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ethyl[(1-methyl-1H-imidazol-2-yl)methyl]{[3-(1H-1,2,4-triazol-5-yl)phenyl]methyl}amine
4-[3-(4-fluorophenyl)-1H-pyrazol-4-yl]-2H,4H,5H,6H,7H-pyrazolo[3,4-b]pyridin-6-one
1-(2-ethoxyethyl)-N-[(2-fluorophenyl)methyl]-2-oxo-2,3-dihydro-1H-1,3-benzodiazole-5-carboxamide
1-{4-[(2-hydroxy-3-methoxyphenyl)methyl]-1,4-diazepan-1-yl}-2-methoxyethan-1-one
[2-(6-methyl-2-phenylpyrimidin-4-yl)phenyl]methanol
1-[3-(4-methyl-1H-pyrazol-1-yl)propyl]-1,2-dihydroquinolin-2-one
2-{2-[4-(1-hydroxypropyl)piperidin-1-yl]pyrimidin-4-yl}pyridine-4-carboxylic acid
(1R,5R)-3-benzoyl-6-[(3-ethyl-1,2-oxazol-5-yl)methyl]-3,6-diazabicyclo[3.2.2]nonane
1-[2-(3-fluorophenyl)ethyl]-6-oxo-N-[2-(pyridin-3-yl)ethyl]piperidine-3-carboxamide
9-(4-methylbenzoyl)-2-[(1r,4r)-4-hydroxycyclohexyl]-2,9-diazaspiro[5.5]undecan-3-one
N-[6,6-dimethyl-1-(2-methylphenyl)-4,5,6,7-tetrahydro-1H-indazol-4-yl]-2-(methylsulfanyl)acetamide
3-(3-hydroxy-3-methylbutyl)-N-{[2-(1H-pyrazol-1-yl)phenyl]methyl}benzamide
4-hydroxy-2-({[(1-methyl-1H-pyrazol-4-yl)methyl](2-methylpropyl)amino}methyl)quinoline-6-carboxamide
5-fluoro-2-(1-{[3-(phenoxymethyl)-1,2,4-oxadiazol-5-yl]methyl}piperidin-4-yl)-1H-1,3-benzodiazole
4-benzyl-3-[1-(5-oxopyrrolidine-3-carbonyl)piperidin-4-yl]-4,5-dihydro-1H-1,2,4-triazol-5-one
2-(dimethylamino)-8-[2-methoxy-5-(propan-2-yl)phenyl]-4H,5H,6H,7H,8H-[1,3]thiazolo[4,5-c]azepin-6-one
N-(3-hydroxypropyl)-1-{1-[(4-methylphenyl)methyl]piperidin-3-yl}-1H-1,2,3-triazole-4-carboxamide
1-(2-{4-[1-(2-methylphenyl)-1H-pyrazol-4-yl]-1,2,3,6-tetrahydropyridin-1-yl}ethyl)-2,3-dihydro-1H-imidazol-2-one
(2R,3R,6R)-5-(1-ethyl-3-methyl-1H-pyrazole-5-carbonyl)-3-phenyl-1,5-diazatricyclo[5.2.2.02,6]undecane
N-[2-(5-methyl-1,2-oxazole-4-carbonyl)-1,2,3,4-tetrahydroisoquinolin-7-yl]-3-(4-methylphenyl)propanamide
3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-1,3,8-triazaspiro[4.5]decane-2,4-dione
(4aR,7aS)-1-(2-hydroxyethyl)-4-[2-(2-methylphenyl)acetyl]-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
1-[7-(3-chlorophenyl)-9-methoxy-2,3,4,5-tetrahydro-1,4-benzoxazepin-4-yl]-2-(5-methyl-1H-pyrazol-1-yl)ethan-1-one
2-[(1S,5R)-6-[(dimethyl-1,2-oxazol-4-yl)methyl]-7-oxo-3,6-diazabicyclo[3.2.2]nonan-3-yl]pyridine-4-carbonitrile
1-(4-tert-butylphenyl)-3-[2-(2-ethyl-1H-imidazol-1-yl)ethyl]urea
