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3-({[(2-aminopyrimidin-5-yl)methyl](methyl)amino}methyl)-3-hydroxy-1-(3-phenylpropyl)piperidin-2-one
N-[(5-ethyl-1,2,4-oxadiazol-3-yl)methyl]-N-methyl-1-(pyridine-2-carbonyl)piperidin-4-amine
N-[(3-chlorophenyl)methyl]-3-[1-(pyridine-3-carbonyl)piperidin-4-yl]propanamide
1-(4-fluorophenyl)-4-{[6-(piperidine-1-carbonyl)imidazo[2,1-b][1,3]thiazol-5-yl]methyl}-1,4-diazepane
5-[(2-hydroxy-5-methylphenyl)methyl]-N-phenyl-4H,5H,6H,7H,8H-pyrazolo[1,5-a][1,4]diazepine-2-carboxamide
(2S)-2-({2-methyl-5-phenylpyrazolo[1,5-a]pyrimidin-7-yl}amino)-4-(methylsulfanyl)butan-1-ol
2-(3-{[(1,4-dioxan-2-ylmethyl)(methyl)amino]methyl}phenoxy)acetamide
ethyl({[5-(oxan-2-yl)furan-2-yl]methyl})[(5-propyl-1,2,4-oxadiazol-3-yl)methyl]amine
[3-(3,5-dimethyl-1H-pyrazol-4-yl)propyl](methyl)[(2E)-2-methylbut-2-en-1-yl]amine
6-[3-(1-phenylpropyl)-1H,4H,5H,6H,7H-pyrazolo[4,3-c]pyridin-5-yl]-9H-purine
1-(2,6-dimethylpyridin-4-yl)-4-{2-methylimidazo[1,2-a]pyrimidine-3-carbonyl}piperazine
1-[(5-methyl-1,3,4-oxadiazol-2-yl)methyl]-3-{4-methyl-5-[(2-methyl-1H-imidazol-1-yl)methyl]-4H-1,2,4-triazol-3-yl}piperidine
6-(2,3-dihydro-1-benzofuran-5-ylmethyl)-N-(2-methyl-1,3-benzothiazol-5-yl)-6-azaspiro[2.5]octane-1-carboxamide
ethyl 1-(but-2-ynoyl)-4-[(4-chlorophenyl)methyl]piperidine-4-carboxylate
3-(2-amino-1,3-thiazol-4-yl)-N-(3-hydroxy-3-phenylpropyl)-N-methylpropanamide
2-[4-(1,3-benzothiazol-2-ylmethyl)-1,4-diazepan-1-yl]-6-ethoxy-4-methylquinazoline
5-hydroxy-N-methyl-N-{[4-(1H-pyrazol-1-yl)phenyl]methyl}pyrazine-2-carboxamide
5-[(4-methyl-1H-pyrazol-1-yl)methyl]-3-(thiophen-2-ylmethyl)-1-(2,2,2-trifluoroethyl)-1H-1,2,4-triazole
2,5-dioxo-6-{2-[3-(trifluoromethyl)phenyl]ethyl}-1,2,5,6-tetrahydro-1,6-naphthyridine-3-carbonitrile
(2S,4S)-N-ethyl-1-(3-methylbut-2-en-1-yl)-4-[2-(4-methylphenoxy)acetamido]pyrrolidine-2-carboxamide
2-methyl-8-(1-methyl-3-propyl-1H-pyrazole-5-carbonyl)-octahydro-1H-pyrazino[1,2-a]piperazine-1,4-dione
5-[(1R,5R)-6-(3-methylbut-2-en-1-yl)-3,6-diazabicyclo[3.2.2]nonane-3-carbonyl]-1H-1,3-benzodiazole
4-{[2-chloro-5-methoxy-4-(propan-2-yloxy)phenyl]methyl}-3-(2-hydroxyethyl)piperazin-2-one
(1S,5R)-3-{[5-(2-methylpropyl)-1,2,4-oxadiazol-3-yl]methyl}-6-(1,3-thiazol-4-ylmethyl)-3,6-diazabicyclo[3.2.2]nonan-7-one
