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4-[3-(oxan-4-yl)-5-(pyrrolidin-3-yl)-1H-1,2,4-triazol-1-yl]benzonitrile
(3aR,6aR)-2-acetyl-5-(9H-fluoren-2-ylmethyl)-octahydropyrrolo[3,4-c]pyrrole-3a-carboxylic acid
4-(4-{[(butan-2-yl)(pyridin-3-ylmethyl)amino]methyl}phenyl)-2-methylbut-3-yn-2-ol
N-(2-{4-[3-(4-methylpiperazine-1-carbonyl)piperidin-1-yl]piperidin-1-yl}-2-oxoethyl)acetamide
1-{[1-(5-chloropyridin-2-yl)-1H-pyrrol-2-yl]methyl}-4-ethyl-1,4-diazepan-5-one
N6-benzyl-N5-methyl-N5-[(2-methyl-1,3-thiazol-4-yl)methyl]-[1,2,5]oxadiazolo[3,4-b]pyrazine-5,6-diamine
2-(morpholin-3-yl)-N-[(2-phenyl-1,3-oxazol-4-yl)methyl]acetamide
(4aS,7aR)-1-(2-chloro-5-methylbenzoyl)-4-(2-hydroxyethyl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-cycloheptyl-6-oxopiperidine-3-carboxylic acid
3-phenyl-N-{2-[6-(pyrrolidin-1-yl)pyrimidin-4-yl]ethyl}-1,2-oxazole-4-carboxamide
4-({4-[4-ethyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]piperidin-1-yl}methyl)-1-methyl-1H-pyrrole-2-carbonitrile
8-methyl-N-(naphthalen-1-ylmethyl)-2-propyl-2,8-diazaspiro[4.5]decane-3-carboxamide
2-[5-(1-methyl-1H-imidazol-2-yl)-4-phenyl-1H-imidazol-1-yl]-1-(piperazin-1-yl)ethan-1-one
N,N-dimethyl-2-{[(quinoxalin-2-yl)amino]methyl}-4H,5H,6H,7H-pyrazolo[1,5-a]pyrazine-5-carboxamide
3-({[1-(carbamoylmethyl)-2-methyl-1H-indol-3-yl]methyl}amino)-N-(2,5-dimethylphenyl)propanamide
(3R,9aR)-3-[(benzylsulfanyl)methyl]-8-[4-(trifluoromethyl)benzoyl]-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
4-[4-cyclopropyl-5-(1H-pyrazol-1-ylmethyl)-4H-1,2,4-triazol-3-yl]-1-(1-methyl-1H-pyrrole-2-carbonyl)piperidine
1-{[2-(3-chlorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-2-methylpiperazine
N-(dimethyl-1,2-oxazol-4-yl)-5-{1-[(2E)-4-methylpent-2-en-1-yl]pyrrolidin-2-yl}thiophene-2-carboxamide
methyl 2-{N-methyl-2-[2-methyl-4-oxo-1-(2-phenylethyl)-4,5,6,7-tetrahydro-1H-indol-3-yl]acetamido}acetate
N-cyclopropyl-4-[1-(2,3-dimethylphenyl)piperidin-4-yl]piperazine-2-carboxamide
1-{4-[(5-methyl-1H-1,2,3,4-tetrazol-1-yl)methyl]benzoyl}-4-(pyrrolidine-1-carbonyl)piperidine
6-(1-{2-chloro-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}piperidin-3-yl)-2-methyl-3,4-dihydropyrimidin-4-one
N-[(1-methyl-1H-pyrazol-4-yl)methyl]-N-(2-methylpropyl)cyclopentanecarboxamide
3-(methylsulfanyl)-1-{3-[4-(trifluoromethyl)phenyl]-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl}propan-1-one
N-{[4-(4-fluorophenyl)-5-(methylsulfanyl)-4H-1,2,4-triazol-3-yl]methyl}-2,3,4-trimethoxybenzamide
4-{[3-(3-methoxyphenyl)-1,2-oxazol-5-yl]methyl}-1-(1H-1,2,3-triazole-5-carbonyl)piperidin-4-ol
2-(cyclopropylmethyl)-7-[(3-hydroxypiperidin-3-yl)methyl]-3H,4H,5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-one
1-[(3R,4R)-3-hydroxy-4-methyl-3-(propan-2-yl)pyrrolidin-1-yl]-2-(1,3-thiazol-4-yl)ethan-1-one
1-methyl-4-[2-(2-oxo-1,2-dihydropyridin-1-yl)acetyl]-1,4,9-triazaspiro[5.6]dodecan-10-one
5-{[(1S,5R)-3-[(4-fluorophenyl)methyl]-3,6-diazabicyclo[3.2.2]nonan-6-yl]methyl}-N-methyl-1,2,4-oxadiazole-3-carboxamide
3-[1-(3-cyclopropyl-1,2,4-oxadiazol-5-yl)ethyl]-1-[2-methoxy-5-(5-methyl-1,3,4-oxadiazol-2-yl)phenyl]urea
3-[(5-methylthiophen-2-yl)methyl]-1-{4-[2-(morpholin-4-yl)-2-oxoethoxy]phenyl}urea
2-{[5-(methoxymethyl)furan-2-yl]methyl}-7-[(3-methoxyphenyl)methyl]-2,7-diazaspiro[4.5]decan-6-one
1-{1,9-dimethyl-10-oxo-1,4,9-triazaspiro[5.6]dodecan-4-yl}-2-(1-methyl-1H-pyrrol-2-yl)ethane-1,2-dione
(2S)-N-(2,3-dihydro-1H-inden-2-yl)-2-acetamido-4-(methylsulfanyl)butanamide
1-{[4-(furan-3-ylmethyl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-7-yl]methyl}piperidin-4-ol
N-(cyclopropylmethyl)-8-methyl-N-propyl-2-(1H-pyrazol-4-yl)quinoline-4-carboxamide
7-[(2E)-3-(4-methoxyphenyl)prop-2-en-1-yl]-2-methyl-2,7-diazaspiro[4.5]decane
1-[1,3-dimethyl-6-(pyridin-4-yl)-1H-pyrazolo[3,4-d]pyrimidin-4-yl]-3-phenylpiperazine
{[2-(4-methoxy-2,5-dimethylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(methyl)[(3-phenyl-1,2,4-oxadiazol-5-yl)methyl]amine
N-[2-(dimethylamino)ethyl]-N-methyl-5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-amine
4-{[(1S,5R)-6-(cyclopropylmethyl)-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]methyl}benzoic acid
2-(3-hydroxypropyl)-9-[2-(4-methyl-1H-pyrazol-1-yl)acetyl]-2,9-diazaspiro[5.5]undecan-3-one
2-(3-methyl-1H-1,2,4-triazol-5-yl)-N-(4-pentylphenyl)pyrrolidine-1-carboxamide
3-(morpholine-4-carbonyl)-N-(naphthalen-1-ylmethyl)-1-(prop-2-en-1-yl)-4,5,6,7-tetrahydro-1H-indazol-5-amine
7-chloro-1-methyl-N-[(5-methylpyrazin-2-yl)methyl]-1H-indole-2-carboxamide
1-[2-({methyl[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]amino}methyl)phenoxy]-3-(piperidin-1-yl)propan-2-ol
N-[(5-cyclopropyl-1H-pyrazol-3-yl)methyl]-1,3-dimethyl-1H-pyrazolo[3,4-d][1,3]thiazol-5-amine
2-{3-[6-amino-5-cyano-4-(pyridin-3-yl)pyridin-2-yl]-1H-indol-1-yl}propanoic acid