2-methyl-4-{[3-(2-methylphenoxy)azetidin-1-yl]methyl}-1,3-oxazole
N-[2-(4-fluorophenyl)-1-[1-(4-phenylbenzoyl)piperidin-4-yl]ethyl]-2-methoxy-N-methylacetamide
4-(1-cyclopropyl-6-oxopiperidine-3-carbonyl)-1-[(3-fluorophenyl)methyl]piperazin-2-one
1-[2-(2-methoxyethoxy)phenyl]-3-[2-oxo-2-(pyrrolidin-1-yl)ethyl]urea
N-[(1-ethylpyrrolidin-2-yl)methyl]-N-{[1-(2-methoxyethyl)piperidin-4-yl]methyl}-3-(1H-1,2,4-triazol-1-yl)propanamide
N-{[5-fluoro-2-(trifluoromethyl)phenyl]methyl}-3-(3-methoxyphenyl)-1H-pyrazole-5-carboxamide
5-chloro-N-[3-(1H-indazol-1-yl)propyl]-2-oxo-1,2-dihydropyridine-3-carboxamide
4-[3-(1H-imidazol-2-yl)piperidine-1-carbonyl]-6-(2-methylpropyl)pyrimidin-2-amine
1-tert-butyl-5-(cyclopent-3-en-1-yl)-3-(oxan-4-yl)-1H-1,2,4-triazole
2-[3-(1H-1,2,3-benzotriazol-1-yl)propanoyl]-7-(2-methoxyethyl)-2,7-diazaspiro[4.5]decan-6-one
(4aS,7aR)-1-{[2-(methylamino)-1,3-thiazol-4-yl]methyl}-4-(pyrimidin-2-yl)-octahydro-6λ6-thieno[3,4-b]piperazine-6,6-dione
methyl 2-{[(2R,6S)-2,6-dimethylmorpholin-4-yl]sulfonyl}-6-(2-phenylacetyl)-4H,5H,6H,7H-thieno[2,3-c]pyridine-3-carboxylate
2-(2-methoxyphenyl)-1-{1-[2-(1H-pyrazol-1-yl)phenyl]ethyl}-1H-imidazole
2-(3,5-dimethyl-1H-pyrazol-4-yl)-2-(naphthalen-1-ylformamido)acetic acid
2-(2-oxo-1,2-dihydropyridin-1-yl)-N-[3-(1,2,3,4-tetrahydroquinolin-1-yl)propyl]acetamide
8-[(5-cyclopentyl-1,2,4-oxadiazol-3-yl)methyl]-2-(propan-2-yl)-2,8-diazaspiro[5.5]undecan-3-one
N-[(3R,4S)-4-cyclopropyl-1-{[5-(methoxymethyl)-1,2,4-oxadiazol-3-yl]methyl}pyrrolidin-3-yl]ethane-1-sulfonamide
2-[3,5-dimethyl-4-({methyl[(5-methylfuran-2-yl)methyl]amino}methyl)-1H-pyrazol-1-yl]ethan-1-ol
2-[1-(2-phenylethyl)-5-[4-(4H-1,2,4-triazol-4-yl)phenyl]-1H-1,2,4-triazol-3-yl]acetamide
N-{[7-methoxy-2-(morpholin-4-yl)quinolin-3-yl]methyl}-N-[3-(2-oxopyrrolidin-1-yl)propyl]cyclohexanecarboxamide
1-cyclopentyl-N-[2-(5-cyclopentyl-1,2,4-oxadiazol-3-yl)ethyl]piperidine-3-carboxamide
N-methyl-N-[(4-methyl-1,3-thiazol-2-yl)methyl]-2-[(prop-2-en-1-yl)amino]benzamide
1-benzyl-N-(2,2-dimethyloxan-4-yl)-5-methanesulfonamido-2-methyl-1H-1,3-benzodiazole-7-carboxamide
2-cyclopropyl-N-methyl-6-oxo-N-[1-(5-phenyl-1H-pyrazol-3-yl)ethyl]-1,6-dihydropyrimidine-5-carboxamide
N-({3-methoxy-4-[2-(4-methyl-1,3-thiazol-5-yl)ethoxy]phenyl}methyl)-N-[(3S)-2-oxoazepan-3-yl]cyclohexanecarboxamide