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9-[2-(3-fluoro-4-hydroxyphenyl)acetyl]-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
methyl 1-oxo-2-(1,3-thiazol-5-ylmethyl)-1,2-dihydroisoquinoline-7-carboxylate
1-[(3-fluorophenyl)methyl]-N-[(1-methyl-1,2,3,4-tetrahydroquinolin-6-yl)methyl]-6-oxopiperidine-3-carboxamide
N-[1-(4-cyclopentyl-4H-1,2,4-triazol-3-yl)ethyl]-2-(1-ethylpiperidin-4-yl)acetamide
1-{2-[(2R,3S,6R)-3-(3-methoxyphenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]-2-oxoethyl}pyrrolidin-2-one
1-[2-(1H-imidazol-2-yl)benzoyl]-2-methyl-4-(2-methylphenyl)piperazine
N-{1-[4-(2-methoxyethyl)-4H-1,2,4-triazol-3-yl]ethyl}thian-4-amine
1-[3-({dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-yl}amino)propyl]pyrrolidin-2-one
N-[3-(dimethyl-1H-1,2,4-triazol-1-yl)propyl]-2-methylthieno[3,2-d]pyrimidin-4-amine
6-ethyl-N-[(2-fluorophenyl)methyl]-N-(2-methoxyethyl)-1,5-dimethyl-2-oxo-1,2-dihydropyridine-3-carboxamide
4-chloro-1-{2-[3-(3,4-difluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]ethyl}-1H-pyrazole
2-[1-(1-cyclopropanecarbonylpiperidin-4-yl)-1H-1,2,3-triazol-4-yl]pyridine
(3S,7S,8aS)-3-benzyl-7-{[(3-methoxyphenyl)methyl]amino}-octahydropyrrolo[1,2-a]piperazine-1,4-dione
({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(2-methoxyethyl)[(2-methyl-1H-imidazol-4-yl)methyl]amine
1-{[2-(4-methoxynaphthalen-1-yl)-5-methyl-1,3-oxazol-4-yl]methyl}-N-methylpyrrolidine-3-carboxamide
N-{[4-(prop-2-en-1-yl)-5-{[2-(pyrrolidin-1-yl)ethyl]sulfanyl}-4H-1,2,4-triazol-3-yl]methyl}propanamide
2,4-difluoro-N-{[(3S,4S)-3-hydroxy-1-[(1-methyl-1H-pyrazol-4-yl)methyl]piperidin-4-yl]methyl}benzamide
N-{1-[(4-fluorophenyl)methyl]-5-oxopyrrolidin-3-yl}-3-(thiophen-3-yl)propanamide
2-[methyl(pyridin-4-ylmethyl)amino]-N-[1-(2-methyl-1,3-thiazol-4-yl)ethyl]acetamide
[3-(1H-imidazol-1-yl)propyl][(3-methyl-1,2-oxazol-5-yl)methyl](pyridin-4-ylmethyl)amine
(1S,5R)-6-cyclopropanecarbonyl-3-[(dimethyl-1,2-oxazol-4-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
2-(dimethyl-1,2-oxazol-4-yl)-N-{[2-(dimethylamino)-7-methylquinolin-3-yl]methyl}-N-[2-(4-fluorophenyl)ethyl]acetamide
N4-(3,4-dihydro-1H-2-benzopyran-1-ylmethyl)-6-(morpholin-4-yl)pyrimidine-2,4-diamine
1-[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]-3-[1-(1,3-thiazol-4-ylmethyl)-1H-imidazol-2-yl]piperidine
1-(5-cyclobutyl-1,3,4-oxadiazol-2-yl)-4-(5-methylpyridin-2-yl)piperidin-4-ol
(2S,4R)-4-amino-N-ethyl-1-[1-(methoxymethyl)cyclobutanecarbonyl]pyrrolidine-2-carboxamide
N-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-(propan-2-yl)quinoxaline-5-carboxamide
N-cyclopropyl-8-methyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
(2S,4S)-4-amino-1-[2-(3,5-dimethoxyphenyl)acetyl]-N,N-diethylpyrrolidine-2-carboxamide
3-ethyl-8-(2-methylpropyl)-1-(2-phenylethyl)-1,3,8-triazaspiro[4.5]decane-2,4-dione
butyl 2-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]pyrrolidine-1-carboxylate
14-[2-(3-methylphenyl)pyrimidin-5-yl]-2,8,11-triazatricyclo[7.5.0.02,7]tetradeca-1(9),3,5,7-tetraen-12-one
3-(3-hydroxy-3-methylbutyl)-N-[2-(oxan-3-yl)ethyl]benzamide
methyl 1-ethoxy-2-oxo-8-[2-(2-oxo-4-phenylpyrrolidin-1-yl)acetyl]-1,8-diazaspiro[4.5]decane-4-carboxylate
2-[3-({[(1R,2S)-2-hydroxycyclohexyl](methyl)amino}methyl)phenoxy]acetamide
N-({1-[2-(4-chlorophenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-2-(propan-2-yl)-1,3-thiazole-4-carboxamide
3-(1-methyl-1H-imidazol-2-yl)-7-thia-2,4,5-triazatricyclo[6.4.0.02,6]dodeca-1(12),3,5,8,10-pentaene
N,N-dimethyl-3-{3-[(methylsulfanyl)methyl]-1,2,4-oxadiazol-5-yl}piperidine-1-carboxamide
2-[2-(1H-imidazol-4-yl)ethyl]-9-(oxane-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
N-[2-(azepan-1-yl)-2-phenylethyl]-1-methyl-3-propyl-1H-pyrazole-5-carboxamide
methyl 6-{[4-(diethylamino)phenyl]methyl}-2-(diethylsulfamoyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
3-(2-methoxyethyl)-1-[(2E)-2-methylbut-2-en-1-yl]piperidine-3-carboxylic acid
1-[2-(benzyloxy)phenyl]-3-[(1R,2S)-2-hydroxycyclohexyl]-3-methylurea
ethyl 5-[(2E)-3-(furan-2-yl)prop-2-en-1-yl]-1-(2-hydroxyethyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine-3-carboxylate
1-(3-phenylbutyl)-4-[2-(piperidine-1-carbonyl)-1-benzofuran-5-yl]piperidin-4-ol
1-(3-cyano-4-ethoxyphenyl)-3-(2-methoxyethyl)-3-propylurea
1-[4-hydroxy-3,3-dimethyl-4-(morpholin-4-ylmethyl)piperidin-1-yl]-2-(trimethyl-1H-pyrazol-1-yl)ethan-1-one
methyl N-{2-[4-(4-methoxyphenyl)-2-methyl-5-oxopiperazin-1-yl]-2-oxoethyl}carbamate
2-benzyl-8-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-2,8-diazaspiro[5.5]undecane
3-[(3R,4S)-4-(4-methylpiperazin-1-yl)-1-(1,3-thiazol-2-yl)piperidin-3-yl]propan-1-ol