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4-(4-methyl-1H-pyrazol-3-yl)-N-[2-methyl-5-(2-oxopyrrolidin-1-yl)phenyl]piperidine-1-carboxamide
5-chloro-2-[4-(pyrrolidin-1-ylmethyl)piperidine-1-carbonyl]phenol
3-[4-(dimethylamino)-2-(pyridin-3-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidine-7-carbonyl]-2-methylphenol
3-(4-ethyl-1H-pyrazol-5-yl)-1-(2-propyl-1,3-thiazole-4-carbonyl)piperidine
N-{[3-(cyclopentyloxy)phenyl]methyl}-1-(pyrimidin-2-yl)piperidin-3-amine
(2S,4S)-1-[(2-chlorophenyl)methyl]-N-(2-methoxyethyl)-4-{[(3-phenoxyphenyl)methyl]amino}pyrrolidine-2-carboxamide
3-{1-[4-(aminomethyl)benzoyl]piperidin-3-yl}-1-[2-(dimethylamino)ethyl]-4-ethyl-4,5-dihydro-1H-1,2,4-triazol-5-one
3-butyl-1-methyl-4-(5-methyl-1-propyl-1H-pyrazole-4-carbonyl)piperazin-2-one
2-(3-fluorophenyl)-N-[1-(5-methyl-1H-1,2,4-triazol-3-yl)ethyl]acetamide
8-(1,3-benzothiazol-2-ylmethyl)-1-(2-methoxyethyl)-3-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
N-{[5-(thiophen-2-ylmethyl)-1,2,4-oxadiazol-3-yl]methyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
3-(1,3-dimethyl-1H-pyrazol-4-yl)-1-[2-(2-fluorophenoxy)ethyl]-1-(2-methoxyethyl)urea
2-methyl-1-(4-{[(3-methylphenyl)(thiophen-2-yl)methyl]amino}piperidin-1-yl)propan-1-one
3-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-1-{4-[(5-methyl-4H-1,2,4-triazol-3-yl)methyl]phenyl}urea
1-cyclopentyl-3-(3-phenylpiperidine-1-carbonyl)-5-(piperidine-1-carbonyl)-1,4-dihydropyridin-4-one
(3S,4R)-1-{2-[(dimethylcarbamoyl)amino]acetyl}-4-(3-methoxyphenyl)pyrrolidine-3-carboxylic acid
7-(1-benzothiophen-3-yl)-4-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
N-methyl-2-[3-oxo-2-(pyridin-3-ylmethyl)-2,9-diazaspiro[5.5]undecan-9-yl]propanamide
{1-[(1-ethyl-1H-1,2,4-triazol-5-yl)methyl]pyrrolidin-3-yl}methanamine
4-(3-ethyl-1H-pyrazole-4-carbonyl)-1-(4-methoxyphenyl)-2,2-dimethylpiperazine
6-[3-(3-methoxyphenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-5-carbonyl]-1,2-dihydropyridin-2-one
[9-(oxan-4-yl)-3-(1H-pyrrole-3-carbonyl)-3,9-diazaspiro[5.5]undecan-1-yl]methanol
2-{4-[4-(3-methoxypiperidine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-1,3-benzoxazole
1-[2-(3-fluorophenyl)ethyl]-2-(6-methoxy-2H-1,3-benzodioxol-5-yl)-1H-imidazole
5-(oxolan-2-yl)-N-[1-(pyrrolidine-1-carbonyl)piperidin-4-yl]thiophene-2-carboxamide
N-(4-chloro-2-methylphenyl)-3-oxo-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecane-9-carboxamide
N-(2,3-dihydro-1H-inden-2-yl)-5-(oxolan-2-yl)thiophene-2-carboxamide
2-[(1R,5R)-6-(cyclobutylmethyl)-3,6-diazabicyclo[3.2.2]nonan-3-yl]-8-methoxy-4-methylquinoline
3-[(2,1,3-benzoxadiazol-4-ylmethyl)(ethyl)amino]-1λ6-thiolane-1,1-dione
N-[2-(1H-indol-1-yl)ethyl]-N-methyl-1H-imidazole-2-carboxamide
1-[(4aR,8aR)-7-(2-amino-5-butyl-6-methylpyrimidin-4-yl)-4a-hydroxy-decahydro-2,7-naphthyridin-2-yl]ethan-1-one
14-(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
3-[3-(4-ethylpiperazin-1-yl)propyl]-8-(2-hydroxyacetyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
5-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-1-[2-(1H-imidazol-5-yl)ethyl]-3-(2-methoxyethyl)-1H-1,2,4-triazole
2-[1-(4-chloro-2-methoxybenzoyl)-1,4-diazepan-6-yl]acetic acid
3-{[3-(4-chlorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]methyl}-5-(oxolan-2-yl)-1,2,4-oxadiazole
N-[2-(dimethylamino)ethyl]-3-(5-methyl-1H-pyrazol-1-yl)-N-[(5-methylthiophen-2-yl)methyl]propanamide
N-(4,5,6,7-tetrahydro-1-benzothiophen-3-ylmethyl)-6-(4H-1,2,4-triazol-4-yl)pyridine-2-carboxamide
3-(2-fluorophenyl)-N-[(3S,4S)-4-methoxy-1-(propan-2-yl)pyrrolidin-3-yl]-1H-pyrazole-5-carboxamide
3-[(1-ethyl-1H-imidazol-2-yl)methyl]-3-methyl-1-[3-(3-methyl-2,5-dioxoimidazolidin-1-yl)phenyl]urea
N,2,4-trimethyl-N-{[3-(pyridin-4-yl)-1,2-oxazol-5-yl]methyl}-1,3-thiazole-5-carboxamide
(4aS,8aR)-6-[2-(morpholin-4-yl)-2-oxoethyl]-1-[2-(pyridin-2-yl)ethyl]-decahydro-1,6-naphthyridin-2-one
5-(1-cyclopentyl-4-hydroxypiperidin-4-yl)-N-methyl-N-(quinolin-8-ylmethyl)-1-benzofuran-2-carboxamide
2-{4-[(4-ethyl-1-methyl-5-oxo-4,5-dihydro-1H-1,2,4-triazol-3-yl)methyl]piperidine-1-carbonyl}pyrrolidine-1-carboxamide
(3R)-3,4,4-trimethyl-1-[2-methyl-2-(piperidin-1-yl)propyl]pyrrolidin-3-ol
2-{[1-(dimethyl-1,3-thiazol-4-yl)ethyl](methyl)amino}-N,N-dimethylacetamide
3-hydroxy-3-{[methyl(propan-2-yl)amino]methyl}-1-(2-phenylethyl)piperidin-2-one
3-[(2E)-3-(2-methoxyphenyl)prop-2-en-1-yl]-7-methyl-3,7,11-triazaspiro[5.6]dodecan-12-one
2-(2-methoxyethyl)-9-(3-methylbenzoyl)-2,9-diazaspiro[5.5]undecan-3-one
N-({4-[(dimethylamino)methyl]phenyl}methyl)-N-methyl-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine