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5-fluoro-N-({1-[2-(2-methoxyphenyl)ethyl]piperidin-3-yl}methyl)-N-methyl-1H-indole-2-carboxamide
6-(4H-1,2,4-triazol-4-yl)-N-[2,2,2-trifluoro-1-(pyridin-3-yl)ethyl]pyridine-3-carboxamide
3-{3-[4-(4-methylphenyl)-1H-pyrazol-5-yl]piperidine-1-carbonyl}pyridin-2-ol
3-[(3R,7S,8aS)-3-[(1S)-1-hydroxyethyl]-1,4-dioxo-octahydropyrrolo[1,2-a]piperazin-7-yl]-1-phenylurea
N-cyclopentyl-3-{[(5-methylthiophen-2-yl)methyl]amino}-5-(phenylsulfamoyl)benzamide
N3-(cyclopropylmethyl)-1-(2-methoxyethyl)-4-oxo-N5-[(1-phenylcyclopentyl)methyl]-1,4-dihydropyridine-3,5-dicarboxamide
3-[3-(3,5-dimethyl-1H-pyrazol-1-yl)propyl]-3-methyl-1-(2-methyl-5-sulfamoylphenyl)urea
3-(quinolin-3-yl)-5-(thiomorpholine-4-sulfonyl)benzoic acid
6-chloro-2-{[4-(1-methyl-1H-imidazol-2-yl)-1H,4H,5H,6H,7H-imidazo[4,5-c]pyridin-5-yl]methyl}quinoline
3-{[1-(6-methylpyridin-2-yl)-1H,2H,3H,4H,9H-pyrido[3,4-b]indol-2-yl]methyl}phenol
N-(3,4-dimethylphenyl)-1-(pyridine-3-sulfonyl)piperidin-3-amine
methyl 4-{4-oxo-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(15),3(8),6,11,13-pentaen-6-yl}piperazine-1-carboxylate
3-chloro-4-({1-[(2-ethyl-4-methyl-1H-imidazol-5-yl)methyl]piperidin-4-yl}oxy)-N-(2-methoxyethyl)benzamide
6-[2-(1-methyl-1H-1,3-benzodiazol-2-yl)pyrrolidine-1-carbonyl]-1,3-benzothiazole
(2R,6R)-11-methoxy-4-[2-(1-methyl-1H-imidazol-2-yl)ethyl]-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-triene-6-carboxylic acid
4-benzyl-3-(1-cyclobutanecarbonylpiperidin-4-yl)-4,5-dihydro-1H-1,2,4-triazol-5-one
N-{[7-chloro-5-(thiophen-3-yl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(3-methyl-1H-pyrazol-1-yl)acetamide
4-(2-methyl-1H-imidazol-1-yl)-1-(1,3-thiazol-2-yl)piperidine-4-carboxylic acid
7-[(2,3-difluorophenyl)methyl]-2-(1-methyl-1H-imidazole-2-carbonyl)-2,7-diazaspiro[4.5]decane
3-methoxy-N-methyl-N-[(3-methyl-1,2,4-oxadiazol-5-yl)methyl]-4-[(1-methylpiperidin-4-yl)oxy]benzamide
2-[(5-fluoro-1H-1,3-benzodiazol-2-yl)methoxy]-N-methyl-N-[2-(4-methyl-1,3-thiazol-5-yl)ethyl]acetamide
3-[5-(2-methylpropyl)-4H-1,2,4-triazol-3-yl]-1-{[2-(thiophen-2-yl)-1,3-thiazol-4-yl]methyl}urea
8-{[3-methyl-1-(prop-2-en-1-yl)-1H-pyrazol-4-yl]methyl}-3-(2-phenoxyethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
N-(1,3-dihydroxypropan-2-yl)-2-{1-[(5-methylfuran-2-yl)methyl]-3-oxopiperazin-2-yl}acetamide
3-{2-oxo-2-[4-(thiophene-2-carbonyl)piperazin-1-yl]ethyl}-4-(propan-2-yl)piperazin-2-one
[4-({1-[3-(trifluoromethyl)-1H-pyrazole-5-carbonyl]pyrrolidin-3-yl}methyl)phenyl]methanol
N-[(5-methylpyrazin-2-yl)methyl]-3-(pyrrolidin-3-yl)benzamide
2-(4-{[1-(1,3-thiazol-2-yl)-1H-pyrrol-2-yl]methyl}-1-(thiophen-3-ylmethyl)piperazin-2-yl)ethan-1-ol
1-[2-(4-chlorophenyl)ethyl]-6-oxopiperidine-3-carboxylic acid
N-[4-(3,5-dimethyl-1H-pyrazol-1-yl)phenyl]-1-[3-(methylsulfanyl)propyl]piperidine-2-carboxamide
2-[(1,5-dimethyl-1H-pyrazol-4-yl)methyl]-4-[4-(5-methylthiophene-2-carbonyl)piperazin-1-yl]-2,3-dihydro-1H-isoindole-1,3-dione
N-[(1R,3R)-3-aminocyclopentyl]-4-methoxy-5,6,7,8-tetrahydronaphthalene-1-sulfonamide
1-(4-{[(1,3-dimethyl-1H-pyrazol-5-yl)methyl]amino}-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-7-yl)-2-methoxyethan-1-one
N-(2-methoxyethyl)-5-{1-[(1-methyl-1H-indol-2-yl)methyl]pyrrolidin-2-yl}thiophene-2-carboxamide
5-(2-methylpropanoyl)-N-(pyridin-2-ylmethyl)-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-2-carboxamide
1-(2-chlorophenyl)-3-{[1-(furan-2-ylmethyl)pyrrolidin-3-yl]methyl}urea
4,6-dimethyl-2-oxo-5-(3-{4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}propanamido)-1,2-dihydropyridine-3-carboxamide
N-[3-hydroxy-3-(prop-2-en-1-yl)hex-5-en-2-yl]-5-methoxyfuran-2-carboxamide
2-[5-(2-methylpropanoyl)thiophen-2-yl]benzamide
4-amino-1-[9-hydroxy-7-(5-methylthiophen-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]butan-1-one
N-cyclopropyl-6-(4-fluoro-2-methoxyphenyl)pyridazin-3-amine
(3S)-1-benzyl-N-[1-methyl-6-(pyridin-3-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]pyrrolidin-3-amine
2-(4-chlorophenyl)-5-{[4-(pyridin-3-ylmethyl)piperazin-1-yl]methyl}pyrimidine
2-(4-{4-[(1-methyl-1H-imidazol-2-yl)methyl]piperazine-1-carbonyl}piperidin-1-yl)acetamide
2-(4-{3,9-diazaspiro[5.5]undecan-3-ylmethyl}phenoxy)-1-(pyrrolidin-1-yl)ethan-1-one
1-(furan-2-ylmethyl)-N-{[4-(1H-1,2,4-triazol-1-yl)phenyl]methyl}piperidine-4-carboxamide
1-{[3-(2-phenylethyl)-1-(propan-2-yl)-1H-1,2,4-triazol-5-yl]methyl}piperidin-2-one
methyl 4-({[(3S,5S)-5-(ethylcarbamoyl)-1-(propan-2-yl)pyrrolidin-3-yl]amino}methyl)benzoate
N-(3-methylphenyl)-3-{1-[2-(phenylsulfanyl)acetyl]piperidin-4-yl}propanamide
N-{5H,6H,7H-cyclopenta[d]pyrimidin-2-ylmethyl}-3-(3-phenyl-1,2,4-oxadiazol-5-yl)propanamide