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5-({[2-amino-6-methyl-5-(prop-2-en-1-yl)pyrimidin-4-yl]amino}methyl)-1,2,3,4-tetrahydropyrimidine-2,4-dione
3-{2-[3-(oxolan-3-yl)-1,2,4-oxadiazol-5-yl]ethyl}pyridine
2-cyclopropyl-4-phenyl-9-(pyridin-4-ylmethyl)-2,9-diazaspiro[5.5]undecane
N-{1-[4-(3-methoxypropyl)-4H-1,2,4-triazol-3-yl]ethyl}imidazo[2,1-b][1,3]thiazole-6-carboxamide
8-(pyridin-2-ylmethyl)-1-oxa-8-azaspiro[4.6]undecan-9-one
7-methoxy-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-3,4-dihydro-2H-1-benzopyran-3-carboxamide
4-methyl-N-(2-{[(4-methyl-1H-imidazol-5-yl)methyl]sulfanyl}ethyl)-3-(2-oxoimidazolidin-1-yl)benzamide
N-[1-(1H-1,2,4-triazol-5-yl)ethyl]-2-(2,3,6-trimethylphenoxy)acetamide
4-(pyridin-3-yl)-1-[2-(pyrrolidin-3-yl)benzoyl]piperidin-4-ol
N-(1-tert-butyl-4-phenyl-1H-pyrazol-5-yl)thiomorpholine-4-carboxamide
N-(3,4-difluorophenyl)-5-[1-(furan-2-ylmethyl)-4-hydroxypiperidin-4-yl]-1-benzofuran-2-carboxamide
5-{4-[(4-propyl-1H-1,2,3-triazol-1-yl)methyl]piperidine-1-carbonyl}pyrazin-2-ol
2-{1-[(2,3-difluorophenyl)methyl]-3-oxopiperazin-2-yl}-N-methyl-N-[(3-methyl-1H-indol-2-yl)methyl]acetamide
5-(2H-1,3-benzodioxol-5-ylmethyl)-1-{[5-(methoxymethyl)-1H-pyrazol-3-yl]methyl}-5-methylpiperidin-2-one
3-(4-methoxyphenyl)-5-{[1,2,3,4]tetrazolo[1,5-a]pyridine-6-carbonyl}-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridine
5-(4-cyclohexyl-1,4-diazepane-1-carbonyl)-N-(thiophen-3-ylmethyl)pyridin-2-amine
7-[5-fluoro-4-(pyrrolidin-1-yl)pyrimidin-2-yl]-3-methyl-1-oxa-3,7-diazaspiro[4.5]decan-2-one
1-[3-(dimethylamino)phenyl]-3-[2-(pyrrolidine-1-sulfonyl)ethyl]urea
1-(4-methyl-1,2,3-thiadiazole-5-carbonyl)-4-[(2-methylphenyl)sulfanyl]piperidine
(3aR,6aR)-2-cyclopropanecarbonyl-N-[(3,5-dimethyl-1H-pyrazol-4-yl)methyl]-octahydropyrrolo[3,4-c]pyrrole-3a-carboxamide
(2S,4S)-4-amino-N-[(1R)-1-(3-methoxyphenyl)ethyl]-1-methylpyrrolidine-2-carboxamide
1-[({3-hydroxy-1-[(3-methoxyphenyl)methyl]-2-oxopiperidin-3-yl}methyl)amino]cyclohexane-1-carboxamide
N-benzyl-4-(pyridin-3-ylmethoxy)piperidine-1-sulfonamide
2-(2-ethylpyrimidin-5-yl)-7-methyl-4-(2-methylpiperidine-1-carbonyl)quinoline
(1S,5R)-3-[2-(phenylsulfanyl)ethyl]-6-(pyridin-2-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
