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N-butyl-N,1-dimethyl-3-(thiomorpholine-4-carbonyl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
4-(3-cyano-4,6-dimethylpyridin-2-yl)-N,N-dimethylbenzamide
{9-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-3,9-diazaspiro[5.5]undecan-1-yl}methanol
N-[(3S,4R)-1-(2-methoxypyridine-4-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
5-[(isoquinolin-5-yloxy)methyl]-N-(3-phenylpropyl)-1,2-oxazole-3-carboxamide
6-(4-{[4-(pyridin-3-yl)-1H-1,2,3-triazol-1-yl]methyl}piperidin-1-yl)-9H-purine
N-[3-(dimethyl-1,3-thiazol-2-yl)propyl]-3-(1-methylpiperidin-3-yl)propanamide
2-{9-[(2S)-2-hydroxy-2-phenylacetyl]-3-oxo-2,9-diazaspiro[5.5]undecan-2-yl}acetic acid
1-(2-oxo-1,2-dihydroquinoline-4-carbonyl)azetidine-2-carboxylic acid
3-[(3-{2-ethyl-3-oxo-2,8-diazaspiro[4.5]decan-8-yl}-3-oxopropyl)(methyl)amino]-1λ6-thiolane-1,1-dione
(1S,6R)-3-methyl-9-[6-(morpholin-4-yl)pyrimidin-4-yl]-3,9-diazabicyclo[4.2.1]nonan-4-one
2-(2-fluoro-6-methoxyphenyl)-1,3-benzothiazole
2-(4-fluorophenyl)-1-[3-(4-methoxyphenyl)-1H-pyrazole-5-carbonyl]piperidine
2-(2-{methyl[(4-methylphenyl)methyl]amino}pyrimidin-4-yl)pyridine-4-carboxylic acid
4-[(3R,4R)-4-hydroxy-4-(2-methoxyethyl)-3-methylpiperidine-1-carbonyl]benzene-1-sulfonamide
5-methoxy-2-{[3-(3-methoxyphenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}pyridin-4-ol
N-[2-(morpholin-4-yl)butyl]-5-propyl-1,2-oxazole-3-carboxamide
N-[(1r,4r)-4-(4H-1,2,4-triazol-4-yl)cyclohexyl]spiro[2.4]heptane-1-carboxamide
1-{3-[(3,4-dimethylphenyl)amino]piperidin-1-yl}-4-methylpentane-1,2-dione
9-[(3-fluoro-4-methylphenyl)methyl]-2-(3-hydroxypropyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 6-methyl-2-{[1-(3-phenylpropyl)piperidin-3-yl]amino}pyrimidine-4-carboxylate
(3aR,6aS)-2-[(2-chloro-5-fluorophenyl)methyl]-5-methyl-octahydropyrrolo[3,4-c]pyrrole
N-[2-(4-chlorophenyl)propyl]-5-(methoxymethyl)furan-2-carboxamide
2-(4-acetylphenoxy)-1-(10-methoxy-3,4,5,6-tetrahydro-2H-1,5-benzoxazocin-5-yl)ethan-1-one
4-[4-(2-chlorophenyl)-1H-1,2,3-triazol-1-yl]-1-(1,3-thiazol-2-ylmethyl)piperidine
1-[({[7-chloro-2-(thiophen-3-yl)quinolin-3-yl]methyl}amino)methyl]cyclohexan-1-ol
2-[3-(2-hydroxy-4,6-dimethylpyrimidin-5-yl)propanoyl]-7-methyl-2,7-diazaspiro[4.5]decan-6-one
3-{[methyl({[2-(pyrrolidin-1-ylmethyl)phenyl]methyl})amino]methyl}piperidin-3-ol
5-{1-ethyl-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazine-2-carbonyl}-2,4-dimethyl-1,3-thiazole
1-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-3-[2-(3-methoxyphenyl)ethyl]piperidine
3-{3-[(3,4-dimethoxyphenyl)amino]piperidine-1-carbonyl}-N-methylpyridin-2-amine
1-[2-(dimethylamino)ethyl]-5-oxo-N-{[2-(1H-pyrazol-1-ylmethyl)phenyl]methyl}pyrrolidine-3-carboxamide
(3S,4R)-4-(3-fluorophenyl)-1-[3-(4-hydroxyphenyl)propanoyl]pyrrolidine-3-carboxylic acid
2-[3-tert-butyl-5-(2-hydroxy-3-methylphenyl)-1H-1,2,4-triazol-1-yl]acetic acid
5-[5-methyl-2-(4H-1,2,4-triazol-4-yl)pyridin-3-yl]pyridin-3-amine
2-cyclobutyl-5-fluoro-1-{1-[5-(4-methoxyphenyl)furan-2-carbonyl]piperidin-4-yl}-1H-1,3-benzodiazole
[1-(4-methanesulfonylbenzenesulfonyl)-4-(3-phenylpropyl)piperidin-4-yl]methanol
5-cyclopropyl-1-[4-(3-fluoro-4-methoxyphenyl)pyrimidin-2-yl]-N-methyl-N-(2-methylpropyl)-1H-pyrazole-4-carboxamide
2-(5-phenyl-1,2,4-oxadiazol-3-yl)-1H,4H,5H,6H,7H,8H-imidazo[4,5-c]azepin-4-one
N-[2-(dimethylamino)-2-(2-methylphenyl)ethyl]-1-methyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-({[7-chloro-2-(2-phenylethoxy)quinolin-3-yl]methyl}amino)propan-1-ol
3-[(3R,4R)-3-(hydroxymethyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidine-1-carbonyl]-4-methylbenzene-1-sulfonamide
N-[(3S,4R)-4-(4-methoxyphenyl)-1-[2-(piperidin-1-yl)acetyl]pyrrolidin-3-yl]acetamide
(3aR,6aS)-2-ethyl-5-{[(4-fluorophenyl)methyl]carbamoyl}-1-oxo-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
N-cyclohexyl-2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]acetamide
6-methyl-5-{5-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
4-(1-tert-butyl-1H-pyrazol-4-yl)-1-[(4-methanesulfonylphenyl)methyl]-1,2,3,6-tetrahydropyridine
3-[(3S,7S,8aS)-3-[(1R)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-[2-(trifluoromethyl)phenyl]urea
4-{2-[3-(4-fluorophenyl)pyrrolidin-1-yl]pyridine-4-carbonyl}morpholine
1-methyl-9-(prop-2-en-1-yl)-4-[3-(1H-pyrazol-4-yl)propanoyl]-1,4,9-triazaspiro[5.6]dodecan-10-one