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4-[5-(1-benzofuran-2-yl)-4-phenyl-1H-imidazol-1-yl]-1-methylpiperidine
6-methyl-5-{5-[3-(5-methylfuran-2-yl)-1H-pyrazol-5-yl]-1,2,4-oxadiazol-3-yl}-1,2,3,4-tetrahydro-2,7-naphthyridine
3-(1-butyl-1H-1,2,3,4-tetrazol-5-yl)-1-{[5-(4-fluorophenyl)-1H-pyrazol-4-yl]methyl}-1-methylurea
N-[4-(pyridin-3-yloxy)phenyl]-1-(thiophen-3-ylmethyl)piperidine-2-carboxamide
9-[2-(4-methyl-1H-pyrazol-1-yl)propanoyl]-2-(prop-2-en-1-yl)-2,9-diazaspiro[5.5]undecan-3-one
3-[1-({1-methyl-4-oxo-1H,4H,5H-pyrazolo[3,4-d]pyrimidin-6-yl}methyl)piperidin-3-yl]benzoic acid
4-[(1-cyclopropanecarbonylpiperidin-4-yl)oxy]-N-[2-(2-oxo-1,3-oxazolidin-3-yl)ethyl]benzamide
4-[4-(3-acetamidopyrrolidin-1-yl)-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-2-yl]benzamide
N-[(3S,4R)-1-(2,3-dihydro-1,4-benzodioxine-6-carbonyl)-4-(5-methylfuran-2-yl)pyrrolidin-3-yl]acetamide
1-ethyl-4-[4-(pyridin-2-ylmethyl)-1,4-diazepane-1-carbonyl]pyrrolidin-2-one
4-{3-[4-methyl-5-(pyrrolidin-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}pyridine
2-[2-({[2-(1H-imidazol-1-yl)phenyl]methyl}amino)pyrimidin-4-yl]pyridine-4-carboxylic acid
1-(1-oxo-1,2-dihydroisoquinoline-4-carbonyl)-4-phenylpiperidine-4-carbonitrile
(3S,9aR)-3-benzyl-8-(cyclopropylmethyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
2-ethyl-N-[(1R,2S)-2-hydroxy-2,3-dihydro-1H-inden-1-yl]-4-methyl-1,3-oxazole-5-carboxamide
4-(3,3-dimethylpyrrolidine-1-carbonyl)-2-[1-(propan-2-yl)-1H-pyrazol-4-yl]quinoline
N-(2,3-dihydro-1-benzofuran-2-ylmethyl)-3-[2-(furan-2-ylmethyl)-5-oxopyrrolidin-2-yl]-N-methylpropanamide
(3aR,6aR)-2-cyclobutanecarbonyl-5-(4-fluorobenzoyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{3-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}-3-(oxolan-2-ylmethyl)urea
4-{[5-(pyridin-3-yl)-1,3,4-oxadiazol-2-yl]methyl}-3,4-dihydro-2H-1,4-benzothiazin-3-one
2-(2H-1,3-benzodioxol-5-yl)-N-cyclopropyl-N-[(1-methyl-1H-pyrazol-4-yl)methyl]acetamide
(3E)-N-[(5-chloro-2-methoxyphenyl)methyl]-N-ethylpent-3-enamide
8-methyl-2-{2-oxo-2-[2-(1,3-thiazol-2-yl)pyrrolidin-1-yl]ethyl}-2,8-diazaspiro[4.5]decan-3-one
6-{1-[4-(dimethylamino)-5-methylpyrimidin-2-yl]piperidin-3-yl}pyrimidin-4-ol
N-methyl-N-{[3-(methylsulfanyl)phenyl]methyl}-4-(trimethyl-1H-pyrazol-4-yl)pyrimidin-2-amine
2-(2-methoxyethyl)-6-[2-(pyridin-2-yl)pyrrolidine-1-carbonyl]-1,3-benzoxazole
(3aS,6aS)-2-cyclopentanecarbonyl-5-(2-methylpyridin-4-yl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
1-{3-[2-(4-methoxyphenyl)ethyl]piperidin-1-yl}pent-4-en-1-one
8-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-(2-phenylpropyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-[1-(2,2-dimethylpropyl)-5-oxopyrrolidin-3-yl]-4-methyl-1,2,3-thiadiazole-5-carboxamide
N-[4-(furan-2-yl)phenyl]-1-{[5-(propan-2-yl)-1,2,4-oxadiazol-3-yl]methyl}piperidine-3-carboxamide
N3-[3-(3-ethylphenoxy)propyl]-N1,N1,N3-trimethylpiperidine-1,3-dicarboxamide
9-(5,6-dimethylpyridine-3-carbonyl)-2-(oxolan-2-ylmethyl)-2,9-diazaspiro[5.5]undecan-3-one
1-methyl-2-(morpholin-4-yl)-N-[2-(2-oxoimidazolidin-1-yl)ethyl]-1H-1,3-benzodiazole-5-carboxamide
(1S,5R)-3-(5-hydroxy-1,2-dimethyl-1H-indole-3-carbonyl)-6-propyl-3,6-diazabicyclo[3.2.2]nonan-7-one
N-[(2,2-dimethyl-2,3-dihydro-1-benzofuran-5-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d]pyrimidin-4-amine
3-methyl-1-(2-methylpropyl)-4-{4-[3-(pyridin-4-yl)-1,2,4-oxadiazol-5-yl]butanoyl}piperazin-2-one
1-(2-chlorophenyl)-3-(1-{1-[(3-methylphenyl)methyl]piperidin-4-yl}-1H-pyrazol-5-yl)urea
N-{2-[(2-methylquinolin-8-yl)oxy]ethyl}imidazo[1,2-a]pyrimidine-2-carboxamide
4-[(2,5-dimethylphenyl)methyl]-1,3λ6,4-oxathiazinane-3,3-dione
3-benzyl-1-methyl-3-{2-oxo-2-[3-(1H-pyrazol-1-yl)azetidin-1-yl]ethyl}-2,3-dihydro-1H-indol-2-one
N-[2-(2-chlorophenoxy)ethyl]-2-methyl-2-(thiophen-2-ylformamido)propanamide
3-{2-[4-(4-chlorophenyl)-2-methyl-5-oxopiperazin-1-yl]-2-oxoethyl}imidazolidine-2,4-dione
3-[(3S,4R)-1-(2,2-diphenylethyl)-4-(morpholin-4-yl)piperidin-3-yl]-1-[4-(pyridin-2-yl)piperazin-1-yl]propan-1-one
5-ethyl-N-[2-(hexahydro-1H-pyrrolizin-7a-yl)ethyl]pyrimidin-2-amine
ethyl 4-[3-({[(3-chlorophenyl)methyl]amino}methyl)-6-methylquinolin-2-yl]piperazine-1-carboxylate
2,2-dimethyl-N-({1-[(2E)-2-methylbut-2-en-1-yl]piperidin-4-yl}methyl)propanamide
N-[4-(3-methoxypyrazin-2-yl)-1H-pyrrolo[2,3-b]pyridin-6-yl]piperidin-4-amine
1-[(1-{2-amino-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-yl}piperidin-3-yl)methyl]pyrrolidin-2-one
2-(1,3-benzoxazol-2-yl)-N-{[4-(morpholin-4-yl)phenyl]methyl}acetamide