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2-(1,1-dioxo-1λ6-thiolan-3-yl)-N-methyl-N-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}acetamide
2-{1-butyl-5-[2-(methylamino)pyridin-4-yl]-1H-1,2,4-triazol-3-yl}acetamide
4-({3-[4-(trifluoromethyl)benzoyl]piperidin-1-yl}methyl)-1H-pyrazole-3-carboxylic acid
N-cyclopentyl-5-methoxy-N-[(5-methylthiophen-2-yl)methyl]-4-oxo-1,4-dihydropyridine-2-carboxamide
3-[2-({4-[3-(propan-2-yl)-1H-pyrazol-5-yl]piperidin-1-yl}methyl)-1H-pyrrol-1-yl]pyridine
3-(azepane-1-carbonyl)-N-[(3,4-difluorophenyl)methyl]-1-ethyl-4,5,6,7-tetrahydro-1H-indazol-5-amine
N-(diphenylmethyl)-3-{2-[(4-methoxyphenyl)methyl]-5-oxopyrrolidin-2-yl}propanamide
ethyl 2-[(2-{methyl[1-(4-methyl-1,3-thiazol-2-yl)ethyl]carbamoyl}phenyl)amino]acetate
1-[(4,5-dimethylfuran-2-yl)methyl]-8-(quinolin-6-yl)-1,8-diazaspiro[4.5]decane
4-[1-(2-methyl-6-propylpyrimidin-4-yl)piperidin-4-yl]thiomorpholine
8-[(3aS,6aS)-1-methyl-octahydropyrrolo[3,4-b]pyrrole-5-carbonyl]-2,3,4,9-tetrahydro-1H-carbazole
1-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}-3-(1H-1,2,4-triazol-1-yl)propan-1-one
1-{[1-(3-methoxyphenyl)-1H-pyrazol-4-yl]methyl}-5-{2-[(pyridin-2-ylmethyl)amino]ethyl}pyrrolidin-2-one
2-(3-fluorophenyl)-N-[2-(furan-2-yl)ethyl]-1,3-benzoxazole-5-carboxamide
3-[2-(dimethylamino)ethyl]-8-[(1-methyl-1H-pyrazol-4-yl)methyl]-1-(3-methylbutyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
1-[2-(4-methoxyphenyl)ethyl]-3-(2-methylpropyl)-8-[1-(methylsulfanyl)propan-2-yl]-1,3,8-triazaspiro[4.5]decane-2,4-dione
2-amino-7-[2-(3-methoxyphenoxy)acetyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
3-{5-[1-(4-chlorophenyl)cyclobutyl]-1,3,4-oxadiazol-2-yl}-N-[(5-methylthiophen-2-yl)methyl]propanamide
8-{[(2-fluorophenyl)methyl]carbamoyl}-2-methyl-2,8-diazaspiro[4.5]decane-3-carboxylic acid
N-[4-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]azocane-1-carboxamide
N-[(2,2-dimethyl-1-phenylcyclopropyl)methyl]-1-(propan-2-yl)-1H-pyrazole-4-carboxamide
5,6-dimethyl-N4-{1-[5-(propan-2-yl)-1,3,4-oxadiazol-2-yl]ethyl}pyrimidine-2,4-diamine
1-(6-ethoxy-4-methylquinazolin-2-yl)-N-[2-(2-methyl-1H-imidazol-1-yl)ethyl]pyrrolidine-2-carboxamide
N-{2-[(4-methyl-1,2,5-oxadiazol-3-yl)oxy]ethyl}-2-oxo-1-phenylpyrrolidine-3-carboxamide
[(5-cyclopentylthiophen-2-yl)methyl][2-methoxy-1-(pyridin-2-yl)ethyl]methylamine
5-fluoro-1-methyl-2-[3-(2-methylpiperidin-1-yl)azetidine-1-carbonyl]-1H-indole
4-{4-[2-(3-chlorophenoxy)acetyl]-2-oxopiperazin-1-yl}benzonitrile
3-(7-methyl-1H-indol-3-yl)-5-(morpholine-4-sulfonyl)benzoic acid
4-[(2-methylprop-2-en-1-yl)oxy]-N-[3-(propan-2-yloxy)propyl]benzamide
(3aS,6aS)-2-(cyclopropylmethyl)-1-oxo-5-[3-(1H-pyrrol-1-yl)propyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
({4-[2-(dimethylamino)ethoxy]phenyl}methyl)(methyl)(1,3-thiazol-2-ylmethyl)amine
1-{3-[(4-ethoxypiperidin-1-yl)methyl]-6-methylquinolin-2-yl}piperidin-3-ol
3-(3-hydroxybutyl)-6,8-dimethyl-3,4-dihydroquinazolin-4-one
[(1-ethyl-1H-imidazol-2-yl)methyl]({1-[(2-methylphenyl)methyl]piperidin-4-yl}methyl)(pyridin-3-ylmethyl)amine
1-[(3S,4R)-3-benzyl-4-hydroxy-4-methylpiperidin-1-yl]-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
1-[(3R,4R)-4-hydroxy-3-methyl-4-(oxan-4-yl)piperidin-1-yl]-3-(5-methyl-1H-1,2,4-triazol-3-yl)propan-1-one
2-(4-{2-[2-(3-chlorophenyl)-1H-imidazol-1-yl]ethyl}-1,3-thiazol-2-yl)pyrimidine
4-(2-methylpiperidin-1-yl)-3-(2-{[1,2,4]triazolo[1,5-a]pyrimidin-6-yl}acetamido)benzamide
3-cyclohexyl-N-[(3-methyl-5,6,7,8-tetrahydro-2,7-naphthyridin-4-yl)methyl]-1H-pyrazole-4-carboxamide
N-[(2R,3R)-2-hydroxy-2,3-dihydrospiro[indene-1,4'-piperidine]-3-yl]-4-methoxy-3,5-dimethylbenzamide
methyl 5-[(butan-2-yl)amino]-3-(oxolane-2-amido)-1-(2-phenylethyl)-1H-pyrrolo[2,3-b]pyridine-2-carboxylate
1'-(2-{imidazo[1,2-a]pyridin-3-yl}acetyl)-1,2-dihydrospiro[indole-3,3'-piperidine]-2-one
3-({5-[4-(2-phenylethyl)piperidine-1-carbonyl]pyridin-2-yl}amino)propane-1,2-diol
2-[1-(2-phenylethyl)-5-{[1,2,3,4]tetrazolo[1,5-a]pyridin-7-yl}-1H-1,2,4-triazol-3-yl]acetamide
(1s,4s)-4-hydroxy-N-{2-[3-(propan-2-yloxy)phenyl]ethyl}cyclohexane-1-carboxamide
N-[(4-cyclohexyl-4H-1,2,4-triazol-3-yl)methyl]-3-(4-methyl-1,3-thiazol-5-yl)propanamide
2-methyl-N4-{3-[(pyridin-3-yl)amino]propyl}pyrimidine-4,6-diamine
1-ethyl-4-{4-[2-(2-methyl-1H-imidazol-1-yl)ethyl]piperidine-1-carbonyl}pyrrolidin-2-one
2-methyl-5-(4-{2-oxo-1-oxaspiro[4.4]nonane-4-carbonyl}piperazin-1-yl)-2,3-dihydropyridazin-3-one
1-[(2-fluoro-4,5-dimethoxyphenyl)methyl]azepan-2-one