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4-[(3,5-difluorophenyl)methyl]-1-methyl-9-(prop-2-en-1-yl)-1,4,9-triazaspiro[5.6]dodecan-10-one
2-(1-ethylpiperidin-4-yl)-1-(4-methoxy-4-phenylpiperidin-1-yl)ethan-1-one
methyl 2-[8-(furan-3-ylmethyl)-1-(2-methoxyethyl)-2,4-dioxo-1,3,8-triazaspiro[4.5]decan-3-yl]acetate
(4S)-3,3,4-trimethyl-1-[2-(pyridin-2-yl)pyrimidine-5-carbonyl]piperidin-4-ol
5-[2-(3-methoxypropyl)piperidine-1-carbonyl]-2,1,3-benzoxadiazole
1-[(3R,4R)-3-(hydroxymethyl)-4-(piperidin-1-ylmethyl)pyrrolidin-1-yl]-2-(naphthalen-2-yloxy)ethan-1-one
(4-{[methyl({6-methyl-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3,5,7,12,14-hexaen-4-yl})amino]methyl}oxan-4-yl)methanol
1-{[3-(4-methoxyphenyl)-1,2,4-oxadiazol-5-yl]methyl}-4-(pyrimidin-2-yl)-1,4-diazepane
(1R,5R)-3-methanesulfonyl-6-[3-(1-methyl-1H-pyrrol-2-yl)-1H-pyrazole-5-carbonyl]-3,6-diazabicyclo[3.2.2]nonane
2-[4-chloro-2-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]pyrazine
N-[2-(dimethylamino)ethyl]-N-methyl-1-[1-(pyridin-4-ylmethyl)piperidin-4-yl]piperidine-3-carboxamide
4-{4-[(2-ethoxyphenyl)methyl]piperazin-1-yl}-2-[(1-hydroxycyclohexyl)methyl]-2,3-dihydro-1H-isoindole-1,3-dione
N-{[5-(2-methylpropyl)-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl]methyl}morpholine-2-carboxamide
2-(1-butyl-5-{hydroxy[4-(trifluoromethyl)phenyl]methyl}-1H-1,2,4-triazol-3-yl)acetamide
3-({4-[4-(aminomethyl)-1H-1,2,3-triazol-1-yl]piperidin-1-yl}methyl)-6-methylquinolin-2-ol
(4aR,8aS)-1-[4-(furan-2-yl)benzoyl]-6-(2-phenylethyl)-decahydro-1,6-naphthyridine
methyl[(4-methyl-1H-imidazol-5-yl)methyl][(4-propyl-4H-1,2,4-triazol-3-yl)methyl]amine
[(1-ethyl-1H-imidazol-2-yl)methyl](methyl){[1-(3-methylbutyl)-2-(propane-2-sulfonyl)-1H-imidazol-5-yl]methyl}amine
5-{[3-(3-fluorophenyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridin-5-yl]methyl}-2,1,3-benzoxadiazole
N-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-N,2-dimethyl-[1,3]oxazolo[5,4-d]pyrimidin-7-amine
N-[(4-phenylmorpholin-2-yl)methyl]-1H-1,2,3-triazole-5-carboxamide
2-[4-(cyclohexylmethyl)-1-(3-methylbut-2-en-1-yl)piperazin-2-yl]ethan-1-ol
3-[(3R,4S)-1-[(2-methoxy-3,5-dimethylphenyl)methyl]-4-(4-methylpiperazin-1-yl)piperidin-3-yl]propan-1-ol
N-[2-(2,4-difluorophenyl)-1-[1-(3-methylthiophene-2-carbonyl)piperidin-4-yl]ethyl]-N-methylpyridine-3-carboxamide
N-{1H,4H,5H,6H,7H,8H-cyclohepta[c]pyrazol-3-ylmethyl}-N,2,7-trimethyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-benzyl-N-cyclopropyl-4-oxo-5-(4-phenylazepane-1-carbonyl)-1,4-dihydropyridine-3-carboxamide
2-methyl-4-(4-{[3-(pyrrolidine-1-carbonyl)piperidin-1-yl]methyl}phenyl)butan-2-ol
N-[3-(methylsulfanyl)propyl]-2-{[4-(pyrimidin-2-yl)piperazin-1-yl]methyl}-1,3-oxazole-4-carboxamide
N-{2-[(4,6-dimethylpyrimidin-2-yl)amino]ethyl}pyridine-3-carboxamide
(3R,4R)-3-methyl-4-(oxan-4-yl)-1-[3-(1H-1,2,3,4-tetrazol-1-yl)propyl]piperidin-4-ol
6-(difluoromethyl)-2-[3-({methyl[(3-methylthiophen-2-yl)methyl]amino}methyl)phenyl]-3,4-dihydropyrimidin-4-one
6-(4-fluorophenyl)-N-(2-methoxyethyl)-N-methyl-7-(3-methylbut-2-en-1-yl)-8-oxo-7H,8H-imidazo[1,2-a]pyrazine-2-carboxamide
N-[(3S,4R)-1-(6-chloro-1,3-benzothiazol-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]acetamide
2-(2,3-dihydro-1,4-benzodioxin-2-ylmethyl)-4-{4-[4-(furan-2-carbonyl)piperazine-1-carbonyl]piperidin-1-yl}-2,3-dihydro-1H-isoindole-1,3-dione
4-({4-methyl-5-[1-(1H-pyrazole-3-carbonyl)piperidin-4-yl]-4H-1,2,4-triazol-3-yl}methyl)morpholine
2-benzyl-8-[2-(methylsulfanyl)pyrimidin-4-yl]-2,8-diazaspiro[4.5]decan-3-one
2-[3-(diphenylmethyl)-4H,5H,6H,7H-[1,2]oxazolo[4,5-c]pyridine-5-carbonyl]pyridine
1-[3-(2-chlorophenoxy)azetidin-1-yl]-3-(dimethyl-1H-1,2,4-triazol-1-yl)-2-methylpropan-1-one
4-[7-(furan-3-carbonyl)-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl]thiomorpholine
4-[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]piperazine-2-carboxylic acid
butyl 9-oxo-8-(pyridin-3-ylmethyl)-2,8-diazaspiro[5.5]undecane-2-carboxylate
1-[(4-methoxyphenyl)methyl]-4-[4-(1H-pyrazol-1-yl)butanoyl]piperazin-2-one
2-[3-(2-phenylethyl)piperidine-1-carbonyl]pyrazine
1-[2-(4-fluorophenyl)azetidin-1-yl]-2-[(5-hydroxy-6-methyl-1,2,4-triazin-3-yl)sulfanyl]ethan-1-one
(4aR,7aS)-1-(cyclopropylmethyl)-4-{[4-(4-hydroxybut-1-yn-1-yl)phenyl]methyl}-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
N-[3-(3-ethylphenoxy)propyl]-N-methylpyridazine-3-carboxamide
N-[(3,5-dimethyl-1-propyl-1H-pyrazol-4-yl)methyl]-6-fluoro-2-oxo-1,2,3,4-tetrahydroquinoline-4-carboxamide
2-(4-hydroxypiperidin-1-yl)-N-{[1-(propan-2-yl)-1H-1,3-benzodiazol-2-yl]methyl}acetamide
N-ethyl-7-fluoro-N-[(1-methyl-1H-imidazol-2-yl)methyl]-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
N-[3-(3-chlorophenyl)phenyl]-1-cyclopentanecarbonylpiperidine-4-carboxamide