yl)-N-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-ylmethyl}acetamide
4-chloro-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-N-(oxolan-2-ylmethyl)benzamide
2-(dimethylamino)-7-(ethanesulfonyl)-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
2-(4-methoxyphenoxymethyl)-N-[1-(trimethyl-1H-pyrazol-4-yl)ethyl]-1,3-oxazole-4-carboxamide
4-(1,3-benzothiazol-6-yl)-N-[2-(dimethylamino)ethyl]-1H-pyrrolo[2,3-b]pyridin-6-amine
N-(3,4-dimethoxyphenyl)-7-methyl-6-oxo-2,7-diazaspiro[4.5]decane-2-carboxamide
3-[1-(2-methyl-1,3-benzothiazol-6-yl)-1H-1,2,4-triazol-5-yl]-1λ6-thiane-1,1-dione
2-methyl-5-[3-(4-phenoxybenzoyl)piperidine-1-carbonyl]pyridine
[(3R,5S)-5-(morpholin-4-ylmethyl)-1-(pyridin-4-ylmethyl)piperidin-3-yl]methanol
2-(2,3-dimethylphenyl)-2-[methyl(pyrazin-2-ylmethyl)amino]acetic acid
4-(2,3-dimethylquinoxaline-6-carbonyl)-3-(3-fluorophenyl)piperazin-2-one
4-(1H-imidazol-1-ylmethyl)-1-(3-propyl-1H-pyrazole-5-carbonyl)piperidin-4-ol
(3S,4R)-1-[(1R,5S,6S)-3-azabicyclo[3.1.0]hexane-6-carbonyl]-4-(2H-1,3-benzodioxol-5-yl)pyrrolidine-3-carboxylic acid
({2,4-dimethyl-5-[(4-methylpiperazin-1-yl)methyl]phenyl}methyl)(methyl)(1,3-thiazol-2-ylmethyl)amine
N-methyl-5-({4-[1-(N-methylacetamido)ethyl]-1,2,3,6-tetrahydropyridin-1-yl}methyl)furan-2-carboxamide
1-(azocan-1-yl)-3-(5-{[(dicyclopropylmethyl)amino]methyl}-2-methoxyphenoxy)propan-2-ol
2-cycloheptyl-1-{4-[4-(2-hydroxypropan-2-yl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}ethan-1-one
(2R,3S,6R)-3-(2H-1,3-benzodioxol-5-yl)-5-(pyridin-2-yl)-1,5-diazatricyclo[5.2.2.02,6]undecane