methyl 5-[(2R,3R,6R)-3-(2,3-difluorophenyl)-1,5-diazatricyclo[5.2.2.02,6]undecan-5-yl]pentanoate
1-[4-({1-ethyl-3-[(1-methylpiperidin-4-yl)methyl]-1H-1,2,4-triazol-5-yl}methyl)thiophen-2-yl]ethan-1-one
3-(4-methyl-1,3-thiazol-5-yl)-1-[2-(3-phenyl-1,2,4-oxadiazol-5-yl)pyrrolidin-1-yl]propan-1-one
1-{[2-(2-fluoro-4-methoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}-1H-1,3-benzodiazole
N-{[3-(2-fluorophenyl)-1,2-oxazol-5-yl]methyl}-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
methyl 1-[(3S,5S)-5-{[3-(methylsulfanyl)phenyl]carbamoyl}-1-[1-(2-phenylethyl)piperidin-4-yl]pyrrolidin-3-yl]-1H-1,2,3-triazole-4-carboxylate
2-(4-hydroxyphenyl)-1-[(1S,5R)-3-(oxan-4-yl)-3,6-diazabicyclo[3.2.2]nonan-6-yl]ethan-1-one
3-(dimethyl-1,2-oxazol-4-yl)-1-[2-(pyridin-2-yl)pyrrolidin-1-yl]propan-1-one
1-{[3-(2,5-dihydro-1H-pyrrole-1-carbonyl)-1H-pyrazol-5-yl]methyl}-2-methyl-1H-1,3-benzodiazole
(4aR,8aS)-6-(1-benzothiophen-2-ylmethyl)-1-(cyclohexylmethyl)-decahydro-1,6-naphthyridin-2-one
N-{imidazo[2,1-b][1,3]thiazol-6-ylmethyl}-2-methyl-5H,6H,7H,8H,9H-pyrimido[4,5-d]azepin-4-amine
1-{3-methyl-5-[2-(methylamino)pyrimidin-5-yl]-1H-1,2,4-triazol-1-yl}butan-2-ol
N-(2-methylpropyl)-2-(2-oxo-1,2-dihydropyrimidin-1-yl)-N-(thiophen-3-ylmethyl)acetamide
(1R,2R,6S,7S)-4-(2-phenylbenzoyl)-10-oxa-4-azatricyclo[5.2.1.02,6]decane
{[2-(4-fluorophenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(prop-2-en-1-yl)(prop-2-yn-1-yl)amine
5-[({[2-(2,3-dimethoxyphenyl)-5-methyl-1,3-oxazol-4-yl]methyl}(propan-2-yl)amino)methyl]pyrrolidin-2-one
2-(5-amino-1H-1,2,3,4-tetrazol-1-yl)-N-(2,1,3-benzothiadiazol-5-ylmethyl)-N-methylacetamide
2-(3-{[2-(3,4-dimethoxyphenyl)ethyl](methyl)amino}piperidin-1-yl)-2-oxoacetamide
methyl[(4-methyl-1,2,3-thiadiazol-5-yl)methyl]{[2-(naphthalen-1-yl)pyrimidin-5-yl]methyl}amine
2-(3,3-diethylpyrrolidine-1-carbonyl)-5-(methoxymethyl)-1,3,4-oxadiazole
4,5-dimethyl-6-{2-phenyl-5H,6H,7H-pyrrolo[3,4-d]pyrimidin-6-yl}-2-(trifluoromethyl)pyrimidine
1-[2-(4-fluorophenyl)morpholin-4-yl]-4-(1H-1,2,3,4-tetrazol-1-yl)butan-1-one
1-(2-methoxyphenyl)-3-{1-[1-(2-oxopropanoyl)piperidin-4-yl]-1H-pyrazol-5-yl}urea
1-[4-methyl-3-(2-oxoimidazolidin-1-yl)benzoyl]pyrrolidine-2-carboxylic acid
N-[2-(3-phenylpiperidin-1-yl)ethyl]-4,5,6,7-tetrahydro-1H-indazole-3-carboxamide
1-{1-[(3,5-dimethyl-1-benzofuran-2-yl)methyl]piperidin-4-yl}pyrrolidin-2-one