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N-methyl-N-[(2-phenyl-1,3-thiazol-4-yl)methyl]imidazo[1,2-b]pyridazine-3-carboxamide
3-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]-5-propyl-1,2-oxazole
N-[(3S,4R)-1-{1H,4H,5H,6H-cyclopenta[c]pyrazole-3-carbonyl}-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
2-cyclopropyl-8-[2-methyl-6-(1H-pyrazol-1-yl)pyrimidin-4-yl]-2,8-diazaspiro[5.5]undecan-3-one
2-(5-acetylthiophen-3-yl)-N-{[4-(hydroxymethyl)oxan-4-yl]methyl}-N-methylacetamide
1-({1-[3-(5-methyl-1H-1,2,3,4-tetrazol-1-yl)propanoyl]piperidin-4-yl}methyl)pyrrolidin-2-one
N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1-propylpiperidin-4-amine
1-(4-cyclopentyl-1,4-diazepan-1-yl)-2-(2-fluorophenyl)-2-hydroxyethan-1-one
3-(2-amino-1,3-thiazol-4-yl)-N-[(2-phenyl-1,3-thiazol-5-yl)methyl]propanamide
3-(5-{[(furan-2-ylmethyl)(thiophen-3-ylmethyl)amino]methyl}thiophen-3-yl)prop-2-yn-1-ol
7-(2-hydroxyethyl)-2-[(6-methoxy-2,3-dihydro-1H-inden-5-yl)methyl]-2,7-diazaspiro[4.5]decan-6-one
14-[4-(pyridin-2-ylmethoxy)phenyl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
2-[5-({3-oxo-2,8-diazaspiro[4.5]decan-8-yl}methyl)furan-2-yl]benzonitrile
2-[(1S,2S,4S)-bicyclo[2.2.1]hept-5-en-2-yl]-N-(1-methylpiperidin-4-yl)-N-(pyridin-4-ylmethyl)acetamide
4-(1-butyl-1H-imidazol-2-yl)-1-(3-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperidine
N-[4-(3-fluorophenyl)phenyl]-1-[(1-methyl-1H-imidazol-2-yl)methyl]pyrrolidine-2-carboxamide
N-cyclopentyl-N-({3-[(4-fluorophenyl)methoxy]phenyl}methyl)pyrazolo[1,5-a]pyrimidine-3-carboxamide
2-[2-({cyclopentyl[(3-methylthiophen-2-yl)methyl]amino}methyl)phenoxy]acetamide
8-chloro-2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]quinoline
8-(1-ethyl-1H-pyrazole-4-carbonyl)-2-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecan-3-one
5-(2,5-dimethylphenoxymethyl)-N-methyl-N-[1-(1,3-thiazol-2-yl)ethyl]-1,2-oxazole-3-carboxamide
1'-(3-chlorobenzoyl)-5-cyclopropanecarbonyl-1,5,6,7-tetrahydrospiro[imidazo[4,5-c]pyridine-4,4'-piperidine]
N-[2-(dimethylamino)-2-(3-methylphenyl)ethyl]-3-(2-oxopiperidin-1-yl)propanamide
5-methyl-3-{[3-(pyridin-3-yl)-1,2-oxazol-5-yl]methyl}-3H,4H-thieno[2,3-d]pyrimidin-4-one
(3S,4S)-4-(2H-1,3-benzodioxol-5-yl)-3-hydroxy-N,N-dimethylpiperidine-1-sulfonamide
N-[(4-ethoxyphenyl)methyl]-N-(2-methoxyethyl)-1H-1,3-benzodiazole-2-carboxamide
6-[1-ethyl-3-(oxolan-3-yl)-1H-1,2,4-triazol-5-yl]-4-methyl-3,4-dihydro-2H-1,4-benzoxazin-3-one
1-[2-(dimethylamino)ethyl]-4-[3-(2,6-dimethylphenoxy)azetidine-1-carbonyl]pyrrolidin-2-one
6-(benzyloxy)-1-(oxan-4-ylmethyl)-4-(quinolin-4-ylmethyl)-1,4-diazepan-2-one
3-(2-aminoethyl)-4-(4-tert-butylphenyl)-4,5-dihydro-1H-1,2,4-triazol-5-one
1-(cyclohex-3-en-1-ylmethyl)-3-[4-(3-fluorophenyl)-1H-pyrazol-5-yl]piperidine
1-(4-{[(3-hydroxypropyl)amino]methyl}-2-methoxyphenoxy)-3-(thiomorpholin-4-yl)propan-2-ol
N-{1-[(2-fluorophenyl)methyl]piperidin-3-yl}-6-methoxy-N,1-dimethyl-1H-indole-2-carboxamide
1-[4-(2-methanesulfonylethyl)piperazin-1-yl]-3-(4-methyl-1,3-thiazol-5-yl)propan-1-one
1-{3-oxo-3-[3-(pyridin-2-ylmethoxy)piperidin-1-yl]propyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{benzyl[(4-chloro-1-methyl-1H-indazol-3-yl)methyl]amino}-2-methylpropan-1-ol
N-[3-(3-chlorophenyl)phenyl]-1-(2-hydroxyacetyl)piperidine-4-carboxamide
4-ethyl-1-[2-(phenylsulfanyl)ethyl]-3-(piperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-[(7-methoxy-3,4-dihydro-2H-1-benzopyran-3-yl)methyl]-4-(1H-pyrazol-1-yl)butanamide
5-({[(1-hydroxycyclohexyl)methyl]carbamoyl}amino)-N,N-dimethyl-1-benzothiophene-2-carboxamide
{1-[(5-ethylthiophen-2-yl)sulfonyl]-4-[(4-methoxyphenyl)methyl]piperidin-4-yl}methanol
1-(4-fluorophenyl)-4-(1H-pyrrole-2-carbonyl)-1,4-diazepane
1-(5-methyl-1,2-oxazole-3-carbonyl)-N-[2-(pyridin-3-yloxy)phenyl]piperidine-3-carboxamide
2-[(5-methylpyrazin-2-yl)methyl]-8-[2-(propylsulfanyl)acetyl]-2,8-diazaspiro[5.5]undecan-3-one
1-{4-hydroxy-4-[3-(trifluoromethyl)phenyl]piperidin-1-yl}-2-(4-methyl-1H-pyrazol-1-yl)ethan-1-one
4-{3-[methyl({2-[4-(thiomorpholine-4-carbonyl)-1H-1,2,3-triazol-1-yl]ethyl})amino]butyl}phenol
1-ethyl-4-{[methyl({trimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-yl})amino]methyl}pyrrolidin-2-one
N-{[1-(2,3-dihydro-1H-inden-2-yl)piperidin-4-yl]methyl}-N-[3-(dimethylamino)propyl]cyclopropanecarboxamide
(4aS,7aR)-1-(2-methoxypyrimidine-5-carbonyl)-4-(3-methylbut-2-en-1-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-{3-[(3R,4R)-3-hydroxy-3,4-dimethylpyrrolidin-1-yl]-3-oxopropyl}-1,2,3,4-tetrahydropyrimidine-2,4-dione