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N-[1-(5-chloropyridin-2-yl)piperidin-4-yl]methanesulfonamide
(4aR,8aR)-2-cyclobutanecarbonyl-7-{[3-(difluoromethoxy)phenyl]methyl}-decahydro-2,7-naphthyridin-4a-ol
1-[3-(4-chlorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]-4,4,4-trifluorobutan-1-one
4-(furan-3-ylmethyl)-11-(4-methoxybenzoyl)-1,8-dioxa-4,11-diazaspiro[5.6]dodecane
N-[2-(adamantan-1-yl)-2-hydroxyethyl]-3-(pyridin-4-yl)propanamide
2-({2-[(3-methoxyphenyl)methyl]morpholin-4-yl}methyl)-4,5,6,7-tetrahydro-1,3-benzothiazole
4-[(5-{1-[(4-fluorophenyl)methyl]piperidin-3-yl}-4-methyl-4H-1,2,4-triazol-3-yl)methyl]morpholine
2-methyl-8-[2-(1H-1,2,4-triazol-1-yl)acetyl]-octahydro-1H-pyrazino[1,2-a]piperazin-1-one
N-benzyl-2-{4-[4-({[1-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}amino)piperidin-1-yl]phenyl}acetamide
4-(furan-3-ylmethyl)-9-methoxy-7-(2-methylphenyl)-2,3,4,5-tetrahydro-1,4-benzoxazepine
(4aS,7aR)-1-({4-[(dimethylamino)methyl]thiophen-2-yl}methyl)-4-(2-methylpropyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
(2S,4R)-1-[(3-chlorophenyl)methyl]-4-{[(2-hydroxyphenyl)methyl]amino}-N-(propan-2-yl)pyrrolidine-2-carboxamide
5-{[4-(1,3-benzothiazol-2-yl)-1,4-diazepan-1-yl]methyl}-N,N-dimethylpyridin-2-amine
3-{[3-(2-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-N-methyl-1,2,4-oxadiazole-5-carboxamide
5-methyl-3-phenyl-4-[3-(propan-2-yl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepine-7-carbonyl]-1,2-oxazole
N-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-5-methyl-6-(pyrrolidine-1-carbonyl)thieno[2,3-d]pyrimidin-4-amine
N-(2-hydroxyethyl)-4-methyl-N-{[4-(methylsulfanyl)phenyl]methyl}-2-(propan-2-yl)-1,3-thiazole-5-carboxamide
1-(4-amino-5-methylpyrimidin-2-yl)-4-[(4-fluorophenyl)methyl]-3-(propan-2-yl)-1,4-diazepan-5-one
N-[(1-ethyl-1H-imidazol-2-yl)methyl]-N,2,5-trimethylfuran-3-carboxamide
(2S,4R)-1-[(2-aminopyridin-3-yl)methyl]-4-cyclohexaneamido-N-ethylpyrrolidine-2-carboxamide
4-chloro-1-ethyl-N-(1,2-oxazol-3-ylmethyl)-1H-pyrazole-3-carboxamide
2-methoxy-5-[3-(1H-pyrazol-1-yl)phenyl]benzamide
8-(2H-1,3-benzodioxol-5-ylmethyl)-1-(3-methoxypropyl)-3-(pyridin-2-ylmethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-[2-(2,3-dihydro-1H-indol-1-yl)ethyl]-1-[2-(piperidin-2-yl)ethyl]-1H-1,2,3-triazole-4-carboxamide
N-(2-{[cyclohexyl(methyl)amino]methyl}phenyl)thiomorpholine-4-carboxamide
methyl 1-[(3S,5S)-5-(cycloheptylcarbamoyl)-1-[(6-methylpyridin-2-yl)methyl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
1,9-dimethyl-4-(quinoline-8-carbonyl)-1,4,9-triazaspiro[5.5]undecane
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl]({[3-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl})methylamine
1-[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]-N-[(3-methyl-1,2-oxazol-5-yl)methyl]piperidine-3-carboxamide
N-[4-(2-propyl-1H-imidazol-1-yl)phenyl]acetamide
9-methoxy-7-oxo-3-{[4-(pyrrolidin-1-yl)phenyl]methyl}-N-(1,3-thiazol-2-ylmethyl)-1H,2H,3H,4H,5H,7H-pyrido[1,2-d][1,4]diazepine-10-carboxamide
1-(cyclohexylmethyl)-N3-ethyl-N5-[1-(6-methoxynaphthalen-2-yl)ethyl]-4-oxo-1,4-dihydropyridine-3,5-dicarboxamide
methyl (2S,4S)-4-{3-[(4-fluorophenyl)formamido]propanamido}-1-methylpyrrolidine-2-carboxylate
5-[4-(1H-1,2,4-triazol-3-yl)benzoyl]-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridine-4-carboxylic acid
2-[4-(methoxymethyl)-5-methyl-1,2-oxazole-3-carbonyl]-7-(propan-2-yl)-2,7-diazaspiro[4.5]decan-6-one
3-[4-(1-benzothiophen-3-ylmethyl)piperazin-1-yl]-1,2-dihydropyrazin-2-one
3-methyl-N-{2-[2-(3-methylthiophen-2-yl)-1H-imidazol-1-yl]ethyl}pyridin-4-amine
N,5-dimethyl-N-[2-(1H-pyrazol-1-yl)ethyl]-1-benzofuran-2-carboxamide
1-[cyclopropyl(4-methylpyridin-2-yl)methyl]-3-(4-ethyl-1,3-dimethyl-1H-pyrazol-5-yl)urea
[4-(2-methoxy-5-methylphenyl)-4H-1,2,4-triazol-3-yl]methanamine
(2S,4S)-N-ethyl-4-[2-(1H-imidazol-1-yl)acetamido]-1-(thiophen-3-ylmethyl)pyrrolidine-2-carboxamide
N-[1-(cyclohex-1-en-1-yl)ethyl]-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
3-[2-(3,4-difluorophenyl)ethyl]-1-[(dimethyl-1,2-oxazol-4-yl)sulfonyl]piperidine
3-[5-(2H-1,3-benzodioxol-5-ylmethyl)-1,3,4-oxadiazol-2-yl]-N-(dicyclopropylmethyl)-N-methylpropanamide
5-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-N,N-dimethylpyridin-2-amine
1-(prop-2-en-1-yl)-4-[2-(pyridin-3-yl)-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]piperazine
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]but-3-enamide
1-ethyl-5-[2-(trifluoromethyl)phenyl]-1H,4H-pyrazolo[3,4-d]imidazole
2-methoxy-3-{[(1-methylpiperidin-4-yl)amino]methyl}-6-[2-(pyridin-2-yl)ethyl]-5H,6H,7H-pyrrolo[3,4-b]pyridin-5-one
N-[(3S,4R)-4-(4-methoxyphenyl)-1-(3-methylthiophene-2-carbonyl)pyrrolidin-3-yl]acetamide