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[(1R,3S,3aS,6aR)-1,5-dimethyl-3-{2-[2-(4-methylpiperazin-1-yl)ethoxy]phenyl}-octahydropyrrolo[3,4-c]pyrrol-1-yl]methanol
4-{2-[(4-fluorophenyl)methyl]-3H-imidazo[4,5-b]pyridin-3-yl}-1-[4-(1H-imidazol-1-yl)benzoyl]piperidine
N-(propan-2-yl)-1-(1-propylpiperidin-3-yl)-1H-1,2,3-triazole-4-carboxamide
6-{[(1-propyl-1H-pyrazol-4-yl)methyl]amino}-10-oxa-5,7-diazatricyclo[9.4.0.03,8]pentadeca-1(11),3(8),6,12,14-pentaen-4-one
4-{[3-(1H-pyrazol-1-yl)phenyl]methyl}-4H-1,2,4-triazole
2-(pyridin-3-yl)-6-(pyrrolidine-1-carbonyl)pyrazine
2-(4-{[(3S)-3-ethylmorpholin-4-yl]methyl}phenyl)acetic acid
3-(piperidine-1-carbonyl)-1-(5-propyl-1,3,4-oxadiazol-2-yl)piperidine
[(3R,4R)-1-(5-methylpyrazine-2-carbonyl)-4-(pyrrolidin-1-ylmethyl)pyrrolidin-3-yl]methanol
1-[(2S,6S)-6-(hydroxymethyl)-8-oxa-4-azatricyclo[7.4.0.02,6]trideca-1(13),9,11-trien-4-yl]-2-[methyl(pyridin-2-ylmethyl)amino]ethan-1-one
1-(4-methoxyphenyl)-4-[1-(6-methylpyridine-2-carbonyl)piperidin-3-yl]piperazine
5-ethyl-N-({5-methanesulfonyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepin-2-yl}methyl)-1,2-oxazole-3-carboxamide
7-[1-ethyl-3-(2-methylpropyl)-1H-pyrazole-5-carbonyl]-N,N,2-trimethyl-5H,6H,7H,8H-pyrido[3,4-d]pyrimidin-4-amine
1-(3,5-dimethylphenyl)-4-[6-(1-hydroxyethyl)pyridin-2-yl]piperazin-2-one
1-[2-methoxy-4-({[3-(morpholin-4-yl)propyl]amino}methyl)phenoxy]-3-(thiomorpholin-4-yl)propan-2-ol
1-[3-(4-methyl-1H-1,3-benzodiazol-2-yl)piperidin-1-yl]-3-(pyridin-3-yl)propan-1-one
(3R,4R)-3-cyclopropyl-4-methyl-1-(4-propyl-1,2,3-thiadiazole-5-carbonyl)pyrrolidin-3-ol
1-{2-methoxy-5H,6H,7H-cyclopenta[b]pyridine-3-carbonyl}-3-[3-(propan-2-yl)-1,2,4-oxadiazol-5-yl]piperidine
ethyl({[5-(methoxymethyl)furan-2-yl]methyl})({1-[2-(2-methylphenyl)ethyl]piperidin-4-yl}methyl)amine
1-(5-cyclopropyl-1-{4-[2-(trifluoromethyl)phenyl]pyrimidin-2-yl}-1H-pyrazole-4-carbonyl)-N,N-diethylpyrrolidin-3-amine
methyl 5-[7-(cyclohexylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-5-oxopentanoate
5-(2-chloro-4-methoxyphenoxymethyl)-N-(2,2-dimethylpropyl)-1,2-oxazole-3-carboxamide
1-{4-[({1-[(2-fluorophenyl)methyl]piperidin-4-yl}methyl)(oxolan-2-ylmethyl)amino]piperidin-1-yl}ethan-1-one
6-[3-(2,5-dimethoxyphenyl)-5-(1H-1,2,3,4-tetrazol-1-yl)benzoyl]-1,3,3-trimethyl-6-azabicyclo[3.2.1]octane