2-amino-N,4-dimethyl-N-[2-(1,2,4-oxadiazol-3-yl)ethyl]pyrimidine-5-carboxamide
2-[6-oxo-4-(pyrrolidin-1-yl)-1,6-dihydropyridazin-1-yl]-N-[4-(1H-pyrazol-1-yl)phenyl]acetamide
{[3-(1-benzofuran-2-yl)-1-benzyl-1H-pyrazol-4-yl]methyl}[(1,3-dimethyl-1H-pyrazol-4-yl)methyl]methylamine
1-[6-(2-fluoro-6-methoxyphenyl)pyridin-2-yl]piperazine
1-methyl-1-{2-oxo-2-[3-oxo-2-(2-phenylethyl)-2,9-diazaspiro[5.5]undecan-9-yl]ethyl}urea
(furan-2-ylmethyl)({[2-(4-methoxy-3-methylphenyl)-5-methyl-1,3-oxazol-4-yl]methyl})(prop-2-yn-1-yl)amine
{1-[(1-methyl-1H-1,3-benzodiazol-2-yl)methyl]-3-(2-phenylethyl)piperidin-3-yl}methanol
4-hydroxy-N,2-dimethyl-N-{[3-(thiophen-2-yl)-1H-pyrazol-5-yl]methyl}pyrimidine-5-carboxamide
N-(2-methoxyethyl)-2-methyl-4-phenyl-N-propylpyridine-3-carboxamide
5-{1-[(2,6-difluorophenyl)methyl]-1H-1,2,3-triazol-4-yl}-2-(ethylsulfanyl)pyrimidine
1-[(5-chloro-3-ethyl-1-methyl-1H-pyrazol-4-yl)methyl]-4-(1H-pyrrole-2-carbonyl)piperazine
2-[1-(furan-3-ylmethyl)-3-oxopiperazin-2-yl]-N-[2-(pyridin-3-yloxy)ethyl]acetamide
(3R,4R)-4-(azepan-1-yl)-1-{[1-(3-chlorophenyl)-1H-pyrazol-4-yl]methyl}piperidin-3-ol
1-[4-(methylsulfanyl)phenyl]-2-{4H,5H,6H,7H-pyrazolo[1,5-a]pyrazin-2-yl}-1H-imidazole
4-(4-amino-5-methylpyrimidin-2-yl)-7-(3,6-dimethylpyrazin-2-yl)-2,3,4,5-tetrahydro-1,4-benzoxazepin-9-ol
(2S,4S)-4-amino-N-methyl-1-{2-[4-(1H-1,2,3,4-tetrazol-1-yl)phenoxy]acetyl}pyrrolidine-2-carboxamide
1-phenyl-2-{[5-(propan-2-yl)pyrazolo[1,5-a]pyrimidin-7-yl]amino}ethan-1-ol
N-{[7-chloro-5-(2,5-dimethoxyphenyl)-2,3-dihydro-1-benzofuran-2-yl]methyl}-2-(pyridin-4-ylsulfanyl)acetamide
1-(benzenesulfonyl)-3-[1-(propan-2-yl)-1H-imidazol-2-yl]piperidine
7-methyl-3-{[1-(pyridin-2-yl)-1H,2H,3H,4H-pyrrolo[1,2-a]pyrazin-2-yl]methyl}-1,2-dihydroquinolin-2-one
N-[(3R,4S)-1-(3-chloropyridin-2-yl)-4-(propan-2-yl)pyrrolidin-3-yl]methanesulfonamide
N-methyl-6-(morpholin-4-yl)-N-[2-(1,2,3,4-tetrahydroisoquinolin-2-yl)ethyl]-[1,2,5]oxadiazolo[3,4-b]pyrazin-5-amine
2-[4-(cyclobutylmethyl)piperazin-1-yl]-4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]pyrimidine
2-[(1-phenyl-1H-pyrazol-5-yl)methyl]-2,8-diazaspiro[4.5]decane
5-(3-fluorophenoxymethyl)-N-[1-(1H-1,2,3,4-tetrazol-5-yl)ethyl]-1H-pyrazole-3-carboxamide