2-[3-(3,4-difluorophenyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-N-(2-methylbutan-2-yl)acetamide
7-[(2E)-hex-2-en-1-yl]-2,3-dimethyl-3H,4H,5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-one
2-phenyl-N-{[7-(quinolin-8-ylmethyl)-5H,6H,7H,8H,9H-[1,2,4]triazolo[4,3-d][1,4]diazepin-3-yl]methyl}acetamide
5-[2-(3-methyl-1,2-oxazol-5-yl)pyrrolidine-1-carbonyl]-N-phenylpyrimidin-2-amine
1-(2-methyl-1-benzofuran-5-carbonyl)-4-{[1,2,4]triazolo[4,3-a]pyridin-3-yl}piperidine
3-(2-oxo-2-{2-[5-(propan-2-yl)-1,2-oxazol-3-yl]pyrrolidin-1-yl}ethyl)-1-oxa-3,8-diazaspiro[4.5]decan-2-one
2-methyl-4-[3-(2-phenylethyl)piperidine-1-carbonyl]-1H-1,3-benzodiazole
(3S,4S)-1-{[4-ethoxy-3-(prop-2-en-1-yl)phenyl]methyl}-4-(4-methylpiperazin-1-yl)pyrrolidin-3-ol
2-methyl-4-phenyl-9-(thiophene-2-carbonyl)-2,9-diazaspiro[5.5]undecan-3-one
2-chloro-5-acetamido-N-[(5-methylpyrazin-2-yl)methyl]benzamide
2-(pyridin-2-yl)-1-[1-(2,3,4-trimethoxybenzoyl)piperidin-4-yl]-1H-1,3-benzodiazole
{3-[(3-chlorophenyl)methyl]-1-[(2,4,5-trimethoxyphenyl)methyl]piperidin-3-yl}methanol
2-ethyl-9-{[4-(propan-2-yl)-4H-1,2,4-triazol-3-yl]methyl}-2,9-diazaspiro[5.5]undecan-3-one
(1R,5R)-N,N-dimethyl-6-[(1-methyl-1H-imidazol-2-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane-3-sulfonamide
N-{2-[(4-ethyl-5-methyl-4H-1,2,4-triazol-3-yl)sulfanyl]ethyl}-2-methyl-1-benzofuran-5-carboxamide
1-[(5-ethyl-1,3,4-oxadiazol-2-yl)methyl]-N-[3-(1H-1,2,3,4-tetrazol-1-yl)phenyl]piperidine-3-carboxamide
1-(3-phenylpropyl)-3-[3-(piperidine-1-carbonyl)phenyl]urea
3-[(4aS,7aR)-4-(2-methoxyethyl)-6,6-dioxo-octahydro-6λ6-thieno[3,4-b]piperazin-1-yl]-N-tert-butylpropanamide
5-acetyl-N-[1-(4-methanesulfonylphenyl)propyl]thiophene-3-carboxamide
9-(5-tert-butyl-1,3,4-oxadiazol-2-yl)-1-oxa-9-azaspiro[5.5]undecan-5-ol
N-(2-methylpropyl)-5-[1-(2-methylpropyl)pyrrolidin-2-yl]thiophene-2-carboxamide
2-(1-methyl-1H-pyrazol-3-yl)-1-[5-(propan-2-yl)-1,2-oxazole-3-carbonyl]piperidine
N-{1-[1-(2,2-difluoroethyl)piperidin-4-yl]-1H-pyrazol-5-yl}-3-phenoxypropanamide
4-[7-(cyclopropylmethyl)-6-oxo-2,7-diazaspiro[4.5]decan-2-yl]-2-methoxypyridine-3-carbonitrile
5-{[3-cyclopropyl-1-(2,3-dihydro-1,4-benzodioxin-6-yl)-1H-1,2,4-triazol-5-yl]methyl}-2,6-dimethyl-3,4-dihydropyrimidin-4-one
7-(pyridin-3-ylmethyl)-2-[2-(thiophen-3-yl)acetyl]-2,7-diazaspiro[4.5]decan-6-one